A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons
Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša
Published in Angewandte Chemie International Edition (11.10.2021)
Published in Angewandte Chemie International Edition (11.10.2021)
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Frontispiece: A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons
Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša
Published in Angewandte Chemie International Edition (11.10.2021)
Published in Angewandte Chemie International Edition (11.10.2021)
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Identification and Characterization of Inhibitors of Multidrug Resistance Efflux Pumps in Pseudomonas aeruginosa: Novel Agents for Combination Therapy
LOMOVSKAYA, Olga, WARREN, Mark S, LEGER, Roger, HECKER, Scott, WATKINS, Will, HOSHINO, Kazuki, ISHIDA, Hiroko, LEE, Ving J, LEE, Angela, GALAZZO, Jorge, FRONKO, Richard, MAY LEE, BLAIS, Johanne, CHO, Deidre, CHAMBERLAND, Suzanne, RENAU, Tom
Published in Antimicrobial Agents and Chemotherapy (01.01.2001)
Published in Antimicrobial Agents and Chemotherapy (01.01.2001)
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Mcl-1 antagonism is a potential therapeutic strategy in a subset of solid cancers
Modugno, Michele, Banfi, Patrizia, Gasparri, Fabio, Borzilleri, Robert, Carter, Percy, Cornelius, Lyndon, Gottardis, Marco, Lee, Ving, Mapelli, Claudio, Naglich, Joseph G., Tebben, Andrew, Vite, Gregory, Pastori, Wilma, Albanese, Clara, Corti, Emiliana, Ballinari, Dario, Galvani, Arturo
Published in Experimental cell research (15.03.2015)
Published in Experimental cell research (15.03.2015)
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MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: Highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate
Yoshida, Ken-ichi, Nakayama, Kiyoshi, Ohtsuka, Masami, Kuru, Noriko, Yokomizo, Yoshihiro, Sakamoto, Atsunobu, Takemura, Makoto, Hoshino, Kazuki, Kanda, Hiroko, Nitanai, Hironobu, Namba, Kenji, Yoshida, Kumi, Imamura, Yuichiro, Zhang, Jason Z., Lee, Ving J., Watkins, William J.
Published in Bioorganic & medicinal chemistry (15.11.2007)
Published in Bioorganic & medicinal chemistry (15.11.2007)
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Frontispiz: A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons
Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša
Published in Angewandte Chemie (11.10.2021)
Published in Angewandte Chemie (11.10.2021)
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Journal Article
A Selection of Macrocyclic Peptides That Bind STING From an mRNA‐Display Library With Split Degenerate Codons
Lin, Chi‐Wang, Harner, Mary J., Douglas, Andrew E., Lafont, Virginie, Yu, Fei, Lee, Ving G., Poss, Michael A., Swain, Joanna F., Wright, Martin, Lipovšek, Daša
Published in Angewandte Chemie (11.10.2021)
Published in Angewandte Chemie (11.10.2021)
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Eleven Amino Acid Glucagon-like Peptide-1 Receptor Agonists with Antidiabetic Activity
Mapelli, Claudio, Natarajan, Sesha I, Meyer, Jean-Philippe, Bastos, Margarita M, Bernatowicz, Michael S, Lee, Ving G, Pluscec, Jelka, Riexinger, Douglas J, Sieber-McMaster, Ellen S, Constantine, Keith L, Smith-Monroy, Constance A, Golla, Rajasree, Ma, Zhengping, Longhi, Daniel A, Shi, Dan, Xin, Li, Taylor, Joseph R, Koplowitz, Barry, Chi, Cecilia L, Khanna, Ashish, Robinson, Gordon W, Seethala, Ramakrishna, Antal-Zimanyi, Ildiko A, Stoffel, Robert H, Han, Songping, Whaley, Jean M, Huang, Christine S, Krupinski, John, Ewing, William R
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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Use of a Genetic Approach To Evaluate the Consequences of Inhibition of Efflux Pumps in Pseudomonas aeruginosa
OLGALOMOVSKAYA, LEE, A, HOSHINO, K, ISHIDA, H, MISTRY, A, WARREN, M. S, BOYER, E, CHAMBERLAND, S, LEE, V. J
Published in Antimicrobial Agents and Chemotherapy (01.06.1999)
Published in Antimicrobial Agents and Chemotherapy (01.06.1999)
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MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 6: Exploration of aromatic substituents
Yoshida, Ken-ichi, Nakayama, Kiyoshi, Yokomizo, Yoshihiro, Ohtsuka, Masami, Takemura, Makoto, Hoshino, Kazuki, Kanda, Hiroko, Namba, Kenji, Nitanai, Hironobu, Zhang, Jason Z., Lee, Ving J., Watkins, William J.
Published in Bioorganic & medicinal chemistry (15.12.2006)
Published in Bioorganic & medicinal chemistry (15.12.2006)
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Identification of potent 11mer Glucagon-Like Peptide-1 Receptor agonist peptides with novel C-terminal amino acids: Homohomophenylalanine analogs
Haque, Tasir S., Lee, Ving G., Riexinger, Douglas, Lei, Ming, Malmstrom, Sarah, Xin, Li, Han, Songping, Mapelli, Claudio, Cooper, Christopher B., Zhang, Ge, Ewing, William R., Krupinski, John
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
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MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 5: Carbon-substituted analogues at the C-2 position
Yoshida, Ken-ichi, Nakayama, Kiyoshi, Kuru, Noriko, Kobayashi, Shozo, Ohtsuka, Masami, Takemura, Makoto, Hoshino, Kazuki, Kanda, Hiroko, Zhang, Jason Z., Lee, Ving J., Watkins, William J.
Published in Bioorganic & medicinal chemistry (15.03.2006)
Published in Bioorganic & medicinal chemistry (15.03.2006)
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MexAB-OprM-Specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 1: Discovery and early strategies for lead optimization
Nakayama, Kiyoshi, Ishida, Yohei, Ohtsuka, Masami, Kawato, Haruko, Yoshida, Ken-ichi, Yokomizo, Yoshihiro, Hosono, Shigeru, Ohta, Toshiharu, Hoshino, Kazuki, Ishida, Hiroko, Yoshida, Kumi, Renau, Thomas E., Léger, Roger, Zhang, Jason Z., Lee, Ving J., Watkins, William J.
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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An Inhibitor Binding Pocket Distinct from the Catalytic Active Site on Human β-APP Cleaving Enzyme
Kornacker, Michael G, Lai, Zhihong, Witmer, Mark, Ma, Jianghong, Hendrick, Joseph, Lee, Ving G, Riexinger, Douglas J, Mapelli, Claudio, Metzler, William, Copeland, Robert A
Published in Biochemistry (Easton) (30.08.2005)
Published in Biochemistry (Easton) (30.08.2005)
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MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 2: achieving activity in vivo through the use of alternative scaffolds
Nakayama, Kiyoshi, Ishida, Yohei, Ohtsuka, Masami, Kawato, Haruko, Yoshida, Ken-ichi, Yokomizo, Yoshihiro, Ohta, Toshiharu, Hoshino, Kazuki, Otani, Tsuyoshi, Kurosaka, Yuichi, Yoshida, Kumi, Ishida, Hiroko, Lee, Ving J., Renau, Thomas E., Watkins, William J.
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Conformationally-restricted analogues of efflux pump inhibitors that potentiate the activity of levofloxacin in Pseudomonas aeruginosa
Renau, Thomas E, Léger, Roger, Filonova, Lubov, Flamme, Eric M, Wang, Michael, Yen, Rose, Madsen, Deidre, Griffith, David, Chamberland, Suzanne, Dudley, Michael N, Lee, Ving J, Lomovskaya, Olga, Watkins, William J, Ohta, Toshiharu, Nakayama, Kiyoshi, Ishida, Yohei
Published in Bioorganic & medicinal chemistry letters (18.08.2003)
Published in Bioorganic & medicinal chemistry letters (18.08.2003)
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Exploration of structure–activity relationships at the two C-terminal residues of potent 11mer Glucagon-Like Peptide-1 receptor agonist peptides via parallel synthesis
Haque, Tasir S., Martinez, Rogelio L., Lee, Ving G., Riexinger, Douglas G., Lei, Ming, Feng, Ming, Koplowitz, Barry, Mapelli, Claudio, Cooper, Christopher B., Zhang, Ge, Huang, Christine, Ewing, William R., Krupinski, John
Published in Peptides (New York, N.Y. : 1980) (01.07.2010)
Published in Peptides (New York, N.Y. : 1980) (01.07.2010)
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Journal Article
Peptidomimetics of Efflux Pump Inhibitors Potentiate the Activity of Levofloxacin in Pseudomonas aeruginosa
Renau, Thomas E., Léger, Roger, Yen, Rose, She, Miles W., Flamme, Eric M., Sangalang, Joan, Gannon, Carla L., Chamberland, Suzanne, Lomovskaya, Olga, Lee, Ving J.
Published in Bioorganic & medicinal chemistry letters (11.03.2002)
Published in Bioorganic & medicinal chemistry letters (11.03.2002)
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MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 4: Addressing the problem of poor stability due to photoisomerization of an acrylic acid moiety
Nakayama, Kiyoshi, Kuru, Noriko, Ohtsuka, Masami, Yokomizo, Yoshihiro, Sakamoto, Atsunobu, Kawato, Haruko, Yoshida, Ken-ichi, Ohta, Toshiharu, Hoshino, Kazuki, Akimoto, Katsuya, Itoh, Junko, Ishida, Hiroko, Cho, Aesop, Palme, Monica H., Zhang, Jason Z., Lee, Ving J., Watkins, William J.
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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