A Reversible and Selective Inhibitor of Monoacylglycerol Lipase Ameliorates Multiple Sclerosis
Hernández-Torres, Gloria, Cipriano, Mariateresa, Hedén, Erika, Björklund, Emmelie, Canales, Ángeles, Zian, Debora, Feliú, Ana, Mecha, Miriam, Guaza, Carmen, Fowler, Christopher J., Ortega-Gutiérrez, Silvia, López-Rodríguez, María L.
Published in Angewandte Chemie (International ed.) (08.12.2014)
Published in Angewandte Chemie (International ed.) (08.12.2014)
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Monoacylglycerol lipase (MAGL) as a promising therapeutic target
Gil-Ordóñez, Ana, Martín-Fontecha, Mar, Ortega-Gutiérrez, Silvia, López-Rodríguez, María L.
Published in Biochemical pharmacology (01.11.2018)
Published in Biochemical pharmacology (01.11.2018)
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Journal Article
Blocking Ras inhibition as an antitumor strategy
Marín-Ramos, Nagore I., Ortega-Gutiérrez, Silvia, López-Rodríguez, María L.
Published in Seminars in cancer biology (01.02.2019)
Published in Seminars in cancer biology (01.02.2019)
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Journal Article
2‐AG limits Theiler's virus induced acute neuroinflammation by modulating microglia and promoting MDSCs
Mecha, Miriam, Feliú, Ana, Machín, Isabel, Cordero, Cesar, Carrillo‐Salinas, Francisco, Mestre, Leyre, Hernández‐Torres, Gloria, Ortega‐Gutiérrez, Silvia, López‐Rodríguez, María L, de Castro, Fernando, Clemente, Diego, Guaza, Carmen
Published in Glia (01.07.2018)
Published in Glia (01.07.2018)
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A Potent Isoprenylcysteine Carboxylmethyltransferase (ICMT) Inhibitor Improves Survival in Ras-Driven Acute Myeloid Leukemia
Marín-Ramos, Nagore I, Balabasquer, Moisés, Ortega-Nogales, Francisco J, Torrecillas, Iván R, Gil-Ordóñez, Ana, Marcos-Ramiro, Beatriz, Aguilar-Garrido, Pedro, Cushman, Ian, Romero, Antonio, Medrano, Francisco J, Gajate, Consuelo, Mollinedo, Faustino, Philips, Mark R, Campillo, Mercedes, Gallardo, Miguel, Martín-Fontecha, Mar, López-Rodríguez, María L, Ortega-Gutiérrez, Silvia
Published in Journal of medicinal chemistry (11.07.2019)
Published in Journal of medicinal chemistry (11.07.2019)
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Journal Article
Novel Antagonist of the Type 2 Lysophosphatidic Acid Receptor (LPA2), UCM-14216, Ameliorates Spinal Cord Injury in Mice
Khiar-Fernández, Nora, Zian, Debora, Vázquez-Villa, Henar, Martínez, R. Fernando, Escobar-Peña, Andrea, Foronda-Sainz, Román, Ray, Manisha, Puigdomenech-Poch, Maria, Cincilla, Giovanni, Sánchez-Martínez, Melchor, Kihara, Yasuyuki, Chun, Jerold, López-Vales, Rubèn, López-Rodríguez, María L., Ortega-Gutiérrez, Silvia
Published in Journal of medicinal chemistry (25.08.2022)
Published in Journal of medicinal chemistry (25.08.2022)
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Targeting the FtsZ Allosteric Binding Site with a Novel Fluorescence Polarization Screen, Cytological and Structural Approaches for Antibacterial Discovery
Huecas, Sonia, Araújo-Bazán, Lidia, Ruiz, Federico M, Ruiz-Ávila, Laura B, Martínez, R. Fernando, Escobar-Peña, Andrea, Artola, Marta, Vázquez-Villa, Henar, Martín-Fontecha, Mar, Fernández-Tornero, Carlos, López-Rodríguez, María L, Andreu, José M
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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A Positive Allosteric Modulator of the Serotonin 5‑HT2C Receptor for Obesity
García-Cárceles, Javier, Decara, Juan M., Vázquez-Villa, Henar, Rodríguez, Ramón, Codesido, Eva, Cruces, Jacobo, Brea, José, Loza, María I., Alén, Francisco, Botta, Joaquin, McCormick, Peter J., Ballesteros, Juan A., Benhamú, Bellinda, Rodríguez de Fonseca, Fernando, López-Rodríguez, María L.
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Journal Article
Discovery of V‑0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide‑1 Receptor toward Oral Treatment for “Diabesity”
Decara, Juan M, Vázquez-Villa, Henar, Brea, José, Alonso, Mónica, Srivastava, Raj Kamal, Orio, Laura, Alén, Francisco, Suárez, Juan, Baixeras, Elena, García-Cárceles, Javier, Escobar-Peña, Andrea, Lutz, Beat, Rodríguez, Ramón, Codesido, Eva, Garcia-Ladona, F. Javier, Bennett, Teresa A, Ballesteros, Juan A, Cruces, Jacobo, Loza, María I, Benhamú, Bellinda, Rodríguez de Fonseca, Fernando, López-Rodríguez, María L
Published in Journal of medicinal chemistry (14.04.2022)
Published in Journal of medicinal chemistry (14.04.2022)
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Chemical Probes for the Recognition of Cannabinoid Receptors in Native Systems
Martín-Couce, Lidia, Martín-Fontecha, Mar, Palomares, Óscar, Mestre, Leyre, Cordomí, Arnau, Hernangomez, Miriam, Palma, Sara, Pardo, Leonardo, Guaza, Carmen, López-Rodríguez, María L., Ortega-Gutiérrez, Silvia
Published in Angewandte Chemie (International ed.) (09.07.2012)
Published in Angewandte Chemie (International ed.) (09.07.2012)
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2‑(Fluoromethoxy)-4′‑(S‑methanesulfonimidoyl)-1,1′-biphenyl (UCM-1306), an Orally Bioavailable Positive Allosteric Modulator of the Human Dopamine D1 Receptor for Parkinson’s Disease
García-Cárceles, Javier, Vázquez-Villa, Henar, Brea, José, Ladron de Guevara-Miranda, David, Cincilla, Giovanni, Sánchez-Martínez, Melchor, Sánchez-Merino, Anabel, Algar, Sergio, Teresa de los Frailes, María, Roberts, Richard S., Ballesteros, Juan A., Rodríguez de Fonseca, Fernando, Benhamú, Bellinda, Loza, María I., López-Rodríguez, María L.
Published in Journal of medicinal chemistry (22.09.2022)
Published in Journal of medicinal chemistry (22.09.2022)
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Journal Article
Development of a Nucleotide Exchange Inhibitor That Impairs Ras Oncogenic Signaling
Marín‐Ramos, Nagore I., Piñar, Carmen, Vázquez‐Villa, Henar, Martín‐Fontecha, Mar, González, Ángel, Canales, Ángeles, Algar, Sergio, Mayo, Paloma P., Jiménez‐Barbero, Jesús, Gajate, Consuelo, Mollinedo, Faustino, Pardo, Leonardo, Ortega‐Gutiérrez, Silvia, Viso, Alma, López‐Rodríguez, María L.
Published in Chemistry : a European journal (31.01.2017)
Published in Chemistry : a European journal (31.01.2017)
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Journal Article
Chemoproteomic Approach to Explore the Target Profile of GPCR ligands: Application to 5-HT1A and 5-HT6 Receptors
Gamo, Ana M., González-Vera, Juan A., Rueda-Zubiaurre, Ainoa, Alonso, Dulce, Vázquez-Villa, Henar, Martín-Couce, Lidia, Palomares, Óscar, López, Juan A., Martín-Fontecha, Mar, Benhamú, Bellinda, López-Rodríguez, María L., Ortega-Gutiérrez, Silvia
Published in Chemistry : a European journal (22.01.2016)
Published in Chemistry : a European journal (22.01.2016)
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Journal Article
Isoprenylcysteine Carboxylmethyltransferase-Based Therapy for Hutchinson–Gilford Progeria Syndrome
Marcos-Ramiro, Beatriz, Gil-Ordóñez, Ana, Marín-Ramos, Nagore I, Ortega-Nogales, Francisco J, Balabasquer, Moisés, Gonzalo, Pilar, Khiar-Fernández, Nora, Rolas, Loïc, Barkaway, Anna, Nourshargh, Sussan, Andrés, Vicente, Martín-Fontecha, Mar, López-Rodríguez, María L, Ortega-Gutiérrez, Silvia
Published in ACS central science (25.08.2021)
Published in ACS central science (25.08.2021)
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Journal Article
New Synthetic Inhibitors of Fatty Acid Synthase with Anticancer Activity
Turrado, Carlos, Puig, Teresa, García-Cárceles, Javier, Artola, Marta, Benhamú, Bellinda, Ortega-Gutiérrez, Silvia, Relat, Joana, Oliveras, Gloria, Blancafort, Adriana, Haro, Diego, Marrero, Pedro F, Colomer, Ramón, López-Rodríguez, María L
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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The structural assembly switch of cell division protein FtsZ probed with fluorescent allosteric inhibitors
Artola, Marta, Ruiz-Avila, Laura B., Ramirez-Aportela, Erney, Fernando Martinez, R., Araujo-Bazan, Lidia, Vazquez-Villa, Henar, Martin-Fontecha, Mar, Oliva, Maria A., Javier Martin-Galiano, A., Chacon, Pablo, Lopez-Rodriguez, Maria L., Andreu, Jose M., Huecas, Sonia
Published in Chemical science (Cambridge) (01.02.2017)
Published in Chemical science (Cambridge) (01.02.2017)
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Journal Article
Benzimidazole Derivatives as New Serotonin 5-HT6 Receptor Antagonists. Molecular Mechanisms of Receptor Inactivation
de la Fuente, Tania, Martín-Fontecha, Mar, Sallander, Jessica, Benhamú, Bellinda, Campillo, Mercedes, Medina, Rocío A, Pellissier, Lucie P, Claeysen, Sylvie, Dumuis, Aline, Pardo, Leonardo, López-Rodríguez, María L
Published in Journal of medicinal chemistry (11.02.2010)
Published in Journal of medicinal chemistry (11.02.2010)
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Journal Article
Synthetic Inhibitors of Bacterial Cell Division Targeting the GTP-Binding Site of FtsZ
Ruiz-Avila, Laura B, Huecas, Sonia, Artola, Marta, Vergoñós, Albert, Ramírez-Aportela, Erney, Cercenado, Emilia, Barasoain, Isabel, Vázquez-Villa, Henar, Martín-Fontecha, Mar, Chacón, Pablo, López-Rodrı́guez, María L, Andreu, José M
Published in ACS chemical biology (20.09.2013)
Published in ACS chemical biology (20.09.2013)
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Journal Article
Synthesis of New Serotonin 5-HT7 Receptor Ligands. Determinants of 5-HT7/5-HT1A Receptor Selectivity
Medina, Rocío A, Sallander, Jessica, Benhamú, Bellinda, Porras, Esther, Campillo, Mercedes, Pardo, Leonardo, López-Rodríguez, María L
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Journal Article
New Serotonin 5‑HT1A Receptor Agonists Endowed with Antinociceptive Activity in Vivo
Valhondo, Margarita, Marco, Isabel, Martín-Fontecha, Mar, Vázquez-Villa, Henar, Ramos, José A, Berkels, Reinhard, Lauterbach, Thomas, Benhamú, Bellinda, López-Rodríguez, María L
Published in Journal of medicinal chemistry (24.10.2013)
Published in Journal of medicinal chemistry (24.10.2013)
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