Autoinhibitory regulation of S100A8/S100A9 alarmin activity locally restricts sterile inflammation
Vogl, Thomas, Stratis, Athanasios, Wixler, Viktor, Völler, Tom, Thurainayagam, Sumita, Jorch, Selina K, Zenker, Stefanie, Dreiling, Alena, Chakraborty, Deblina, Fröhling, Mareike, Paruzel, Peter, Wehmeyer, Corinna, Hermann, Sven, Papantonopoulou, Olympia, Geyer, Christiane, Loser, Karin, Schäfers, Michael, Ludwig, Stephan, Stoll, Monika, Leanderson, Tomas, Schultze, Joachim L, König, Simone, Pap, Thomas, Roth, Johannes
Published in The Journal of clinical investigation (01.05.2018)
Published in The Journal of clinical investigation (01.05.2018)
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Journal Article
CD14 Is a Co-Receptor for TLR4 in the S100A9-Induced Pro-Inflammatory Response in Monocytes
He, Zhifei, Riva, Matteo, Björk, Per, Swärd, Karl, Mörgelin, Matthias, Leanderson, Tomas, Ivars, Fredrik
Published in PloS one (26.05.2016)
Published in PloS one (26.05.2016)
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Journal Article
Identification of human S100A9 as a novel target for treatment of autoimmune disease via binding to quinoline-3-carboxamides
Björk, Per, Björk, Anders, Vogl, Thomas, Stenström, Martin, Liberg, David, Olsson, Anders, Roth, Johannes, Ivars, Fredrik, Leanderson, Tomas
Published in PLoS biology (28.04.2009)
Published in PLoS biology (28.04.2009)
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Paquinimod prevents development of diabetes in the non-obese diabetic (NOD) mouse
Tahvili, Sahar, Törngren, Marie, Holmberg, Dan, Leanderson, Tomas, Ivars, Fredrik
Published in PloS one (09.05.2018)
Published in PloS one (09.05.2018)
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Journal Article
Paquinimod reduces skin fibrosis in tight skin 1 mice, an experimental model of systemic sclerosis
Stenström, Martin, Nyhlén, Helén Carlsson, Törngren, Marie, Liberg, David, Sparre, Birgitta, Tuvesson, Helén, Eriksson, Helena, Leanderson, Tomas
Published in Journal of dermatological science (01.07.2016)
Published in Journal of dermatological science (01.07.2016)
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Journal Article
S100A9 interaction with TLR4 promotes tumor growth
Källberg, Eva, Vogl, Thomas, Liberg, David, Olsson, Anders, Björk, Per, Wikström, Pernilla, Bergh, Anders, Roth, Johannes, Ivars, Fredrik, Leanderson, Tomas
Published in PloS one (28.03.2012)
Published in PloS one (28.03.2012)
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Journal Article
Type I IFN Signaling Is Crucial for Host Resistance against Different Species of Pathogenic Bacteria
Mancuso, Giuseppe, Midiri, Angelina, Biondo, Carmelo, Beninati, Concetta, Zummo, Sebastiana, Galbo, Roberta, Tomasello, Francesco, Gambuzza, Maria, Macri, Giancarlo, Ruggeri, Alessia, Leanderson, Tomas, Teti, Giuseppe
Published in Journal of Immunology (01.03.2007)
Published in Journal of Immunology (01.03.2007)
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Journal Article
Human S100A9 protein is stabilized by inflammatory stimuli via the formation of proteolytically-resistant homodimers
Riva, Matteo, He, Zhifei, Källberg, Eva, Ivars, Fredrik, Leanderson, Tomas
Published in PloS one (23.04.2013)
Published in PloS one (23.04.2013)
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Journal Article
Myeloid-Related Protein 14 Promotes Inflammation and Injury in Meningitis
Wache, Christina, Klein, Matthias, Ostergaard, Christian, Angele, Barbara, Häcker, Hans, Pfister, Hans-Walter, Pruenster, Monika, Sperandio, Markus, Leanderson, Tomas, Roth, Johannes, Vogl, Thomas, Koedel, Uwe
Published in The Journal of infectious diseases (15.07.2015)
Published in The Journal of infectious diseases (15.07.2015)
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Journal Article
S100A9 as a Pharmacological Target Molecule in Inflammation and Cancer
Leanderson, Tomas, Liberg, David, Ivars, Fredrik
Published in Endocrine, metabolic & immune disorders drug targets (01.01.2015)
Published in Endocrine, metabolic & immune disorders drug targets (01.01.2015)
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Journal Article
Inhibition of metastasis in a castration resistant prostate cancer model by the quinoline-3-carboxamide tasquinimod (ABR-215050)
Jennbacken, Karin, Welén, Karin, Olsson, Anders, Axelsson, Bengt, Törngren, Marie, Damber, Jan-Erik, Leanderson, Tomas
Published in The Prostate (01.06.2012)
Published in The Prostate (01.06.2012)
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Journal Article
Tasquinimod modulates suppressive myeloid cells and enhances cancer immunotherapies in murine models
Shen, Li, Sundstedt, Anette, Ciesielski, Michael, Miles, Kiersten Marie, Celander, Mona, Adelaiye, Remi, Orillion, Ashley, Ciamporcero, Eric, Ramakrishnan, Swathi, Ellis, Leigh, Fenstermaker, Robert, Abrams, Scott I, Eriksson, Helena, Leanderson, Tomas, Olsson, Anders, Pili, Roberto
Published in Cancer immunology research (01.02.2015)
Published in Cancer immunology research (01.02.2015)
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Journal Article
Tasquinimod (ABR-215050), a quinoline-3-carboxamide anti-angiogenic agent, modulates the expression of thrombospondin-1 in human prostate tumors
Olsson, Anders, Björk, Anders, Vallon-Christersson, Johan, Isaacs, John T, Leanderson, Tomas
Published in Molecular cancer (17.05.2010)
Published in Molecular cancer (17.05.2010)
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Journal Article
Vesicular Location and Transport of S100A8 and S100A9 Proteins in Monocytoid Cells
Chakraborty, Paramita, Bjork, Per, Källberg, Eva, Olsson, Anders, Riva, Matteo, Mörgelin, Matthias, Liberg, David, Ivars, Fredrik, Leanderson, Tomas
Published in PloS one (14.12.2015)
Published in PloS one (14.12.2015)
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Journal Article
Common interactions between S100A4 and S100A9 defined by a novel chemical probe
Björk, Per, Källberg, Eva, Wellmar, Ulf, Riva, Matteo, Olsson, Anders, He, Zhifei, Törngren, Marie, Liberg, David, Ivars, Fredrik, Leanderson, Tomas
Published in PloS one (08.05.2013)
Published in PloS one (08.05.2013)
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Journal Article
Tasquinimod triggers an early change in the polarization of tumor associated macrophages in the tumor microenvironment
Olsson, Anders, Nakhlé, Jessica, Sundstedt, Anette, Plas, Pascale, Bauchet, Anne-Laure, Pierron, Valérie, Bruetschy, Luce, Deronic, Adnan, Törngren, Marie, Liberg, David, Schmidlin, Fabien, Leanderson, Tomas
Published in Journal for immunotherapy of cancer (15.12.2015)
Published in Journal for immunotherapy of cancer (15.12.2015)
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Journal Article
Mice lacking NCF1 exhibit reduced growth of implanted melanoma and carcinoma tumors
Kelkka, Tiina, Pizzolla, Angela, Laurila, Juha Petteri, Friman, Tomas, Gustafsson, Renata, Källberg, Eva, Olsson, Olof, Leanderson, Tomas, Rubin, Kristofer, Salmi, Marko, Jalkanen, Sirpa, Holmdahl, Rikard
Published in PloS one (16.12.2013)
Published in PloS one (16.12.2013)
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Journal Article
CD11b+Ly6C++Ly6G- cells show distinct function in mice with chronic inflammation or tumor burden
Källberg, Eva, Stenström, Martin, Liberg, David, Ivars, Fredrik, Leanderson, Tomas
Published in BMC immunology (12.12.2012)
Published in BMC immunology (12.12.2012)
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Journal Article
Identification of ABR-215050 as lead second generation quinoline-3-carboxamide anti-angiogenic agent for the treatment of prostate cancer
Isaacs, John T., Pili, Roberto, Qian, David Z., Dalrymple, Susan L., Garrison, Jason B., Kyprianou, Natasha, Björk, Anders, Olsson, Anders, Leanderson, Tomas
Published in The Prostate (01.12.2006)
Published in The Prostate (01.12.2006)
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