Algorithm-aided engineering of aliphatic halogenase WelO5 for the asymmetric late-stage functionalization of soraphens
Büchler, Johannes, Malca, Sumire Honda, Patsch, David, Voss, Moritz, Turner, Nicholas J, Bornscheuer, Uwe T, Allemann, Oliver, Le Chapelain, Camille, Lumbroso, Alexandre, Loiseleur, Olivier, Buller, Rebecca
Published in Nature communications (18.01.2022)
Published in Nature communications (18.01.2022)
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Journal Article
Rational Design of Proteasome Inhibitors as Antimalarial Drugs
Le Chapelain, Camille, Groll, Michael
Published in Angewandte Chemie (International ed.) (23.05.2016)
Published in Angewandte Chemie (International ed.) (23.05.2016)
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Journal Article
Activation, Structure, Biosynthesis and Bioactivity of Glidobactin‐like Proteasome Inhibitors from Photorhabdus laumondii
Zhao, Lei, Le Chapelain, Camille, Brachmann, Alexander O., Kaiser, Marcel, Groll, Michael, Bode, Helge B.
Published in Chembiochem : a European journal of chemical biology (04.05.2021)
Published in Chembiochem : a European journal of chemical biology (04.05.2021)
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Journal Article
Synthesis and Biological Evaluation of Chlorinated Analogs of Leukotoxin Diol
Nilewski, Christian, Chapelain, Camille Le, Wolfrum, Susanne, Carreira, Erick M
Published in Organic letters (20.11.2015)
Published in Organic letters (20.11.2015)
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Journal Article
A Collaborative Journey towards the Late‐Stage Functionalization of Added‐Value Chemicals Using Engineered Halogenases
Büchler, Johannes, Hegarty, Eimear, Schroer, Kirsten, Snajdrova, Radka, Turner, Nicholas J., Loiseleur, Olivier, Buller, Rebecca, Le Chapelain, Camille
Published in Helvetica chimica acta (01.01.2023)
Published in Helvetica chimica acta (01.01.2023)
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Journal Article
Structural Elucidation of a Nonpeptidic Inhibitor Specific for the Human Immunoproteasome
Cui, Haissi, Baur, Regina, Le Chapelain, Camille, Dubiella, Christian, Heinemeyer, Wolfgang, Huber, Eva M., Groll, Michael
Published in Chembiochem : a European journal of chemical biology (16.03.2017)
Published in Chembiochem : a European journal of chemical biology (16.03.2017)
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Journal Article
Strategy towards the enantioselective synthesis of schiglautone AThis work was carried out between March 2011 and December 2014 in the laboratory of Prof. Carreira at ETH Zürich and is part of the author's PhD thesis (C. Le Chapelain, ETH Zürich, April 2015, DOI 10.3929/ethz-a-010510664).Electronic supplementary information (ESI) available: Full experimental, copies of NMR spectra for all new compounds, SFC chromatograms. See DOI: 10.1039/c7ob00766c
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Journal Article
Front Cover: Activation, Structure, Biosynthesis and Bioactivity of Glidobactin‐like Proteasome Inhibitors from Photorhabdus laumondii (ChemBioChem 9/2021)
Zhao, Lei, Le Chapelain, Camille, Brachmann, Alexander O., Kaiser, Marcel, Groll, Michael, Bode, Helge B.
Published in Chembiochem : a European journal of chemical biology (04.05.2021)
Published in Chembiochem : a European journal of chemical biology (04.05.2021)
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Journal Article
Design, synthesis, and evaluation of cystargolide-based β-lactones as potent proteasome inhibitors
Niroula, Doleshwar, Hallada, Liam P., Le Chapelain, Camille, Ganegamage, Susantha K., Dotson, Devon, Rogelj, Snezna, Groll, Michael, Tello-Aburto, Rodolfo
Published in European journal of medicinal chemistry (05.09.2018)
Published in European journal of medicinal chemistry (05.09.2018)
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Journal Article
Sequential Inactivation of Gliotoxin by the S‑Methyltransferase TmtA
Duell, Elke R, Glaser, Manuel, Le Chapelain, Camille, Antes, Iris, Groll, Michael, Huber, Eva M
Published in ACS chemical biology (15.04.2016)
Published in ACS chemical biology (15.04.2016)
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Journal Article
Imidazole- and Benzimidazole-Based Inhibitors of the Kinase IspE: Targeting the Substrate-Binding Site and the Triphosphate-Binding Loop of the ATP Site
Mombelli, Paolo, Le Chapelain, Camille, Munzinger, Noah, Joliat, Evelyne, Illarionov, Boris, Schweizer, W. Bernd, Hirsch, Anna K. H., Fischer, Markus, Bacher, Adelbert, Diederich, François
Published in European journal of organic chemistry (01.02.2013)
Published in European journal of organic chemistry (01.02.2013)
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Journal Article
IMIDAZO[1,2-A]PYRIDINE DERIVATIVES
POULIOT, Martin, FINKBEINER, Peter, JEANMART, Stephane André Marie, LE CHAPELAIN, Camille, SCARBOROUGH, Christopher Charles, GERMAIN, Nicolas, BONVALOT, Damien
Year of Publication 20.06.2024
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Year of Publication 20.06.2024
Patent
BENZIMIDAZOLE DERIVATIVES
POULIOT, Martin, JEANMART, Stephane André Marie, DAPIAGGI, Federico, LE CHAPELAIN, Camille, GERMAIN, Nicolas, GROSHEVA, Daria, BONVALOT, Damien
Year of Publication 20.06.2024
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Year of Publication 20.06.2024
Patent
PESTICIDALLY ACTIVE DIAZINE-AMIDE COMPOUNDS
PHADTE, Mangala, WEISS, Matthias, BERARDOZZI, Simone, EL QACEMI, Myriem, LE CHAPELAIN, Camille, JEANGUENAT, André, HALL, Roger Graham, PITTERNA, Thomas, KILARU, Jagadeesh Prathap
Year of Publication 29.08.2024
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Year of Publication 29.08.2024
Patent
PESTICIDALLY ACTIVE DIAZINE-AMIDE COMPOUNDS
PHADTE, Mangala, WEISS, Matthias, BERARDOZZI, Simone, EL QACEMI, Myriem, LE CHAPELAIN, Camille, JEANGUENAT, André, HALL, Roger Graham, PITTERNA, Thomas, KILARU, Jagadeesh Prathap
Year of Publication 17.04.2024
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Year of Publication 17.04.2024
Patent
PESTICIDALLY ACTIVE PYRAZINE-AMIDE COMPOUNDS
RENDLER, Sebastian, GAGNEPAIN, Julien Daniel Henri, EMERY, Daniel, SCHAETZER, Jürgen Harry, LE CHAPELAIN, Camille, PITTERNA, Thomas
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
Patent