Chk1 inhibition and Wee1 inhibition combine synergistically to impede cellular proliferation
Davies, Kurtis D., Cable, P. LouAnn, Garrus, Jennifer E., Sullivan, Francis X., von Carlowitz, Ira, Huerou, Yvan Le, Wallace, Eli, Woessner, Richard D., Gross, Stefan
Published in Cancer biology & therapy (01.11.2011)
Published in Cancer biology & therapy (01.11.2011)
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Novel acyl coenzyme A (CoA): Diacylglycerol acyltransferase-1 inhibitors: Synthesis and biological activities of diacylethylenediamine derivatives
Nakada, Yoshihisa, Aicher, Thomas D., Huerou, Yvan Le, Turner, Timothy, Pratt, Scott A., Gonzales, Stephen S., Boyd, Steve A., Miki, Hiroshi, Yamamoto, Toshihiro, Yamaguchi, Hiroshi, Kato, Koki, Kitamura, Shuji
Published in Bioorganic & medicinal chemistry (01.04.2010)
Published in Bioorganic & medicinal chemistry (01.04.2010)
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Journal Article
Abstract 2939: Chk1 inhibition and Wee1 inhibition combine synergistically to inhibit cellular proliferation
Davies, Kurtis D., Sullivan, Francis, von Carlowitz, Ira, Huerou, Yvan Le, Wallace, Eli, Woessner, Richard D., Gross, Stefan
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Single-agent inhibition of Chk1 is antiproliferative in human cancer cell lines in vitro and inhibits tumor xenograft growth in vivo
Davies, Kurtis D, Humphries, Michael J, Sullivan, Francis X, von Carlowitz, Ira, Le Huerou, Yvan, Mohr, Peter J, Wang, Bin, Blake, James F, Lyon, Michael A, Gunawardana, Indrani, Chicarelli, Mark, Wallace, Eli, Gross, Stefan
Published in Oncology research (01.01.2011)
Published in Oncology research (01.01.2011)
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Abstract 3874: Single-agent Chk1 inhibition is anti-proliferative in leukemia cells in vitro and in vivo
Davies, Kurtis D., Humphries, Michael J., Sullivan, Francis, von Carlowitz, Ira, Huerou, Yvan Le, Mohr, Peter J., Wang, Bin, Blake, Jim F., Lyon, Michael A., Gunawardana, Indrani, Chicarelli, Mark, Wallace, Eli, Gross, Stefan
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Abstract B254: Extended target-coverage by selective Chk1 inhibitors enhances pharmacodynamic inhibition of Chk1 signaling and antitumor activity in vivo
Humphries, Michael J., von Carlowitz, Ira, Le Huerou, Yvan, Randolph, Nikole, Mohr, Peter J., Wang, Bin, Lyon, Michael A., Gunawardana, Indrani, Chicarelli, Mark, Blake, Jim F., Schrag, Michael L., Winski, Shannon L., Wallace, Eli
Published in Molecular cancer therapeutics (10.12.2009)
Published in Molecular cancer therapeutics (10.12.2009)
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Prodrug thiamine analogs as inhibitors of the enzyme transketolase
Le Huerou, Yvan, Gunawardana, Indrani, Thomas, Allen A., Boyd, Steven A., de Meese, Jason, deWolf, Walter, Gonzales, Steven S., Han, May, Hayter, Laura, Kaplan, Tomas, Lemieux, Christine, Lee, Patrice, Pheneger, Jed, Poch, Gregory, Romoff, Todd T., Sullivan, Francis, Weiler, Solly, Wright, S. Kirk, Lin, Jie
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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New cytotoxic analogues of annonaceous acetogenins
Rodier, S, Le Huerou, Y, Renoux, B, Doyon, J, Renard, P, Pierré, A, Gesson, J P, Grée, R
Published in Anti-cancer drug design (01.04.2001)
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Published in Anti-cancer drug design (01.04.2001)
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The microbiological hydroxylation of 3α,5-cycloandrostanes by Cephalosporium aphidicola
Bensasson, Caroline S., Hanson, James R., Le Huerou, Yvan
Published in Phytochemistry (Oxford) (01.12.1999)
Published in Phytochemistry (Oxford) (01.12.1999)
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Journal Article
Pyrrolopyridines as kinase inhibitors
Lyon, Michael, Mohr, Peter J, Blake, James F, Wang, Bin, Chicarelli, Mark Joseph, Le Huerou, Yvan, Gunawardana, Indrani W, Wallace, Eli M
Year of Publication 15.05.2018
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Year of Publication 15.05.2018
Patent
PYRROLOPYRIDINES AS KINASE INHIBITORS
Le Huerou Yvan, Lyon Michael, Chicarelli Mark Joseph, Wallace Eli M, Wang Bin, Blake James F, Gunawardana Indrani W, Mohr Peter J
Year of Publication 22.12.2016
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Year of Publication 22.12.2016
Patent
Triazolopyridine compounds as PIM kinase inhibitors
Xu, Rui, Lyon, Michael, Blake, James F, Wang, Bin, Le Huerou, Yvan, Robinson, John E, De Meese, Lisa A, Delisle, Robert Kirk, Wallace, Eli M, Graham, James M
Year of Publication 08.12.2016
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Year of Publication 08.12.2016
Patent
TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS
Xu, Rui, Lyon, Michael, Blake, James F, Wang, Bin, Le Huerou, Yvan, Robinson, John E, De Meese, Lisa A, Delisle, Robert Kirk, Wallace, Eli M, Graham, James M
Year of Publication 08.04.2016
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Year of Publication 08.04.2016
Patent
Pyrrolopyridines as kinase inhibitors
Le Huerou, Yvan, Blake, James F, Gunawardana, Indrani W, Mohr, Peter J, Wallace, Eli M, Wang, Bin, Chicarelli, Mark Joseph, Lyon, Michael
Year of Publication 15.05.2012
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Year of Publication 15.05.2012
Patent
Thioalkeneamides as transketolase inhibitors
Boyd, Steven A, Condroski, Kevin R, Thomas, Allen, Gonzales, Stephen S, Gunawardana, Indrani W, Huerou, Yvan Le, Romoff, Todd T, Sullivan, Francis X
Year of Publication 01.02.2011
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Year of Publication 01.02.2011
Patent