High-throughput mechanistic screening of non-equilibrium inhibitors by a fully automated data analysis pipeline in early drug-discovery
Srinivasan, Bharath, Flórez Weidinger, Juan Daniel, Zhai, Xiang, Lemercier, Guillaume, Ikeda, Timothy, Brewer, Mark, Zhang, Bairu, Heyse, Stephan, Wingfield, Jonathan, Steigele, Stephan
Published in SLAS discovery (01.12.2022)
Published in SLAS discovery (01.12.2022)
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Journal Article
Identification and Characterization of Novel Small Molecules as Potent Inhibitors of the Plasmodial Calcium-Dependent Protein Kinase 1
Lemercier, Guillaume, Fernandez-Montalvan, Amaury, Shaw, Jeffrey P, Kugelstadt, Dominik, Bomke, Joerg, Domostoj, Mathias, Schwarz, Matthias K, Scheer, Alexander, Kappes, Barbara, Leroy, Didier
Published in Biochemistry (Easton) (14.07.2009)
Published in Biochemistry (Easton) (14.07.2009)
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Journal Article
A Pyrophosphatase Regulating Polyphosphate Metabolism in Acidocalcisomes Is Essential for Trypanosoma brucei Virulence in Mice
Lemercier, Guillaume, Espiau, Benoit, Ruiz, Felix A, Vieira, Mauricio, Luo, Shuhong, Baltz, Theo, Docampo, Roberto, Bakalara, Norbert
Published in The Journal of biological chemistry (30.01.2004)
Published in The Journal of biological chemistry (30.01.2004)
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Journal Article
A Vacuolar-type H+-Pyrophosphatase Governs Maintenance of Functional Acidocalcisomes and Growth of the Insect and Mammalian Forms of Trypanosoma brucei
Lemercier, Guillaume, Dutoya, Sandrine, Luo, Shuhong, Ruiz, Felix A., Rodrigues, Claudia O., Baltz, Théo, Docampo, Roberto, Bakalara, Norbert
Published in The Journal of biological chemistry (04.10.2002)
Published in The Journal of biological chemistry (04.10.2002)
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Journal Article
A Novel C-terminal Kinesin Is Essential for Maintaining Functional Acidocalcisomes in Trypanosoma brucei
Dutoya, Sandrine, Gibert, Stephanie, Lemercier, Guillaume, Santarelli, Xavier, Baltz, Dominique, Baltz, Theo, Bakalara, Norbert
Published in The Journal of biological chemistry (28.12.2001)
Published in The Journal of biological chemistry (28.12.2001)
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Journal Article
Multifaceted C-X-C Chemokine Receptor 4 (CXCR4) Inhibition Interferes with Anti–Vascular Endothelial Growth Factor Therapy–Induced Glioma Dissemination
Gagner, Jean-Pierre, Sarfraz, Yasmeen, Ortenzi, Valerio, Alotaibi, Fawaz M., Chiriboga, Luis A., Tayyib, Awab T., Douglas, Garry J., Chevalier, Eric, Romagnoli, Barbara, Tuffin, Gérald, Schmitt, Michel, Lemercier, Guillaume, Dembowsky, Klaus, Zagzag, David
Published in The American journal of pathology (01.09.2017)
Published in The American journal of pathology (01.09.2017)
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Journal Article
Inducing and Sensing Protein-Protein Interactions in Living Cells by Selective Cross-linking
Lemercier, Guillaume, Gendreizig, Susanne, Kindermann, Maik, Johnsson, Kai
Published in Angewandte Chemie (04.06.2007)
Published in Angewandte Chemie (04.06.2007)
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Journal Article
Trypanosomatid flagellum biogenesis: ARL-3A is involved in several species
Sahin, Annelise, Lemercier, Guillaume, Tetaud, Emmanuel, Espiau, Benoît, Myler, Peter, Stuart, Kenneth, Bakalara, Norbert, Merlin, Gilles
Published in Experimental parasitology (01.11.2004)
Published in Experimental parasitology (01.11.2004)
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Journal Article
Monitor – biology
Gerlai, Robert, Hains, Bryan C, Barnes, Matt J, Miller, David J, Davies, William, Misteli, Tom, Sarker, Dipak K, Perretti, Mauro, Spitzer, Eric D, Lenz, Laurel L, Bakalara, Norbert, Lemercier, Guillaume, Insall, Robert H
Published in Drug discovery today (2004)
Published in Drug discovery today (2004)
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Journal Article
TEMPLATE-FIXED PEPTIDOMIMETICS AS INHIBITORS OF FPR1
CHEVALIER, ERIC, JUNG, FRANCOISE, OBRECHT, DANIEL, ZIMMERMANN, JOHANN, LEMERCIER, GUILLAUME, LOWE, RALF
Year of Publication 24.03.2020
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Year of Publication 24.03.2020
Patent
Template -fixed peptidomimetics as inhibitors of FPR1
JUNG, Francoise, LEMERCIER, Guillaume, LOWE, Ralf, ZIMMERMANN, Johann, OBRECHT, Daniel, CHEVALIER, Eric
Year of Publication 02.05.2019
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Year of Publication 02.05.2019
Patent
Inducing and Sensing Protein–Protein Interactions in Living Cells by Selective Cross‐linking
Lemercier, Guillaume, Gendreizig, Susanne, Kindermann, Maik, Johnsson, Kai
Published in Angewandte Chemie (04.06.2007)
Published in Angewandte Chemie (04.06.2007)
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Journal Article
Template-fixed peptidomimetics as inhibitors of FPR1
Lemercier, Guillaume, Löwe, Ralf, Zimmermann, Johann, Chevalier, Eric, Obrecht, Daniel, Jung, Françoise
Year of Publication 01.05.2018
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Year of Publication 01.05.2018
Patent
Template -fixed peptidomimetics as inhibitors of FPR1
JUNG, Francoise, LEMERCIER, Guillaume, LOWE, Ralf, ZIMMERMANN, Johann, OBRECHT, Daniel, CHEVALIER, Eric
Year of Publication 06.07.2017
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Year of Publication 06.07.2017
Patent
Peptidomiméticos fijados sobre plantilla como inhibidores del FPR1
JUNG, Françoise, LEMERCIER, Guillaume, LÖWE, Ralf, ZIMMERMANN, Johann, OBRECHT, Daniel, CHEVALIER, Eric
Year of Publication 29.05.2017
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Year of Publication 29.05.2017
Patent