Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester
LEAHY, DAVID K, LAPORTE, THOMAS L, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, DISCORDIA, ROBERT P, LOBBEN, PAUL C, PESTI, JAAN A, HAMEDI, MOURAD, XU, ZHONGMIN, THORNTON, JOHN E, SPANGLER, LORI ANN
Year of Publication 12.04.2012
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Year of Publication 12.04.2012
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ΜΕΘΟΔΟΣ ΓΙΑ ΤΗΝ ΠΑΡΑΣΚΕΥΗ [(1R),2S]-2-ΑΜΙΝΟΠΡΟΠΙΟΝΙΚΟΥ 2-[4-(4-ΦΘΟΡΟ-2-ΜΕΘΥΛΟ-1Η-ΙΝΔΟΛ-5-ΥΛΟΞΥ)-5-ΜΕΘΥΛΠΥΡΡΟΛΟ]2,1-F[1,2,4]ΤΡΙΑΖΙΝ-6-ΥΛΟΞΥ]-1-ΜΕΘΥΛΑΙΘΥΛΕΣΤΕΡΑ
LAI Chiajen, LAPORTE Thomas L, PESTI Jaan A, XU Zhongmin, CRISPINO Gerard A, LEAHY David K, MUSLEHIDDINOGLU Jale, HAMEDI Mourad, LOBBEN Paul C, THORNTON John E, DISCORDIA Robert P, SPANGLER Lori Ann
Year of Publication 22.06.2016
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Year of Publication 22.06.2016
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Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2, 1-F][1,2,4]triazin-6-yloxy]-1-methylethyl ester
LEAHY DAVID K, LOBBEN PAUL C, THORNTON JOHN E, MUSLEHIDDINOGLU JALE, HAMEDI MOURAD, GIBSON FRANCIS S, XU ZHONGMIN, DISCORDIA ROBERT P, LAI CHIAJEN, CRISPINO GERARD A, PESTI JAAN A, SPANGLER LORI ANN, LAPORTE THOMAS L
Year of Publication 02.03.2010
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Year of Publication 02.03.2010
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Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2, 1-F][1,2,4]triazin-6-yloxy]-1-methylethyl ester
Crispino, Gerard A, Hamedi, Mourad, LaPorte, Thomas L, Thornton, John E, Pesti, Jaan A, Xu, Zhongmin, Lobben, Paul C, Leahy, David K, Muslehiddinoglu, Jale, Lai, Chiajen, Spangler, Lori Ann, Discordia, Robert P, Gibson, Francis S
Year of Publication 02.03.2010
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Year of Publication 02.03.2010
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PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-F][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LEAHY DAVID K, LOBBEN PAUL C, THORNTON JOHN E, MUSLEHIDDINOGLU JALE, HAMEDI MOURAD, XU ZHONGMIN, DISCORDIA ROBERT P, LAI CHIAJEN, CRISPINO GERARD A, PESTI JAAN A, SPANGLER LORI ANN, LAPORTE THOMAS L
Year of Publication 21.01.2009
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Year of Publication 21.01.2009
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PROCESS FOR THE PREPARATION OF Ý(1R), 2S¨-2-AMINOPROPIONIC ACID 2-Ý4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLOÝ2,1-f¨Ý1,2,4¨TRIAZIN-6-YLOXY¨-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 07.01.2009
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Year of Publication 07.01.2009
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Continuous process for producing hydroxyazapirones by oxidation
DEPUE JEFFREY S, HAMEDI MOURAD, WATSON DANIEL J, CHAN YEUNG Y, DOWDY ERIC D, LAPORTE THOMAS L, SHEN LIFEN
Year of Publication 28.07.2005
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Year of Publication 28.07.2005
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CONTINUOUS PROCESS FOR PRODUCING HYDROXYAZAPIRONES BY OXIDATION
DEPUE, JEFFREY S, CHAN, YEUNG YU, LAPORTE, THOMAS L, WATSON, DANIEL J, DOWDY, ERIC D, SHEN, LIFEN, HAMEDI, MOURAD
Year of Publication 27.07.2006
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Year of Publication 27.07.2006
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Synthesis and Activity of a C-8 Keto Pleuromutilin Derivative
Springer, Dane M., Sorenson, Margaret E., Huang, Stella, Connolly, Timothy P., Bronson, Joanne J., Matson, James A., Hanson, Ronald L., Brzozowski, David B., LaPorte, Thomas L., Patel, Ramesh N.
Published in ChemInform (16.09.2003)
Published in ChemInform (16.09.2003)
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Journal Article
PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 01.11.2007
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Year of Publication 01.11.2007
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Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester
GERARD A. CRISPINO, THOMAS L. LAPORTE, JALE MUSLEHIDDINOGLU, PAUL C. LOBBEN, DAVID K. LEAHY, MOURAD HAMEDI, CHIAJEN LAI, ROBERT P. DISCORDIA, ZHONGMIN XU, JOHN E. THORNTON, JAAN A. PESTI, LORI ANN SPANGLER
Year of Publication 01.11.2007
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Year of Publication 01.11.2007
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PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-F][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, LOBBEN, PAUL C, CRISPINO, GERARD A, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 01.11.2007
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Year of Publication 01.11.2007
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PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LEAHY DAVID K, LOBBEN PAUL C, THORNTON JOHN E, MUSLEHIDDINOGLU JALE, HAMEDI MOURAD, SPANGLER LORI A, XU ZHONGMIN, DISCORDIA ROBERT P, LAI CHIAJEN, CRISPINO GERARD A, PESTI JAAN A, LAPORTE THOMAS L
Year of Publication 25.10.2007
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Year of Publication 25.10.2007
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PROCESS FOR THE PREPARATION OF [(1R),2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO[2,1-f][1,2,4]TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LOBBEN PAUL, C, MUSLEHIDDINOGLU JALE, HAMEDI MOURAD, XU ZHONGMIN, LEAHY DAVID, K, LAI CHIAJEN, DISCORDIA ROBERT, P, LAPORTE THOMAS, L, CRISPINO GERARD, A, PESTI JAAN, A, THORNTON JOHN, E, SPANGLER LORI, ANN
Year of Publication 30.05.2014
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Year of Publication 30.05.2014
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CONTINUOUS PROCESS FOR PRODUCING HYDROXYAZAPIRONES BY OXIDATION
DEPUE, JEFFREY S, CHAN, YEUNG YU, LAPORTE, THOMAS L, WATSON, DANIEL J, DOWDY, ERIC D, SHEN, LIFEN, HAMEDI, MOURAD
Year of Publication 02.06.2005
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Year of Publication 02.06.2005
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Procedimiento de preparación del éster de 2-[4-(4-fluoro-2-metil-1H-indol-5-iloxi)-5-metilpirrolo]2,1-f-[1,2,4-triazin-6-iloxi]-1-metílico del ácido [(1R),2S]-2-aminopropiónico
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 01.04.2013
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Year of Publication 01.04.2013
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Fremgangsmåde til fremstilling af [(1R), 2S]-2-aminopropionsyre 2-[4-(4-fluor-2-methyl-1H-indol-5-yloxy)-5-methylpyrrol]2,1-f-[1,2,4-triazin-6-yloxy]-1-methylethylester
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 18.03.2013
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Year of Publication 18.03.2013
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