An efficient site-selective, dual bioconjugation approach exploiting N-terminal cysteines as minimalistic handles to engineer tailored anti-HER2 affibody conjugates
Novak, Ana, Kersaudy, Florian, Berger, Sylvie, Morisset-Lopez, Séverine, Lefoulon, François, Pifferi, Carlo, Aucagne, Vincent
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
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Active targeting with particulate drug carriers in tumor therapy: fundamentals and recent progress
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Book Review
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Exploiting the Biocatalytic Toolbox for the Asymmetric Synthesis of the Heart‐Rate Reducing Agent Ivabradine
Pedragosa‐Moreau, Sandrine, Le Flohic, Alexandre, Thienpondt, Vivien, Lefoulon, François, Petit, Anne‐Marie, Ríos‐Lombardía, Nicolás, Morís, Francisco, González‐Sabín, Javier
Published in Advanced synthesis & catalysis (02.02.2017)
Published in Advanced synthesis & catalysis (02.02.2017)
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Drug solubilization and in vitro toxicity evaluation of lipoamino acid surfactants
Ménard, Nathalie, Tsapis, Nicolas, Poirier, Cécile, Arnauld, Thomas, Moine, Laurence, Lefoulon, François, Péan, Jean-Manuel, Fattal, Elias
Published in International journal of pharmaceutics (28.02.2012)
Published in International journal of pharmaceutics (28.02.2012)
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Extending the Structural Diversity of α-Flavonoid Glycosides with Engineered Glucansucrases
Malbert, Yannick, Pizzut-Serin, Sandra, Massou, Stéphane, Cambon, Emmanuelle, Laguerre, Sandrine, Monsan, Pierre, Lefoulon, François, Morel, Sandrine, André, Isabelle, Remaud-Simeon, Magali
Published in ChemCatChem (01.08.2014)
Published in ChemCatChem (01.08.2014)
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Anti-Cancer Stem-like Cell Compounds in Clinical Development - An Overview and Critical Appraisal
Marcucci, Fabrizio, Rumio, Cristiano, Lefoulon, François
Published in Frontiers in oncology (10.05.2016)
Published in Frontiers in oncology (10.05.2016)
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Journal Article
Original Design of Fluorescent Ligands by Fusing BODIPY and Melatonin Neurohormone
Thireau, Jérémy, Marteaux, Justine, Delagrange, Philippe, Lefoulon, Francois, Dufourny, Laurence, Guillaumet, Gérald, Suzenet, Franck
Published in ACS medicinal chemistry letters (13.02.2014)
Published in ACS medicinal chemistry letters (13.02.2014)
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Journal Article
Pyridine to aniline: An exceptional biologically driven rearrangement
Arnauld, Thomas, Beaumal, Jean-Yves, Lefoulon, François, Petit, Alain, Renaud, Tristan
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
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Journal Article
Branching pattern of gluco-oligosaccharides and 1.5 kDa dextran grafted by the α-1,2 branching sucrase GBD-CD2
BRISON, Yoann, LAGUERRE, Sandrine, LEFOULON, François, MOREL, Sandrine, MONTIES, Nelly, POTOCKI-VERONESE, Gabrielle, MONSAN, Pierre, REMAUD-SIMEON, Magali
Published in Carbohydrate polymers (15.04.2013)
Published in Carbohydrate polymers (15.04.2013)
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Journal Article
Novel Surfactants with Diglutamic Acid Polar Head Group: Drug Solubilization and Toxicity Studies
Ménard, Nathalie, Tsapis, Nicolas, Poirier, Cécile, Arnauld, Thomas, Moine, Laurence, Gignoux, Claire, Lefoulon, François, Péan, Jean-Manuel, Fattal, Elias
Published in Pharmaceutical research (01.07.2012)
Published in Pharmaceutical research (01.07.2012)
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Journal Article
Physicochemical characterization and toxicity evaluation of steroid-based surfactants designed for solubilization of poorly soluble drugs
Ménard, Nathalie, Tsapis, Nicolas, Poirier, Cécile, Arnauld, Thomas, Moine, Laurence, Lefoulon, François, Péan, Jean-Manuel, Fattal, Elias
Published in European journal of pharmaceutical sciences (18.12.2011)
Published in European journal of pharmaceutical sciences (18.12.2011)
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Journal Article
A convenient microwave-assisted 5-amination of flavones
Lecoutey, Cédric, Fossey, Christine, Demuynck, Luc, Lefoulon, François, Fabis, Frédéric, Rault, Sylvain
Published in Tetrahedron (01.12.2008)
Published in Tetrahedron (01.12.2008)
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Journal Article
Molecular pharmacology of the ovine melatonin receptor: comparison with recombinant human MT1 and MT2 receptors
MAILLIET, Francois, AUDINOT, Valérie, RENARD, Pierre, BOUTIN, Jean A, MALPAUX, Benoit, BONNAUD, Anne, DELAGRANGE, Philippe, MIGAUD, Martine, BARRETT, Perry, VIAUD-MASSUARD, Marie-Claude, LESIEUR, Daniel, LEFOULON, Francois
Published in Biochemical pharmacology (15.02.2004)
Published in Biochemical pharmacology (15.02.2004)
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Journal Article
New radioligands for describing the molecular pharmacology of MT1 and MT2 melatonin receptors
Legros, Céline, Matthey, Ulrich, Grelak, Teresa, Pedragona-Moreau, Sandrine, Hassler, Werner, Yous, Saïd, Thomas, Emmanuel, Suzenet, Franck, Folleas, Benoît, Lefoulon, François, Berthelot, Pascal, Caignard, Daniel-Henri, Guillaumet, Gérald, Delagrange, Philippe, Brayer, Jean-Louis, Nosjean, Olivier, Boutin, Jean A
Published in International journal of molecular sciences (25.04.2013)
Published in International journal of molecular sciences (25.04.2013)
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Journal Article
Enhanced drug loading in polymerized micellar cargo
Ogier, Julien, Arnauld, Thomas, Carrot, Geraldine, Lhumeau, Antoine, Delbos, Jean-Marie, Boursier, Claire, Loreau, Olivier, Lefoulon, Francois, Doris, Eric
Published in Organic & biomolecular chemistry (07.09.2010)
Published in Organic & biomolecular chemistry (07.09.2010)
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