In vitro and In vivo Activity of Novel Small-Molecule Inhibitors Targeting the Pleckstrin Homology Domain of Protein Kinase B/AKT
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An Inhibitor of the Pleckstrin Homology Domain of CNK1 Selectively Blocks the Growth of Mutant KRAS Cells and Tumors
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Novel inhibitors induce large conformational changes of GAB1 pleckstrin homology domain and kill breast cancer cells
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Molecular pharmacology and antitumor activity of PHT-427, a novel Akt/phosphatidylinositide-dependent protein kinase 1 pleckstrin homology domain inhibitor
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Recent development of anticancer therapeutics targeting Akt
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Published in Alzheimer's & dementia (01.12.2023)
Published in Alzheimer's & dementia (01.12.2023)
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Correction: An Inhibitor of the Pleckstrin Homology Domain of CNK1 Selectively Blocks the Growth of Mutant KRAS Cells and Tumors
Indarte, Martin, Puentes, Roisin, Maruggi, Marco, Ihle, Nathan T, Grandjean, Geoffrey, Scott, Michael, Ahmed, Zamal, Meuillet, Emmanuelle J, Zhang, Shuxing, Lemos, Jr, Robert, Du-Cuny, Lei, Layng, Fabiana I A L, Correa, Ricardo G, Bankston, Laurie A, Liddington, Robert C, Kirkpatrick, Lynn, Powis, Garth
Published in Cancer research (Chicago, Ill.) (15.10.2019)
Published in Cancer research (Chicago, Ill.) (15.10.2019)
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Computational aqueous solubility prediction for drug-like compounds in congeneric series
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Published in European journal of medicinal chemistry (01.03.2008)
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Abstract 2166: In silico identification and biological evaluation of potent small molecule inhibitors targeting GAB1 pleckstrin homology domain
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Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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Novel Inhibitors Induce Large Conformational Changes of GAB1 Pleckstrin Homology Domain and Kill Breast Cancer Cells: e1004021
Chen, Lu, Du-Cuny, Lei, Moses, Sylvestor, Dumas, Sabrina, Song, Zuohe, Rezaeian, Abdol Hossein, Lin, Hui-Kuan, Meuillet, Emmanuelle J, Zhang, Shuxing
Published in PLoS computational biology (01.01.2015)
Published in PLoS computational biology (01.01.2015)
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Development of sulfonamide AKT PH domain inhibitors
Ahad, Ali Md, Zuohe, Song, Du-Cuny, Lei, Moses, Sylvestor A., Zhou, Li Li, Zhang, Shuxing, Powis, Garth, Meuillet, Emmanuelle J., Mash, Eugene A.
Published in Bioorganic & medicinal chemistry (15.03.2011)
Published in Bioorganic & medicinal chemistry (15.03.2011)
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