Common activation mechanism of class A GPCRs
Zhou, Qingtong, Yang, Dehua, Wu, Meng, Guo, Yu, Guo, Wanjing, Zhong, Li, Cai, Xiaoqing, Dai, Antao, Jang, Wonjo, Shakhnovich, Eugene I, Liu, Zhi-Jie, Stevens, Raymond C, Lambert, Nevin A, Babu, M Madan, Wang, Ming-Wei, Zhao, Suwen
Published in eLife (19.12.2019)
Published in eLife (19.12.2019)
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Structure of formylpeptide receptor 2-Gi complex reveals insights into ligand recognition and signaling
Zhuang, Youwen, Liu, Heng, Edward Zhou, X., Kumar Verma, Ravi, de Waal, Parker W., Jang, Wonjo, Xu, Ting-Hai, Wang, Lei, Meng, Xing, Zhao, Gongpu, Kang, Yanyong, Melcher, Karsten, Fan, Hao, Lambert, Nevin A., Eric Xu, H., Zhang, Cheng
Published in Nature communications (14.02.2020)
Published in Nature communications (14.02.2020)
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Blockade of Dendritic Cell Development by Bacterial Fermentation Products Butyrate and Propionate through a Transporter (Slc5a8)-dependent Inhibition of Histone Deacetylases
Singh, Nagendra, Thangaraju, Muthusamy, Prasad, Puttur D., Martin, Pamela M., Lambert, Nevin A., Boettger, Thomas, Offermanns, Stefan, Ganapathy, Vadivel
Published in The Journal of biological chemistry (03.09.2010)
Published in The Journal of biological chemistry (03.09.2010)
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GPR109A Is a G-protein―Coupled Receptor for the Bacterial Fermentation Product Butyrate and Functions as a Tumor Suppressor in Colon
THANGARAJU, Muthusamy, CRESCI, Gail A, PRASAD, Puttur D, GANAPATHY, Vadivel, KEBIN LIU, ANANTH, Sudha, GNANAPRAKASAM, Jaya P, BROWNING, Darren D, MELLINGER, John D, SMITH, Sylvia B, DIGBY, Gregory J, LAMBERT, Nevin A
Published in Cancer research (Chicago, Ill.) (01.04.2009)
Published in Cancer research (Chicago, Ill.) (01.04.2009)
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Pathway selectivity in Frizzleds is achieved by conserved micro-switches defining pathway-determining, active conformations
Grätz, Lukas, Kowalski-Jahn, Maria, Scharf, Magdalena M, Kozielewicz, Pawel, Jahn, Michael, Bous, Julien, Lambert, Nevin A, Gloriam, David E, Schulte, Gunnar
Published in Nature communications (29.07.2023)
Published in Nature communications (29.07.2023)
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Agonist-selective recruitment of engineered protein probes and of GRK2 by opioid receptors in living cells
Stoeber, Miriam, Jullié, Damien, Li, Joy, Chakraborty, Soumen, Majumdar, Susruta, Lambert, Nevin A, Manglik, Aashish, von Zastrow, Mark
Published in eLife (25.02.2020)
Published in eLife (25.02.2020)
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A conserved molecular switch in Class F receptors regulates receptor activation and pathway selection
Wright, Shane C, Kozielewicz, Paweł, Kowalski-Jahn, Maria, Petersen, Julian, Bowin, Carl-Fredrik, Slodkowicz, Greg, Marti-Solano, Maria, Rodríguez, David, Hot, Belma, Okashah, Najeah, Strakova, Katerina, Valnohova, Jana, Babu, M Madan, Lambert, Nevin A, Carlsson, Jens, Schulte, Gunnar
Published in Nature communications (08.02.2019)
Published in Nature communications (08.02.2019)
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GLP-1R signaling neighborhoods associate with the susceptibility to adverse drug reactions of incretin mimetics
Wright, Shane C, Motso, Aikaterini, Koutsilieri, Stefania, Beusch, Christian M, Sabatier, Pierre, Berghella, Alessandro, Blondel-Tepaz, Élodie, Mangenot, Kimberley, Pittarokoilis, Ioannis, Sismanoglou, Despoina-Christina, Le Gouill, Christian, Olsen, Jesper V, Zubarev, Roman A, Lambert, Nevin A, Hauser, Alexander S, Bouvier, Michel, Lauschke, Volker M
Published in Nature communications (09.10.2023)
Published in Nature communications (09.10.2023)
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The c-terminus of GRK3 indicates rapid dissociation of G protein heterotrimers
Hollins, Bettye, Kuravi, Sudhakiranmayi, Digby, Gregory J., Lambert, Nevin A.
Published in Cellular signalling (01.06.2009)
Published in Cellular signalling (01.06.2009)
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A Non-Systemic Phosphodiesterase-5 Inhibitor Suppresses Colon Proliferation in Mice
Lee, Avelina, Lebedyeva, Iryna, Zhi, Wenbo, Senthil, Vani, Cheema, Herjot, Brands, Michael W, Bush, Weston, Lambert, Nevin A, Snipes, Madeline, Browning, Darren D
Published in International journal of molecular sciences (28.05.2023)
Published in International journal of molecular sciences (28.05.2023)
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Regulators of G-protein Signaling accelerate GPCR signaling kinetics and govern sensitivity solely by accelerating GTPase activity
Lambert, Nevin A, Johnston, Christopher A, Cappell, Steven D, Kuravi, Sudhakiranmayi, Kimple, Adam J, Willard, Francis S, Siderovski, David P
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (13.04.2010)
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Allosteric Modulation of M1 Muscarinic Acetylcholine Receptor Internalization and Subcellular Trafficking
Yeatman, Holly R., Lane, J. Robert, Choy, Kwok Ho Christopher, Lambert, Nevin A., Sexton, Patrick M., Christopoulos, Arthur, Canals, Meritxell
Published in The Journal of biological chemistry (30.05.2014)
Published in The Journal of biological chemistry (30.05.2014)
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