Recent Advances in the Discovery of HIF-1α-p300/CBP Inhibitors as Anti-Cancer Agents
Wei, Jinlian, Yang, Yingrui, Lu, Mengchen, Lei, Yonghua, Xu, Lili, Jiang, Zhengyu, Xu, Xiaoli, Guo, Xiaoke, Zhang, Xiaojin, Sun, Haopeng, You, Qidong
Published in Mini reviews in medicinal chemistry (01.01.2018)
Published in Mini reviews in medicinal chemistry (01.01.2018)
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Microwave-assisted transition-metal-free intramolecular Ullmann-type O-arylation in water for the synthesis of xanthones and azaxanthones
Zhang, Xiaojin, Yang, Li, Wu, Yue, Du, Jianyao, Mao, Yingle, Wang, Xiao, Luan, Shijie, Lei, Yonghua, Li, Xiang, Sun, Haopeng, You, Qidong
Published in Tetrahedron letters (27.08.2014)
Published in Tetrahedron letters (27.08.2014)
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Discovery of Clinical Candidate (5-(3-(4-Chlorophenoxy)prop-1-yn-1-yl)-3-hydroxypicolinoyl)glycine, an Orally Bioavailable Prolyl Hydroxylase Inhibitor for the Treatment of Anemia
Zhang, Xiaojin, Lei, Yonghua, Hu, Tianhan, Wu, Yue, Li, Zhihong, Jiang, Zhensheng, Yang, Changyong, Zhang, Lianshan, You, Qidong
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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CDK2 and CDK4 targeted liensinine inhibits the growth of bladder cancer T24 cells
Jiang, Hanbing, Zhu, Siying, Wu, Bin, Su, Yinyin, Wang, Qiming, Lei, Yonghua, Shao, Qiuju, Gao, Yun, Gao, Ke, Wu, Guojun
Published in Chemico-biological interactions (01.09.2023)
Published in Chemico-biological interactions (01.09.2023)
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Journal Article
miR‑130b regulates PTEN to activate the PI3K/Akt signaling pathway and attenuate oxidative stress‑induced injury in diabetic encephalopathy
Lei, Yonghua, Yang, Ming, Li, Hong, Xu, Rongjuan, Liu, Junbao
Published in International journal of molecular medicine (01.07.2021)
Published in International journal of molecular medicine (01.07.2021)
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Prognostic values of preoperative neutrophil-to-lymphocyte ratio, platelet-to-lymphocyte ratio and lymphocyte- to-monocyte ratio for patients with muscle- invasive bladder cancer undergoing radical cystectomy
Lei, Yonghua, Jiao, Dian, Yao, Zhen, Wang, Lei, Zhao, Zhiguang
Published in Archivos españoles de urología (01.04.2022)
Published in Archivos españoles de urología (01.04.2022)
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Differences of temporomandibular joint symmetry in patients with unilateral complete cleft lip and palate at different developmental stages
Jia, Wanping, Yang, Zhaoxia, Su, Xinying, Shao, Mengying, Lei, Yonghua
Published in Zhong nan da xue xue bao. Journal of Central South University. Yi xue ban (28.04.2023)
Published in Zhong nan da xue xue bao. Journal of Central South University. Yi xue ban (28.04.2023)
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Association of finasteride with prostate cancer: A systematic review and meta-analysis
Wang, Lei, Lei, Yonghua, Gao, Yanyao, Cui, Dong, Tang, Qisheng, Li, Ruixiao, Wang, Dong, Chen, Yu, Zhang, Bo, Wang, He
Published in Medicine (Baltimore) (01.04.2020)
Published in Medicine (Baltimore) (01.04.2020)
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2-Substituted 3-methylnaphtho[1,2-b]furan-4,5-diones as novel L-shaped ortho-quinone substrates for NAD(P)H:quinone oxidoreductase (NQO1)
Bian, Jinlei, Deng, Bang, Xu, Lili, Xu, Xiaoli, Wang, Nan, Hu, Tianhan, Yao, Zeyu, Du, Jianyao, Yang, Li, Lei, Yonghua, Li, Xiang, Sun, Haopeng, Zhang, Xiaojin, You, Qidong
Published in European journal of medicinal chemistry (23.07.2014)
Published in European journal of medicinal chemistry (23.07.2014)
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Microwave-assisted copper- and palladium-catalyzed sonogashira-type coupling of aryl bromides and iodides with trimethylsilylacetylene
Lei, Yonghua, Hu, Tianhan, Wu, Xingsen, Wu, Yue, Xiang, Hua, Sun, Haopeng, You, Qidong, Zhang, Xiaojin
Published in Tetrahedron letters (09.03.2016)
Published in Tetrahedron letters (09.03.2016)
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A squamous odontogenic tumor following an orthodontic micro-screw: A rare case report and review of the literature
Tu, Jingqiu, Yin, Ping, Yuan, Yunyi, Chen, Jie, Yuan, Yongxiang, Lei, Yonghua
Published in Oral oncology (01.02.2018)
Published in Oral oncology (01.02.2018)
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Novel 5-carboxy-8-HQ based histone demethylase JMJD2A inhibitors: Introduction of an additional carboxyl group at the C-2 position of quinoline
Feng, Taotao, Li, Dongdong, Wang, Hai, Zhuang, Jian, Liu, Fang, Bao, Qichao, Lei, Yonghua, Chen, Weilin, Zhang, Xiaojin, Xu, Xiaoli, Sun, Haopeng, You, Qidong, Guo, Xiaoke
Published in European journal of medicinal chemistry (13.11.2015)
Published in European journal of medicinal chemistry (13.11.2015)
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Journal Article
Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 Inhibitors
Lei, Yonghua, Hu, Tianhan, Wu, Xingsen, Wu, Yue, Bao, Qichao, Zhang, Lianshan, Xia, Hua, Sun, Haopeng, You, Qidong, Zhang, Xiaojin
Published in ACS medicinal chemistry letters (10.12.2015)
Published in ACS medicinal chemistry letters (10.12.2015)
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Journal Article
An improved and scalable synthesis of N-(5-(4-cyanophenyl)-3-hydroxypicolinoyl)glycine, a promising PHD2 inhibitor for the treatment of anemia
Lei, Yonghua, Hu, Tianhan, Hu, Mingyang, Yang, Li, Wu, Yue, Xiang, Hua, Zhang, Lianshan, Shen, Lingjia, You, Qidong, Zhang, Xiaojin
Published in Tetrahedron letters (26.08.2015)
Published in Tetrahedron letters (26.08.2015)
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Journal Article
Small-molecule inhibitors of HIF-PHD2: a valid strategy to renal anemia treatment in clinical therapy
Wu, Yue, Wang, Nan, Lei, Yonghua, Hu, Tianhan, You, Qidong, Zhang, Xiaojin
Published in MedChemComm (01.01.2016)
Published in MedChemComm (01.01.2016)
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Small-molecule inhibitors of HIF-PHD2: a valid strategy to renal anemia treatment in clinical therapyThe authors declare no competing interests
Wu, Yue, Wang, Nan, Lei, Yonghua, Hu, Tianhan, You, Qidong, Zhang, Xiaojin
Year of Publication 12.07.2016
Year of Publication 12.07.2016
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Identification of novel JMJD2A inhibitor scaffold using shape and electrostatic similarity search combined with docking method and MM-GBSA approach
Feng, Taotao, Chen, Weilin, Li, Dongdong, Lin, Hongzhi, Liu, Fang, Bao, Qichao, Lei, Yonghua, Zhang, Xiaojin, Xu, Xiaoli, Guo, Xiaoke, You, Qidong, Sun, Haopeng
Published in RSC advances (01.01.2015)
Published in RSC advances (01.01.2015)
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Three-dimensional analysis for changes in dentigerous cyst-associated maxillary canines after marsupialization in adolescents
Yuan, Yunyi, Tu, Jingqiu, Fan, Jiaqian, Lei, Yonghua
Published in Zhong nan da xue xue bao. Journal of Central South University. Yi xue ban (28.02.2019)
Published in Zhong nan da xue xue bao. Journal of Central South University. Yi xue ban (28.02.2019)
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