Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles
Kita, Diogo Henrique, Guragossian, Nathalie, Zattoni, Ingrid Fatima, Moure, Vivian Rotuno, Rego, Fabiane Gomes de Moraes, Lusvarghi, Sabrina, Moulenat, Thomas, Belhani, Billel, Picheth, Geraldo, Bouacida, Sofiane, Bouaziz, Zouhair, Marminon, Christelle, Berredjem, Malika, Jose, Joachim, Gonçalves, Marcos Brown, Ambudkar, Suresh V., Valdameri, Glaucio, Le Borgne, Marc
Published in Scientific reports (19.01.2021)
Published in Scientific reports (19.01.2021)
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Journal Article
Discovery of holoenzyme-disrupting chemicals as substrate-selective CK2 inhibitors
Kufareva, Irina, Bestgen, Benoit, Brear, Paul, Prudent, Renaud, Laudet, Béatrice, Moucadel, Virginie, Ettaoussi, Mohamed, Sautel, Celine F., Krimm, Isabelle, Engel, Matthias, Filhol, Odile, Borgne, Marc Le, Lomberget, Thierry, Cochet, Claude, Abagyan, Ruben
Published in Scientific reports (04.11.2019)
Published in Scientific reports (04.11.2019)
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Journal Article
Tetanus Toxin Fragment C: Structure, Drug Discovery Research and Production
Bayart, Caroline, Mularoni, Angélique, Hemmani, Nada, Kerachni, Soumeya, Jose, Joachim, Gouet, Patrice, Paladino, Joseph, Le Borgne, Marc
Published in Pharmaceuticals (Basel, Switzerland) (17.06.2022)
Published in Pharmaceuticals (Basel, Switzerland) (17.06.2022)
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Journal Article
QSAR Model of Indeno[1,2- b ]indole Derivatives and Identification of N -isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3- b ]furan-3-carboxamide as a Potent CK2 Inhibitor
Haidar, Samer, Marminon, Christelle, Aichele, Dagmar, Nacereddine, Abdelhamid, Zeinyeh, Wael, Bouzina, Abdeslem, Berredjem, Malika, Ettouati, Laurent, Bouaziz, Zouhair, Le Borgne, Marc, Jose, Joachim
Published in Molecules (Basel, Switzerland) (01.01.2020)
Published in Molecules (Basel, Switzerland) (01.01.2020)
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Journal Article
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols
Lebouvier, Nicolas, Pagniez, Fabrice, Na, Young Min, Shi, Da, Pinson, Patricia, Marchivie, Mathieu, Guillon, Jean, Hakki, Tarek, Bernhardt, Rita, Yee, Sook Wah, Simons, Claire, Lézé, Marie-Pierre, Hartmann, Rolf W, Mularoni, Angélique, Le Baut, Guillaume, Krimm, Isabelle, Abagyan, Ruben, Le Pape, Patrice, Le Borgne, Marc
Published in Pharmaceuticals (Basel, Switzerland) (08.08.2020)
Published in Pharmaceuticals (Basel, Switzerland) (08.08.2020)
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Journal Article
Occurrence of the Synthetic Analgesic Tramadol in an African Medicinal Plant
Boumendjel, Ahcène, Sotoing Taïwe, Germain, Ngo Bum, Elisabeth, Chabrol, Tanguy, Beney, Chantal, Sinniger, Valérie, Haudecoeur, Romain, Marcourt, Laurence, Challal, Soura, Ferreira Queiroz, Emerson, Souard, Florence, Le Borgne, Marc, Lomberget, Thierry, Depaulis, Antoine, Lavaud, Catherine, Robins, Richard, Wolfender, Jean-Luc, Bonaz, Bruno, De Waard, Michel
Published in Angewandte Chemie International Edition (04.11.2013)
Published in Angewandte Chemie International Edition (04.11.2013)
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Journal Article
Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2
Alchab, Faten, Ettouati, Laurent, Bouaziz, Zouhair, Bollacke, Andre, Delcros, Jean-Guy, Gertzen, Christoph G W, Gohlke, Holger, Pinaud, Noël, Marchivie, Mathieu, Guillon, Jean, Fenet, Bernard, Jose, Joachim, Borgne, Marc Le
Published in Pharmaceuticals (Basel, Switzerland) (08.06.2015)
Published in Pharmaceuticals (Basel, Switzerland) (08.06.2015)
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Journal Article
Behaviour of Tetrabenazine in Acid Medium: Reassessment and Impact on Formulation
Ettouati, Laurent, Senta-Loys, Zoé, Bourgeois, Sandrine, Fenet, Bernard, Borgne, Marc Le, Fessi, Hatem
Published in Pharmaceutics (01.01.2019)
Published in Pharmaceutics (01.01.2019)
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Journal Article
Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity
Gozzi, Gustavo Jabor, Bouaziz, Zouhair, Winter, Evelyn, Daflon-Yunes, Nathalia, Honorat, Mylène, Guragossian, Nathalie, Marminon, Christelle, Valdameri, Glaucio, Bollacke, Andre, Guillon, Jean, Pinaud, Noël, Marchivie, Mathieu, Cadena, Silvia M, Jose, Joachim, Le Borgne, Marc, Di Pietro, Attilio
Published in Drug design, development and therapy (01.01.2015)
Published in Drug design, development and therapy (01.01.2015)
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Journal Article
1st Joint European Conference on Therapeutic Targets and Medicinal Chemistry (TTMC 2015)
Le Borgne, Marc, Haidar, Samer, Duval, Olivier, Wünsch, Bernhard, Jose, Joachim
Published in Pharmaceuticals (26.12.2015)
Published in Pharmaceuticals (26.12.2015)
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Journal Article
Publication
Toxicological Risks of the Cobalt–Chromium Alloys in Dentistry: A Systematic Review
Grosgogeat, Brigitte, Vaicelyte, Alina, Gauthier, Rémy, Janssen, Christine, Le Borgne, Marc
Published in Materials (23.08.2022)
Published in Materials (23.08.2022)
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Journal Article
Biological exploration of a novel 1,2,4-triazole-indole hybrid molecule as antifungal agent
Pagniez, Fabrice, Lebouvier, Nicolas, Na, Young Min, Ourliac-Garnier, Isabelle, Picot, Carine, Le Borgne, Marc, Le Pape, Patrice
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2
Bouzina, Abdeslem, Berredjem, Malika, Bouacida, Sofiane, Bachari, Khaldoun, Marminon, Christelle, Borgne, Marc Le, Bouaziz, Zouhair, Bouone, Yousra Ouafa
Published in Journal of molecular structure (05.06.2022)
Published in Journal of molecular structure (05.06.2022)
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Journal Article
Solubility enhancement of mefenamic acid by inclusion complex with β-cyclodextrin: in silico modelling, formulation, characterisation, and in vitro studies
Sid, Dounia, Baitiche, Milad, Elbahri, Zineb, Djerboua, Ferhat, Boutahala, Mokhtar, Bouaziz, Zouhair, Le Borgne, Marc
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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Journal Article
The combined use of analytical tools for exploring tetanus toxin and tetanus toxoid structures
Bayart, Caroline, Peronin, Sébastien, Jean, Elisa, Paladino, Joseph, Talaga, Philippe, Borgne, Marc Le
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2017)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2017)
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Journal Article
Toward selective CK2alpha and CK2alpha’ inhibitors: Development of a novel whole-cell kinase assay by Autodisplay of catalytic CK2alpha
Bollacke, Andre, Nienberg, Christian, Borgne, Marc Le, Jose, Joachim
Published in Journal of pharmaceutical and biomedical analysis (20.03.2016)
Published in Journal of pharmaceutical and biomedical analysis (20.03.2016)
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Journal Article