Biological Characterization of a Novel, Orally Active Small Molecule Gonadotropin-Releasing Hormone (GnRH) Antagonist Using Castrated and Intact Rats
Anderes, Kenna L, Luthin, David R, Castillo, Rosemary, Kraynov, Eugenia A, Castro, Mary, Nared-Hood, Karen, Gregory, Margaret L, Pathak, Ved P, Christie, Lance C, Paderes, Genevieve, Vazir, Haresh, Ye, Qiang, Anderson, Mark B, May, John M
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Journal Article
Electrophilic Tetraalkylammonium Nitrate Nitration. II. Improved Anhydrous Aromatic and Heteroaromatic Mononitration with Tetramethylammonium Nitrate and Triflic Anhydride, Including Selected Microwave Examples
Shackelford, Scott A, Anderson, Mark B, Christie, Lance C, Goetzen, Thomas, Guzman, Mark C, Hananel, Martha A, Kornreich, Wayne D, Li, Haitao, Pathak, Ved P, Rabinovich, Alex K, Rajapakse, Ranjan J, Truesdale, Larry K, Tsank, Stella M, Vazir, Haresh N
Published in Journal of organic chemistry (24.01.2003)
Published in Journal of organic chemistry (24.01.2003)
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Journal Article
Discovery of a Novel, Orally Active, Small Molecule Gonadotropin-Releasing Hormone (GnRH) Receptor Antagonist
Li, Haitao, Anderes, Kenna L, Kraynov, Eugenia A, Luthin, David R, Do, Quyen-Quyen, Hong, Yufeng, Tompkins, Eileen, Sun, Eric T, Rajapakse, Ranjan, Pathak, Ved P, Christie, Lance C, Vazir, Haresh, Castillo, Rosemary, Gregory, Margaret L, Castro, Mary, Nared-Hood, Karen, Paderes, Genevieve, Anderson, Mark B
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Journal Article
Pyridine-3-propanoic acids: Discovery of dual PPARα/γ agonists as antidiabetic agents
Humphries, Paul S., Bailey, Simon, Almaden, Jonathon V., Barnum, Sandra J., Carlson, Thomas J., Christie, Lance C., Do, Quyen-Quyen T., Fraser, James D., Hess, Mary, Kellum, Jack, Kim, Young H., McClellan, Guy A., Ogilvie, Kathleen M., Simmons, Brett H., Skalitzky, Donald, Sun, Shaoxian, Wilhite, David, Zehnder, Luke R.
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Journal Article
Discovery of a Novel, Orally Active, Small Molecule Gonadotropin-Releasing Hormone (GnRH) Receptor Antagonist
Li, Haitao, Anderes, Kenna L, Kraynov, Eugenia A, Luthin, David R, Do, Quyen-Quyen, Hong, Yufeng, Tompkins, Eileen, Sun, Eric T, Rajapakse, Ranjan, Pathak, Ved P, Christie, Lance C, Feng, Jun, Vazir, Haresh, Castillo, Rosemary, Gregory, Margaret L, Castro, Mary, Nared-Hood, Karen, Paderes, Genevieve, Anderson, Mark B
Published in Journal of medicinal chemistry (21.09.2006)
Published in Journal of medicinal chemistry (21.09.2006)
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Journal Article
Electrophilic Tetraalkylammonium Nitrate Nitration. II. Improved Anhydrous Aromatic and Heteroaromatic Mononitration with Tetramethylammonium Nitrate and Triflic Anhydride, Including Selected Microwave Examples
Shackelford, Scott A, Anderson, Mark B, Christie, Lance C, Goetzen, Thomas, Guzman, Mark C, Hananel, Martha A, Kornreich, Wayne D, Li, Haitao, Pathak, Ved P, Rabinovich, Alex K, Rajapakse, Ranjan J, Truesdale, Larry K, Tsank, Stella M, Vazir, Haresh N
Published in Journal of organic chemistry (04.04.2003)
Published in Journal of organic chemistry (04.04.2003)
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Journal Article
Pyridine-3-propanoic acids: Discovery of dual PPARalpha/gamma agonists as antidiabetic agents
Humphries, Paul S, Bailey, Simon, Almaden, Jonathon V, Barnum, Sandra J, Carlson, Thomas J, Christie, Lance C, Do, Quyen-Quyen T, Fraser, James D, Hess, Mary, Kellum, Jack, Kim, Young H, McClellan, Guy A, Ogilvie, Kathleen M, Simmons, Brett H, Skalitzky, Donald, Sun, Shaoxian, Wilhite, David, Zehnder, Luke R
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Journal Article
Effect of testosterone suppression on the pharmacokinetics of a potent GnRH receptor antagonist
IATSIMIRSKAIA, Eugenia A, GREGORY, Margaret L, MAY, John M, ANDERES, Kenna L, CASTILLO, Rosemary, MILGRAM, K. Eric, LUTHIN, David R, PATHAK, Ved P, CHRISTIE, Lance C, VAZIR, Haresh, ANDERSON, Mark B
Published in Pharmaceutical research (01.02.2002)
Published in Pharmaceutical research (01.02.2002)
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Journal Article
NICHT-PEPTIDISCHE VERBINDUNGEN, WELCHE DIE WIRKUNG DES GONADOTROPIN-FREISETZENDEN HORMONS (GNRH) BEEINFLUSSEN
VAZIR, HARESH N, HONG, YUFENG, PATHAK,VED P, RAJAPAKSE,RANJAN, ANDERSON, MARK B, TOMPKINS, EILEEN, FENG, JUN, LI, HAITAO, CHRISTIE, LANCE C
Year of Publication 15.05.2006
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Year of Publication 15.05.2006
Patent
Non-peptide compounds affecting the action of gonadotropin-releasing hormone (GnRH)
VAZIR, HARESH N, HONG, YUFENG, PATHAK,VED P, RAJAPAKSE,RANJAN, ANDERSON, MARK B, TOMPKINS, EILEEN, FENG, JUN, LI, HAITAO, CHRISTIE, LANCE C
Year of Publication 19.04.2006
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Year of Publication 19.04.2006
Patent
Non-peptide GnRH agents, Pharmaceutical compositions, and methods for their use
Christie, Lance C, Anderson, Mark B, Feng, Jun, Hong, Yufeng, Pathak, Ved P, Rajapakse, Ranjan J, Tompkins, Eileen V, Vazir, Haresh, Li, Haitao
Year of Publication 21.12.2004
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Year of Publication 21.12.2004
Patent
Non-peptide GnRH agents, Pharmaceutical compositions, and methods for their use
RAJAPAKSE RANJAN J, PATHAK VED P, ANDERSON MARK B, FENG JUN, LI HAITAO, TOMPKINS EILEEN V, VAZIR HARESH, HONG YUFENG, CHRISTIE LANCE C
Year of Publication 21.12.2004
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Year of Publication 21.12.2004
Patent
Non-peptide GnRH agents, pharmaceutical compositions, and methods for their use
RAJAPAKSE RANJAN J, PATHAK VED P, ANDERSON MARK B, FENG JUN, LI HAITAO, TOMPKINS EILEEN V, VAZIR HARESH, HONG YUFENG, CHRISTIE LANCE C
Year of Publication 18.03.2004
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Year of Publication 18.03.2004
Patent
Non-peptide GnRH agents, pharmaceutical compositions and methods for their use
RAJAPAKSE RANJAN J, SUN ERIC T, PATHAK VED P, ANDERSON MARK B, FENG JUN, LI HAITAO, TOMPKINS EILEEN V, DO QUYEN-QUYEN T, HONG YUFENG, CHRISTIE LANCE C
Year of Publication 10.11.2005
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Year of Publication 10.11.2005
Patent
Non-peptide compounds affecting the action of gonadotropin-releasing hormone (GnRH)
VAZIR, HARESH N, HONG, YUFENG, PATHAK,VED P, RAJAPAKSE,RANJAN, ANDERSON, MARK B, TOMPKINS, EILEEN, FENG, JUN, LI, HAITAO, CHRISTIE, LANCE C
Year of Publication 13.08.2003
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Year of Publication 13.08.2003
Patent
NON-PEPTIDE GnRH AGENTS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR THEIR USES, AND PROCESSES FOR PREPARING THEM
TOMPKINS, EILEEN, VALENZUELA, SUN, ERIC, T, CHRISTIE, LANCE, C, PADERES, GENEVIEVE, D, IATSIMIRSKAIA, EUGENIA, A, PATHAK, VED, P, FENG, JUN, RAJAPAKSE, RANJAN, JAGATH, LUTHIN, DAVID, R, HONG, YUFENG, SHACKELFORD, SCOTT, VAZIR, HARESH, ANDERES, KENNA, L, ANDERSON, MARK, B, LI, HAITAO, DO, QUYEN-QUYEN, T, GOETZEN, THOMAS, TRUESDALE, LARRY, K
Year of Publication 20.03.2003
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Year of Publication 20.03.2003
Patent
Non-peptide gnrh agents, pharmaceutical compositions and methods for their uses, and processes for preparing them
DAVID R. LUTHIN, HAITAO LI, VED P. PATHAK, HARESH VAZIR, SCOTT SHACKELFORD, QUYEN-QUYEN T. DO, GENEVIEVE D. PADERES, THOMAS GOETZEN, RANJAN JAGATH RAJAPAKSE, ERIC T. SUN, LARRY K. TRUESDALE, JUN FENG, MARK B. ANDERSON, LANCE C. CHRISTIE, EILEEN VALENZUELA TOMPKINS, KENNA L. ANDERES, EUGENIA A. IATSIMIRSKAIA, YUFENG HONG
Year of Publication 16.12.2002
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Year of Publication 16.12.2002
Patent
NON-PEPTIDE GNRH AGENTS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR THEIR USE, AND PROCESSES FOR PREPARING THEM AND THEIR INTERMEDIATES
TOMPKINS, EILEEN, VALENZUELA, SUN, ERIC, T, CHRISTIE, LANCE, C, PADERES, GENEVIEVE, D, IATSIMIRSKAIA, EUGENIA, A, PATHAK, VED, P, FENG, JUN, RAJAPAKSE, RANJAN, JAGATH, LUTHIN, DAVID, R, HONG, YUFENG, SHACKELFORD, SCOTT, VAZIR, HARESH, ANDERES, KENNA, L, ANDERSON, MARK, B, LI, HAITAO, DO, QUYEN-QUYEN, T, GOETZEN, THOMAS, TRUESDALE, LARRY, K
Year of Publication 12.12.2002
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Year of Publication 12.12.2002
Patent
ZAT-ZAT GnRH NON-PEPTIDA, METODE-METODE DAN ZAT-ZAT ANTARA PEMBUATANNYA
DAVID R. LUTHIN, HARESH N. VAZIR, JAMES FAUST, VED P. PATHAK, GENEVIEVE DEGUZMAN PADERES, EILEEN VALENZUELA TOMPKINS, HAITO LI, MARK BARIAN ANDERSON, LANCE CH. CHRISTIE, YUFENG HONG
Year of Publication 16.08.2001
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Year of Publication 16.08.2001
Patent