Search Results - "LASSALLE, GILBERT" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Characterization of Glycosaminoglycan (GAG) Sulfatases from the Human Gut Symbiont Bacteroides thetaiotaomicron Reveals the First GAG-specific Bacterial Endosulfatase

Characterization of Glycosaminoglycan (GAG) Sulfatases from the Human Gut Symbiont Bacteroides thetaiotaomicron Reveals the First GAG-specific Bacterial Endosulfatase

by Ulmer, Jonathan E., Vilén, Eric Morssing, Namburi, Ramesh Babu, Benjdia, Alhosna, Beneteau, Julie, Malleron, Annie, Bonnaffé, David, Driguez, Pierre-Alexandre, Descroix, Karine, Lassalle, Gilbert, Le Narvor, Christine, Sandström, Corine, Spillmann, Dorothe, Berteau, Olivier
Published in The Journal of biological chemistry (29.08.2014)

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Journal Article

5‑Chlorothiophene-2-carboxylic Acid [(S)‑2-[2-Methyl-3-(2-oxopyrrolidin-1-yl)benzenesulfonylamino]-3-(4-methylpiperazin-1-yl)-3-oxopropyl]amide (SAR107375), a Selective and Potent Orally Active Dual Thrombin and Factor Xa Inhibitor

5‑Chlorothiophene-2-carboxylic Acid [(S)‑2-[2-Methyl-3-(2-oxopyrrolidin-1-yl)benzenesulfonylamino]-3-(4-methylpiperazin-1-yl)-3-oxopropyl]amide (SAR107375), a Selective and Potent Orally Active Dual Thrombin and Factor Xa Inhibitor

by Meneyrol, Jerome, Follmann, Markus, Lassalle, Gilbert, Wehner, Volkmar, Barre, Guillaume, Rousseaux, Tristan, Altenburger, Jean-Michel, Petit, Frederic, Bocskei, Zsolt, Schreuder, Herman, Alet, Nathalie, Herault, Jean-Pascal, Millet, Laurence, Dol, Frederique, Florian, Peter, Schaeffer, Paul, Sadoun, Freddy, Klieber, Sylvie, Briot, Christophe, Bono, Françoise, Herbert, Jean-Marc
Published in Journal of medicinal chemistry (12.12.2013)

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Journal Article

SSR182289A, a selective and potent orally active thrombin inhibitor

SSR182289A, a selective and potent orally active thrombin inhibitor

by Altenburger, Jean-Michel, Lassalle, Gilbert Y., Matrougui, Mostapha, Galtier, Daniel, Jetha, Jean-Claude, Bocskei, Zsolt, Berry, Christopher N., Lunven, Catherine, Lorrain, Janine, Herault, Jean-Pascal, Schaeffer, Paul, O'Connor, Stephen E., Herbert, Jean-Marc
Published in Bioorganic & medicinal chemistry (01.04.2004)

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Influence of Heparin Mimetics on Assembly of the FGF·FGFR4 Signaling Complex

Influence of Heparin Mimetics on Assembly of the FGF·FGFR4 Signaling Complex

by Saxena, Krishna, Schieborr, Ulrich, Anderka, Oliver, Duchardt-Ferner, Elke, Elshorst, Bettina, Gande, Santosh Lakshmi, Janzon, Julia, Kudlinzki, Denis, Sreeramulu, Sridhar, Dreyer, Matthias K., Wendt, K. Ulrich, Herbert, Corentin, Duchaussoy, Philippe, Bianciotto, Marc, Driguez, Pierre-Alexandre, Lassalle, Gilbert, Savi, Pierre, Mohammadi, Moosa, Bono, Françoise, Schwalbe, Harald
Published in The Journal of biological chemistry (20.08.2010)

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Journal Article

SSR182289A, a Novel, Orally Active Thrombin Inhibitor: In Vitro Profile and ex Vivo Anticoagulant Activity

by Berry, Christopher N, Lassalle, Gilbert, Lunven, Catherine, Altenburger, Jean-Michel, Guilbert, Frédérique, Lalé, Alain, Hérault, Jean-Pascal, Lecoffre, Catherine, Pfersdorff, Christian, Herbert, Jean-Marc, O'Connor, Stephen E
Published in The Journal of pharmacology and experimental therapeutics (01.12.2002)

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Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling

Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling

by Herbert, Corentin, Schieborr, Ulrich, Saxena, Krishna, Juraszek, Jarek, De Smet, Frederik, Alcouffe, Chantal, Bianciotto, Marc, Saladino, Giorgio, Sibrac, David, Kudlinzki, Denis, Sreeramulu, Sridhar, Brown, Alan, Rigon, Patrice, Herault, Jean-Pascal, Lassalle, Gilbert, Blundell, Tom L., Rousseau, Frederic, Gils, Ann, Schymkowitz, Joost, Tompa, Peter, Herbert, Jean-Marc, Carmeliet, Peter, Gervasio, Francesco Luigi, Schwalbe, Harald, Bono, Françoise
Published in Cancer cell (15.04.2013)

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European Medicinal Chemistry Leaders in Industry (EMCL) – On the Status and Future of Medicinal Chemistry Research in Europe

European Medicinal Chemistry Leaders in Industry (EMCL) – On the Status and Future of Medicinal Chemistry Research in Europe

by Ali, Amjad, Bauser, Marcus, Bertrand, Sophie, Blackaby, Wesley, Boss, Christoph, Bossart, Martin, Hall, Adrian, Binch, Hayley, Czechtizky, Werngard, Gijsen, Harrie, Haning, Helmut, Hartung, Ingo V., Kilburn, Paul, Lassalle, Gilbert, Lücking, Ulrich, Mack, Jürgen, Missbach, Martin, Otsomaa, Leena, Torrens, Antoni, Wagner, Michael, Walter, Magnus, Weinstabl, Harald, Hijfte, Luc, Nussbaum, Franz
Published in ChemMedChem (03.07.2023)

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N‑[6-(4-Butanoyl-5-methyl‑1H‑pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]‑1H‑indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist

N‑[6-(4-Butanoyl-5-methyl‑1H‑pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]‑1H‑indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist

by Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)

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Journal Article

N -[6-(4-Butanoyl-5-methyl-1 H -pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1 H -indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist

N -[6-(4-Butanoyl-5-methyl-1 H -pyrazol-1-yl)pyridazin-3-yl]-5-chloro-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1 H -indole-3-carboxamide (SAR216471), a Novel Intravenous and Oral, Reversible, and Directly Acting P2Y12 Antagonist

by Boldron, Christophe, Besse, Angélina, Bordes, Marie-Françoise, Tissandié, Stéphanie, Yvon, Xavier, Gau, Benjamin, Badorc, Alain, Rousseaux, Tristan, Barré, Guillaume, Meneyrol, Jérôme, Zech, Gernot, Nazare, Marc, Fossey, Valérie, Pflieger, Anne-Marie, Bonnet-Lignon, Sandrine, Millet, Laurence, Briot, Christophe, Dol, Frédérique, Hérault, Jean-Pascal, Savi, Pierre, Lassalle, Gilbert, Delesque, Nathalie, Herbert, Jean-Marc, Bono, Françoise
Published in Journal of medicinal chemistry (11.09.2014)

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Journal Article

Approaches targeting the FGF-FGFR system: a review of the recent patent literature and associated advanced therapeutic agents

Approaches targeting the FGF-FGFR system: a review of the recent patent literature and associated advanced therapeutic agents

by Herbert, Corentin, Lassalle, Gilbert, Alcouffe, Chantal, Bono, Françoise
Published in Pharmaceutical patent analyst (2014)

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Journal Article

Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling

Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling

by Herbert, Corentin, Schieborr, Ulrich, Saxena, Krishna, Juraszek, Jarek, De Smet, Frederik, Alcouffe, Chantal, Bianciotto, Marc, Saladino, Giorgio, Sibrac, David, Kudlinzki, Denis, Sreeramulu, Sridhar, Brown, Alan, Rigon, Patrice, Herault, Jean-Pascal, Lassalle, Gilbert, Blundell, Tom L., Rousseau, Frederic, Gils, Ann, Schymkowitz, Joost, Tompa, Peter, Herbert, Jean-Marc, Carmeliet, Peter, Gervasio, Francesco Luigi, Schwalbe, Harald, Bono, Françoise
Published in Cancer cell (11.07.2016)

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Journal Article

Studies directed toward the total synthesis of cerorubenic acid-III. 2. Analysis of the inability to realize D ring formation by means of extraannular Robinson annulation

Studies directed toward the total synthesis of cerorubenic acid-III. 2. Analysis of the inability to realize D ring formation by means of extraannular Robinson annulation

by Paquette, Leo A, Lassalle, Gilbert Y, Lovely, Carl J
Published in Journal of organic chemistry (01.07.1993)

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Journal Article

Characterization of Gglycosaminoglycan (GAG) sulfatases from the human gut symbiont bacteroides thetaiotaomicron reveals the first GAG-specific bacterial endosulfatase

Characterization of Gglycosaminoglycan (GAG) sulfatases from the human gut symbiont bacteroides thetaiotaomicron reveals the first GAG-specific bacterial endosulfatase

by Ulmer, Jonathan, Vilen, Eric Morssing, Namburi, Ramesh Babu, Benjdia, Alhosna, Beneteau, Julie, Malleron, Annie, Bonnaffe, David, Driguez, Pierre-Alexandre, Descroix, Karine, Lassalle, Gilbert, Le Narvor, Christine, Sandstrom, Corine, Spillmann, Dorothe, Berteau, Olivier
Published in The Journal of biological chemistry (2014)

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Journal Article

INDOLIZINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

INDOLIZINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

by ALCOUFFE CHANTAL, HERBERT CORENTIN, LASSALLE GILBERT
Year of Publication 26.11.2013

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Patent

IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

by ALCOUFFE CHANTAL, KIRSCH REINHARD, HERBERT CORENTIN, LASSALLE GILBERT
Year of Publication 26.11.2013

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Patent

PYRIDINE-PYRIDINONE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

PYRIDINE-PYRIDINONE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

by VOLLE CHALLIER CECILE, MARTIN VALERIE, LASSALLE GILBERT, MCCORT GARY
Year of Publication 11.09.2012

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Patent

PYRAZOLOQUINOLINONE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

PYRAZOLOQUINOLINONE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF

by MACARY KARIM, GUILLO NATHALIE, VIN VALERIE, LASSALLE GILBERT, BENAZET ALEXANDRE, DUCLOS OLIVIER
Year of Publication 02.07.2014

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Patent

DERIVATIVES OF N-[(1H-PYRAZOL-1-YL)ARYL]-1H-INDOLE OR 1H-INDAZOLE-3-CARBOXAMIDE, THEIR PREPARATION AND THEIR USE AS P2Y12 ANTAGONISTS

DERIVATIVES OF N-[(1H-PYRAZOL-1-YL)ARYL]-1H-INDOLE OR 1H-INDAZOLE-3-CARBOXAMIDE, THEIR PREPARATION AND THEIR USE AS P2Y12 ANTAGONISTS

by YVON XAVIER, FOSSEY VALERIE, BADORC ALAIN, BOLDRON CHRISTOPHE, LASSALLE GILBERT, DELESQUE NATHALIE
Year of Publication 27.03.2014

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Patent

2-AMINO-3-(IMIDAZOL-2-YL)-PYRIDIN-4-ONE DERIVATIVES AND THEIR USE AS VEGF RECEPTOR KINASE INHIBITORS

2-AMINO-3-(IMIDAZOL-2-YL)-PYRIDIN-4-ONE DERIVATIVES AND THEIR USE AS VEGF RECEPTOR KINASE INHIBITORS

by STRUB AURELIE, MARTIN VALERIE, LASSALLE GILBERT, RITZELER OLAF, LORGE FRANZ, DUCLOS OLIVIER, BRAUN ALAIN
Year of Publication 04.03.2014

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Patent

SULPHONYLAMINOPYRROLIDINONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

SULPHONYLAMINOPYRROLIDINONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

by KIRSCH REINHARD, PHILIPPO ORTS MARIE CLAIRE, ALET NATHALIE, LASSALLE GILBERT, HERAULT JEAN PASCAL, MALLART SERGIO, ALTENBURGER JEAN MICHEL
Year of Publication 03.09.2014

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Patent

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