Total Syntheses of Ningalin A, Lamellarin O, Lukianol A, and Permethyl Storniamide A Utilizing Heterocyclic Azadiene Diels−Alder Reactions
Boger, Dale L, Boyce, Christopher W, Labroli, Marc A, Sehon, Clark A, Jin, Qing
Published in Journal of the American Chemical Society (13.01.1999)
Published in Journal of the American Chemical Society (13.01.1999)
Get full text
Journal Article
Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. IV. Discovery of 1-[(4,6-Dimethyl-5-pyrimidinyl)carbonyl]- 4-[4-{2-methoxy-1(R)-4-(trifluoromethyl)phenyl}ethyl-3(S)-methyl-1-piperazinyl]- 4-methylpiperidine (Sch-417690/Sch-D), a Potent, Highly Selective, and Orally Bioavailable CCR5 Antagonist
Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis, Labroli, Marc A, Xiao, Yushi, Steensma, Ruo W, Strizki, Julie M, Baroudy, Bahige M, Cox, Kathleen, Lachowicz, Jean, Varty, Geoffrey, Watkins, Robert
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
Get full text
Journal Article
Discovery of potent wall teichoic acid early stage inhibitors
Labroli, Marc A., Caldwell, John P., Yang, Christine, Lee, Sang Ho, Wang, Hao, Koseoglu, Sandra, Mann, Paul, Yang, Shu-Wei, Xiao, Jing, Garlisi, Charles G., Tan, Christopher, Roemer, Terry, Su, Jing
Published in Bioorganic & medicinal chemistry letters (15.08.2016)
Published in Bioorganic & medicinal chemistry letters (15.08.2016)
Get full text
Journal Article
The identification of novel 5′-amino gemcitabine analogs as potent RRM1 inhibitors
Labroli, Marc A., Dwyer, Michael P., Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Wyss, Daniel, McCoy, Mark, Barrett, Dianah, Davis, Nicole, Seghezzi, Wolfgang, Shanahan, Frances, Taricani, Lorena, Beaumont, Maribel, Malinao, Maria-Christina, Parry, David, Guzi, Timothy J.
Published in Bioorganic & medicinal chemistry (01.04.2014)
Published in Bioorganic & medicinal chemistry (01.04.2014)
Get full text
Journal Article
10-Formyl-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid (10-formyl-ddacthf) : A potent cytotoxic agent acting by selective inhibition of human GAR Tfase and the de novo purine biosynthetic pathway
MARSILJE, Thomas H, LABROLI, Marc A, WILSON, Ian A, BEARDSLEY, G. Peter, BENKOVIC, Stephen J, BOGER, Dale L, HEDRICK, Michael P, QING JIN, DESHARNAIS, Joel, BAKER, Stephen J, GOOLJARSINGH, Lata T, RAMCHARAN, Joseph, TAVASSOLI, Ali, YAN ZHANG
Published in Bioorganic & medicinal chemistry (01.08.2002)
Published in Bioorganic & medicinal chemistry (01.08.2002)
Get full text
Journal Article
A convergent preparation of the CHK1 inhibitor MK-8776 (SCH 900776)
Labroli, Marc A., Dwyer, Michael P., Poker, Cory, Keertikar, Kerry M., Rossman, Randall, Guzi, Timothy J.
Published in Tetrahedron letters (15.06.2016)
Published in Tetrahedron letters (15.06.2016)
Get full text
Journal Article
ChemInform Abstract: Syntheses of 5′-Amino-2′,5′-dideoxy-2′,2′-difluorocytidine Derivatives as Novel Anticancer Nucleoside Analogues
Labroli, Marc A., Dwyer, Michael P., Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Richard, Judson, Rosner, Kristen, Paruch, Kamil, Guzi, Timothy J.
Published in ChemInform (24.06.2014)
Published in ChemInform (24.06.2014)
Get full text
Journal Article
Syntheses of 5′-amino-2′,5′-dideoxy-2′,2′-difluorocytidine derivatives as novel anticancer nucleoside analogs
Labroli, Marc A., Dwyer, Michael P., Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Richard, Judson, Rosner, Kristen, Paruch, Kamil, Guzi, Timothy J.
Published in Tetrahedron letters (15.01.2014)
Published in Tetrahedron letters (15.01.2014)
Get full text
Journal Article
Syntheses of 5'-amino-2',5'-dideoxy-2',2'-dif luorocytidine derivatives as novel anticancer nucleoside analogs
Labroli, Marc A, Dwyer, Michael P, Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Richard, Judson, Rosner, Kristen, Paruch, Kamil, Guzi, Timothy J
Published in Tetrahedron letters (01.01.2014)
Published in Tetrahedron letters (01.01.2014)
Get full text
Journal Article
PYRAZOLOPYRIMIDINE DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPESVIRUSES
LABROLI, Marc, A, ARMACOST, Kira, A, CROWLEY, Brendan, M, COOKE, Andrew, J, SCHLEGEL, Kelly-Ann S, SHAW, Anthony, W, COX, Christopher Douglas, PLOTKIN, Michael, A, RAHEEM, Izzat, T
Year of Publication 23.10.2024
Get full text
Year of Publication 23.10.2024
Patent
AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
HAYES, Robert, Patrick, LABROLI, Marc, A, ARMACOST, Kira, A, SCHUBERT, Jeffrey, W, COOKE, Andrew, John, TELLERS, David, M, PLOTKIN, Michael, Aaron, RAHEEM, Izzat, Tiedje
Year of Publication 29.11.2023
Get full text
Year of Publication 29.11.2023
Patent
Piperazine-based CCR5 antagonists as HIV-1 inhibitors. IV. Discovery of 1-[(4,6-dimethyl-5-pyrimidinyl)carbonyl]- 4-[4-[2-methoxy-1(R)-4-(trifluoromethyl)phenyl]ethyl-3(S)-methyl-1-piperazinyl]- 4-methylpiperidine (Sch-417690/Sch-D), a potent, highly selective, and orally bioavailable CCR5 antagonist
Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis, Labroli, Marc A, Xiao, Yushi, Steensma, Ruo W, Strizki, Julie M, Baroudy, Bahige M, Cox, Kathleen, Lachowicz, Jean, Varty, Geoffrey, Watkins, Robert
Published in Journal of medicinal chemistry (06.05.2004)
Get full text
Published in Journal of medicinal chemistry (06.05.2004)
Journal Article
AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
Plotkin, Michael Aaron, Tellers, David M, Hayes, Robert Patrick, Armacost, Kira A, Cooke, Andrew John, Labroli, Marc A, Schubert, Jeffrey W, Raheem, Izzat Tiedje
Year of Publication 16.03.2023
Get full text
Year of Publication 16.03.2023
Patent
AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
HAYES, Robert, Patrick, LABROLI, Marc, A, ARMACOST, Kira, A, SCHUBERT, Jeffrey, W, COOKE, Andrew, John, TELLERS, David, M, PLOTKIN, Michael, Aaron, RAHEEM, Izzat, Tiedje
Year of Publication 26.10.2022
Get full text
Year of Publication 26.10.2022
Patent
OXAZOLIDINONES AS TARO INHIBITORS
DE JESUS, Reynalda, MANDAL, Mihir, LABROLI, Marc A, TANG, Haifeng, HA, Sookhee N, MADSEN-DUGGAN, Christina, LEE, Sang Ho, WANG, Hao, CALDWELL, John P, DING, Fa-Xiang, GILL, Charles J, TAN, Zheng, KOSEOGLU, Sandra, J, SU, Jing, TAN, Christopher Michael, YANG, Shu-Wei, HO, Ginny Dai, YANG, Christine, ROEMER, Terry
Year of Publication 13.12.2023
Get full text
Year of Publication 13.12.2023
Patent
INHIBITORS OF MSBA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
TONG, Ling, LABROLI, Marc A, ZHANG, Li-Kang, BALIBAR, Carl J, SKUDLAREK, Jason W, WANG, Hao, LIU, Jian, WU, Zhe, MITCHELL, Helen, BABAOGLU, Kerim, COOKE, Andrew J, FORSTER, Ashley, WU, Chengwei, RAHEEM, Izzat, BUEVICH, Alexei, SHAW, Anthony W
Year of Publication 23.11.2023
Get full text
Year of Publication 23.11.2023
Patent