4-{8-아미노-3-[(2S)-1--피롤리딘-2-일]이미다조[1,5-a]-피라진-1-일}N--벤즈아미드의 제조 공정
LAWLER MICHAEL JOSEPH, GOLDEN MICHAEL DAVID, GARREY RUSTAM FERDINAND, WANG ANGANG, TELFORD ALEXANDER JAMES, EVARTS JERRY, CHAN LAI CHUN, SHORT DAVID ALLEN, VERSTAPPEN MATHILDA MARIA HENRICA, JACKSON LUCINDA VICTORIA, MILLARD KIRSTY JANE, VAN EIJK PETER JOHANNES SERVAAS SAVIO, LITJENS REMY E. J. N, COX ROBERT JOHN, ZIJP ERIC JURRIEN, VOS FRANK L. M, HUGHES SHAUN ALAN, COOPER KATIE GRACE, PHILLIPS ANDREW JOHN, BETHEL PAUL ALLEN, JUNYING QIU
Year of Publication 11.05.2021
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Year of Publication 11.05.2021
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-a]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
ZIJP, Eric Jurriën, SHORT, David Allen, LAWLER, Michael Joseph, JACKSON, Lucinda Victoria, HUGHES, Shaun Alan, JUNYING, Qiu, COOPER, Katie Grace, GOLDEN, Michael David, WANG, Angang, EVARTS, Jerry, VERSTAPPEN, Mathilda Maria Henrica, GARREY, Rustam Ferdinand, PHILLIPS, Andrew John, VAN EIJK, Peter Johannes Servaas Savio, VOS, Frank L. M, TELFORD, Alexander James, CHAN, Lai Chun, COX, Robert John, LITJENS, Remy E. J. N, BETHEL, Paul Allen, MILLARD, Kirsty Jane
Year of Publication 26.09.2024
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Year of Publication 26.09.2024
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Processes for the preparation of 4-{8-amino-3-[(2S)-1-(but-2-ynoyl)-pyrrolidin-2-yl]imidazo[1,5-a]-pyrazin-1-yl}N-(pyridin-2-yl)-benzamide
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Litjens, Remy E. J. N, Verstappen, Mathilda Maria Henrica, Vos, Frank L. M, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Chan, Lai Chun, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 02.07.2024
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Year of Publication 02.07.2024
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Litjens, Remy E. J. N, Verstappen, Mathilda Maria Henrica, Vos, Frank L. M, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Chan, Lai Chun, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 02.05.2024
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Year of Publication 02.05.2024
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Litjens, Remy E. J. N, Verstappen, Mathilda Maria Henrica, Vos, Frank L. M, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Chan, Lai Chun, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 25.01.2024
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Year of Publication 25.01.2024
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Litjens, Remy E. J. N, Verstappen, Mathilda Maria Henrica, Vos, Frank L. M, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Chan, Lai Chun, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 03.08.2023
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Year of Publication 03.08.2023
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Verstappen, Mathilda Maria Henrica, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Vos, Frank L.M, Chan, Lai Chun, Litjens, Remy E.J.N, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-a]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
ZIJP, Eric Jurriën, SHORT, David Allen, LAWLER, Michael Joseph, JACKSON, Lucinda Victoria, HUGHES, Shaun Alan, JUNYING, Qiu, COOPER, Katie Grace, GOLDEN, Michael David, WANG, Angang, EVARTS, Jerry, VERSTAPPEN, Mathilda Maria Henrica, GARREY, Rustam Ferdinand, PHILLIPS, Andrew John, VAN EIJK, Peter Johannes Servaas Savio, VOS, Frank L. M, TELFORD, Alexander James, CHAN, Lai Chun, COX, Robert John, LITJENS, Remy E. J. N, BETHEL, Paul Allen, MILLARD, Kirsty Jane
Year of Publication 28.04.2022
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Year of Publication 28.04.2022
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
Cox, Robert John, Garrey, Rustam Ferdinand, Bethel, Paul Allen, Short, David Allen, Telford, Alexander James, Zijp, Eric Jurriën, Jackson, Lucinda Victoria, Cooper, Katie Grace, Van Eijk, Peter Johannes Servaas Savio, Junying, Qiu, Hughes, Shaun Alan, Verstappen, Mathilda Maria Henrica, Lawler, Michael Joseph, Evarts, Jerry, Millard, Kirsty Jane, Vos, Frank L.M, Chan, Lai Chun, Litjens, Remy E.J.N, Wang, Angang, Golden, Michael David, Phillips, Andrew John
Year of Publication 03.03.2022
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Year of Publication 03.03.2022
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Processes for the preparation of 4-{8-amino-3-[(2S)-1-(but-2-ynoyl)-pyrrolidin-2-yl]imidazo[1,5-a]-pyrazin-1-yl}N-(pyridin-2-yl)-benzamide
ZIJP, Eric Jurriën, SHORT, David Allen, LAWLER, Michael Joseph, JACKSON, Lucinda Victoria, HUGHES, Shaun Alan, JUNYING, Qiu, COOPER, Katie Grace, GOLDEN, Michael David, WANG, Angang, EVARTS, Jerry, VERSTAPPEN, Mathilda Maria Henrica, GARREY, Rustam Ferdinand, PHILLIPS, Andrew John, VAN EIJK, Peter Johannes Servaas Savio, VOS, Frank L. M, TELFORD, Alexander James, CHAN, Lai Chun, COX, Robert John, LITJENS, Remy E. J. N, BETHEL, Paul Allen, MILLARD, Kirsty Jane
Year of Publication 27.01.2022
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Year of Publication 27.01.2022
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PROCÉDÉS DE PRÉPARATION DE 4-(8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL] IMIDAZO[1,5-A]-PYRAZIN-1-YL)N-(PYRIDIN-2-YL)-BENZAMIDE
BETHEL, Paul, Allen, COOPER, Katie, Grace, TELFORD, Alexander, James, GOLDEN, Michael, David, MILLARD, Kirsty, Jane, SHORT, David, Allen, JUNYING, Qiu, GARREY, Rustam, Ferdinand, WANG, Angang, EVARTS, Jerry, VOS, Frank, L. M, HUGHES, Shaun, Alan, LITJENS, Remy E. J. N, VERSTAPPEN, Mathilda, Maria, Henrica, CHAN, Lai, Chun, COX, Robert, John, VAN EIJK, Peter, Johannes, Servaas, Savio, ZIJP, Eric, Jurriën, LAWLER, Michael, Joseph, PHILLIPS, Andrew, John, JACKSON, Lucinda, Victoria
Year of Publication 08.12.2021
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Year of Publication 08.12.2021
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
BETHEL, Paul, Allen, COOPER, Katie, Grace, TELFORD, Alexander, James, GOLDEN, Michael, David, MILLARD, Kirsty, Jane, SHORT, David, Allen, JUNYING, Qiu, WANG, Angang, GARREY, Rustam, Ferdinand, EVARTS, Jerry, VOS, Frank, L. M, HUGHES, Shaun, Alan, LITJENS, Remy E. J. N, VERSTAPPEN, Mathilda, Maria, Henrica, CHAN, Lai, Chun, COX, Robert, John, VAN EIJK, Peter, Johannes, Servaas, Savio, ZIJP, Eric, Jurriën, PHILLIPS, Andrew, John, LAWLER, Michael, Joseph, JACKSON, Lucinda, Victoria
Year of Publication 07.07.2021
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Year of Publication 07.07.2021
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Processes for the preparation of 4-{8-amino-3-((2S)-1-(but-2-ynoyl)-pyrrolidin-2-yl)imidazo(1,5-a)-pyrazin-1-yl}N-(pyridin-2-yl)-benzamide
ZIJP, Eric Jurriën, SHORT, David Allen, LAWLER, Michael Joseph, JACKSON, Lucinda Victoria, HUGHES, Shaun Alan, JUNYING, Qiu, COOPER, Katie Grace, GOLDEN, Michael David, WANG, Angang, EVARTS, Jerry, VERSTAPPEN, Mathilda Maria Henrica, GARREY, Rustam Ferdinand, PHILLIPS, Andrew John, VAN EIJK, Peter Johannes Servaas Savio, VOS, Frank L. M, TELFORD, Alexander James, CHAN, Lai Chun, COX, Robert John, LITJENS, Remy E. J. N, BETHEL, Paul Allen, MILLARD, Kirsty Jane
Year of Publication 22.04.2021
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Year of Publication 22.04.2021
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
WANG, ANGANG, LITJENS, REMY E. J. N, VERSTAPPEN, MATHILDA MARIA HENRICA, BETHEL, PAUL ALLEN, MILLARD, KIRSTY JANE, LAWLER, MICHAEL JOSEPH, VOS, FRANK L. M, TELFORD, ALEXANDER JAMES, VAN EIJK, PETER JOHANNES SERVAAS SAVIO, ZIJP, ERIC JURRIEN, CHAN, LAI CHUN, COX, ROBERT JOHN, COOPER, KATIE GRACE, GARREY, RUSTAM FERDINAND, GOLDEN, MICHAEL DAVID, SHORT, DAVID ALLEN, JUNYING, QIU, JACKSON, LUCINDA VICTORIA, EVARTS, JERRY, HUGHES, SHAUN ALAN, PHILLIPS, ANDREW JOHN
Year of Publication 05.03.2020
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Year of Publication 05.03.2020
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOY L)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)- BENZAMIDE
MILLARD Kirsty Jane, VAN EIJK Peter Johannes Servaas Savio, WANG Angang, LAWLER Michael Joseph, COOPER Katie Grace, SHORT David Allen, GOLDEN Michael David, VOS Frank L. M, JUNYING Qiu, VERSTAPPEN Mathilda Maria Henrica, PHILLIPS Andrew John, TELFORD Alexander James, ZIJP Eric Jurriën, BETHEL Paul Allen, EVARTS Jerry, COX Robert John, HUGHES Shaun Alan, LITJENS Remy E. J. N, GARREY Rustam Ferdinand, JACKSON Lucinda Victoria, CHAN Lai Chun
Year of Publication 19.10.2023
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Year of Publication 19.10.2023
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Process for the preparation of N,N-dicyclopropyl-4-(1,5-dimethyl-1H-pyrazol-3-ylamino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide
Eastgate Martin D, Hay Michael Bryan, Zhu Keming, Xiao Yi, Wei Carolyn S, Desai Lopa V, Regens Christopher S, Fitzgerald Monica, Rosner Thorsten, Beutner Gregory L, Zheng Bin, Strotman Neil, Cuniere Nicolas, Cohen Benjamin, Lawler Michael Joseph, Lobben Paul C, Gao Qi
Year of Publication 13.12.2016
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Year of Publication 13.12.2016
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PROCESS FOR THE PREPARATION OF N,N-DICYCLOPROPYL-4-(1,5-DIMETHYL-1H-PYRAZOL-3-YLAMINO)-6-ETHYL-1-METHYL-1,6-DIHYDROIMIDAZO[4,5-d]PYRROLO[2,3-b]PYRIDINE-7-CARBOXAMIDE
Eastgate Martin D, Hay Michael Bryan, Zhu Keming, Xiao Yi, Wei Carolyn S, Desai Lopa V, Regens Christopher S, Fitzgerald Monica, Rosner Thorsten, Beutner Gregory L, Zheng Bin, Strotman Neil, Cuniere Nicolas, Cohen Benjamin, Lawler Michael Joseph, Lobben Paul C, Gao Qi
Year of Publication 11.08.2016
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Year of Publication 11.08.2016
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PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOY L)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)- BENZAMIDE
MILLARD Kirsty Jane, VAN EIJK Peter Johannes Servaas Savio, WANG Angang, LAWLER Michael Joseph, COOPER Katie Grace, SHORT David Allen, GOLDEN Michael David, VOS Frank L. M, JUNYING Qiu, VERSTAPPEN Mathilda Maria Henrica, PHILLIPS Andrew John, TELFORD Alexander James, ZIJP Eric Jurriën, BETHEL Paul Allen, EVARTS Jerry, COX Robert John, HUGHES Shaun Alan, LITJENS Remy E. J. N, GARREY Rustam Ferdinand, JACKSON Lucinda Victoria, CHAN Lai Chun
Year of Publication 27.05.2021
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Year of Publication 27.05.2021
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processos para a preparação de 4-{8-amino-3-[(2s)-1-(but-2-inoil)-pirrolidin-2-il]imidazo[1,5-a]-pirazin-1-il}-n-(piridin-2-il)-benzamida
ERIC JURRIËN ZIJP, PETER JOHANNES SERVAAS SAVIO VAN EIJK, MICHAEL DAVID GOLDEN, LUCINDA VICTORIA JACKSON, KIRSTY JANE MILLARD, MATHILDA MARIA HENRICA VERSTAPPEN, MICHAEL JOSEPH LAWLER, ALEXANDER JAMES TELFORD, FRANK L. M. VOS, JERRY EVARTS, SHAUN ALAN HUGHES, RUSTAM FERDINAND GARREY, QIU JUNYING, REMY E. J. N. LITJENS, LAI CHUN CHAN, ROBERT JOHN COX, ANGANG WANG, DAVID ALLEN SHORT, KATIE GRACE COOPER, ANDREW JOHN PHILLIPS, PAUL ALLEN BETHEL
Year of Publication 18.05.2021
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Year of Publication 18.05.2021
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Procesos para la preparación de 4-{8-amino-3-[(2s)-1-(but-2-inoil)pirrolidin-2-il]imidazo[1,5-a]-pirazin-1-il}-n-(piridin-2-il)benzamida
ZIJP, Eric Jurriën, SHORT, David Allen, LAWLER, Michael Joseph, JACKSON, Lucinda Victoria, HUGHES, Shaun Alan, JUNYING, Qiu, COOPER, Katie Grace, GOLDEN, Michael David, WANG, Angang, EVARTS, Jerry, VERSTAPPEN, Mathilda Maria Henrica, GARREY, Rustam Ferdinand, PHILLIPS, Andrew John, VAN EIJK, Peter Johannes Servaas Savio, VOS, Frank L. M, TELFORD, Alexander James, CHAN, Lai Chun, COX, Robert John, LITJENS, Remy E. J. N, BETHEL, Paul Allen, MILLARD, Kirsty Jane
Year of Publication 08.04.2021
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Year of Publication 08.04.2021
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