Proton stoichiometry associated with human neutrophil respiratory-burst reactions
Gabig, T G, Lefker, B A, Ossanna, P J, Weiss, S J
Published in The Journal of biological chemistry (10.11.1984)
Published in The Journal of biological chemistry (10.11.1984)
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Journal Article
Origin of Stereochemistry in Simple Pyrrolidinone Enolate Alkylations
Meyers, A. I, Seefeld, Mark A, Lefker, Bruce A, Blake, James F
Published in Journal of the American Chemical Society (14.05.1997)
Published in Journal of the American Chemical Society (14.05.1997)
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Journal Article
Discovery of inhibitors of human renin with high oral bioavailability
Hoover, D J, Lefker, B A, Rosati, R L, Wester, R T, Kleinman, E F, Bindra, J S, Holt, W F, Murphy, W R, Mangiapane, M L, Hockel, G M
Published in Advances in experimental medicine and biology (1995)
Published in Advances in experimental medicine and biology (1995)
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Journal Article
An efficient synthesis of enantiomerically enriched aryllactic esters
Lefker, Bruce A., Hada, William A., McGarry, Patrick J.
Published in Tetrahedron letters (18.07.1994)
Published in Tetrahedron letters (18.07.1994)
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Journal Article
An asymmetric synthesis of chiral 4,4-disubstituted cyclohexenones in high enantiomeric purity
Meyers, A. I, Lefker, Bruce A, Wanner, Klaus T, Aitken, R. Alan
Published in Journal of organic chemistry (01.05.1986)
Published in Journal of organic chemistry (01.05.1986)
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Journal Article
Tetrahydroisoquinolines as subtype selective estrogen agonists/antagonists
Chesworth, Richard, Zawistoski, Michael P., Lefker, Bruce A., Cameron, Kimberly O., Day, Robert F., Mangano, F.Michael, Rosati, Robert L., Colella, Stacy, Petersen, Donna N., Brault, Amy, Lu, Bihong, Pan, Lydia C., Perry, Pia, Ng, Oicheng, Castleberry, Tessa A., Owen, Thomas A., Brown, Thomas A., Thompson, David D., DaSilva-Jardine, Paul
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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Journal Article
Stereoselective Alkylations in Rigid Systems. Effect of Remote Substituents on π-Facial Additions to Lactam Enolates. Stereoelectronic and Steric Effects
Meyers, A. I, Seefeld, Mark A, Lefker, Bruce A, Blake, James F, Williard, Paul G
Published in Journal of the American Chemical Society (05.08.1998)
Published in Journal of the American Chemical Society (05.08.1998)
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Journal Article
Discovery of highly selective EP4 receptor agonists that stimulate new bone formation and restore bone mass in ovariectomized rats
Cameron, Kimberly O., Lefker, Bruce A., Chu-Moyer, Margaret Y., Crawford, David T., Jardine, Paul DaSilva, DeNinno, Shari L., Gilbert, Sandra, Grasser, William A., Ke, HuaZhu, Lu, Bihong, Owen, Thomas A., Paralkar, Vishwas M., Qi, Hong, Scott, Dennis O., Thompson, David D., Tjoa, Christina M., Zawistoski, Michael P.
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Journal Article
Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs): Discovery of capromorelin
Carpino, Philip A, Lefker, Bruce A, Toler, Steven M, Pan, Lydia C, Hadcock, John R, Cook, Ewell R, DiBrino, Joseph N, Campeta, Anthony M, DeNinno, Shari L, Chidsey-Frink, Kristin L, Hada, William A, Inthavongsay, John, Mangano, F.Michael, Mullins, Michelle A, Nickerson, David F, Ng, Oicheng, Pirie, Christine M, Ragan, John A, Rose, Colin R, Tess, David A, Wright, Ann S, Yu, Li, Zawistoski, Michael P, DaSilva-Jardine, Paul A, Wilson, Theresa C, Thompson, David D
Published in Bioorganic & medicinal chemistry (20.02.2003)
Published in Bioorganic & medicinal chemistry (20.02.2003)
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Journal Article
Preclinical pharmacology of CP-424,391, an orally active pyrazolinone-piperidine [correction of pyrazolidinone-piperidine] growth hormone secretagogue
Pan, L C, Carpino, P A, Lefker, B A, Ragan, J A, Toler, S M, Pettersen, J C, Nettleton, D O, Ng, O, Pirie, C M, Chidsey-Frink, K, Lu, B, Nickerson, D F, Tess, D A, Mullins, M A, MacLean, D B, DaSilva-Jardine, P A, Thompson, D D
Published in Endocrine (01.02.2001)
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Published in Endocrine (01.02.2001)
Journal Article
A Nonprostanoid EP4 Receptor Selective Prostaglandin E sub(2) Agonist Restores Bone Mass and Strength in Aged, Ovariectomized Rats
Ke, H Z, Crawford, D T, Qi, H, Simmons, HA, Owen, T A, Paralkar, V M, Li, M, Lu, B, Grasser, WA, Cameron, KO, Lefker, BA, DaSilva-Jardine, P, Scott, DO, Zhang, Q
Published in Journal of bone and mineral research (01.04.2006)
Published in Journal of bone and mineral research (01.04.2006)
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Journal Article
A Novel, Non-Prostanoid EP2 Receptor-Selective Prostaglandin E sub(2) Agonist Stimulates Local Bone Formation and Enhances Fracture Healing
Li, M, Ke, H Z, Qi, H, Healy, DR, Li, Y, Crawford, D T, Paralkar, V M, Owen, T A, Cameron, KO, Lefker, BA, Brown, T A, Thompson, D D
Published in Journal of bone and mineral research (01.11.2003)
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Published in Journal of bone and mineral research (01.11.2003)
Journal Article
Discovery and biological characterization of capromorelin analogues with extended half-lives
Carpino, Philip A., Lefker, Bruce A., Toler, Steven M., Pan, Lydia C., Hadcock, John R., Murray, Marianne C., Cook, Ewell R., DiBrino, Joseph N., DeNinno, Shari L., Chidsey-Frink, Kristin L., Hada, William A., Inthavongsay, John, Lewis, Sharon K., Mangano, F.Michael, Mullins, Michelle A., Nickerson, David F., Ng, Oicheng, Pirie, Christine M., Ragan, John A., Rose, Colin R., Tess, David A., Wright, Ann S., Yu, Li, Zawistoski, Michael P., Pettersen, John C., DaSilva-Jardine, Paul A., Wilson, Theresa C., Thompson, David D.
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
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Journal Article
A simple method for the formation of cyclopropylamines: the first synthesis of tricyclopropylamine
Gillaspy, Melissa L., Lefker, Bruce A., Hada, William A, Hoover, Dennis J.
Published in Tetrahedron letters (09.10.1995)
Published in Tetrahedron letters (09.10.1995)
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Journal Article