Search Results - "Lépissier, Luce" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

by Terrett, Jack A, Chen, Huifen, Shore, Daniel G, Villemure, Elisia, Larouche-Gauthier, Robin, Déry, Martin, Beaumier, Francis, Constantineau-Forget, Léa, Grand-Maître, Chantal, Lépissier, Luce, Ciblat, Stéphane, Sturino, Claudio, Chen, Yong, Hu, Baihua, Lu, Aijun, Wang, Yunli, Cridland, Andrew P, Ward, Stuart I, Hackos, David H, Reese, Rebecca M, Shields, Shannon D, Chen, Jun, Balestrini, Alessia, Riol-Blanco, Lorena, Lee, Wyne P, Liu, John, Suto, Eric, Wu, Xiumin, Zhang, Juan, Ly, Justin Q, La, Hank, Johnson, Kevin, Baumgardner, Matt, Chou, Kang-Jye, Rohou, Alexis, Rougé, Lionel, Safina, Brian S, Magnuson, Steven, Volgraf, Matthew
Published in Journal of medicinal chemistry (08.04.2021)

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Journal Article

Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

by Terrett, Jack A., Ly, Justin Q., Katavolos, Paula, Hasselgren, Catrin, Laing, Steven, Zhong, Fiona, Villemure, Elisia, Déry, Martin, Larouche-Gauthier, Robin, Chen, Huifen, Shore, Daniel G., Lee, Wyne P., Suto, Eric, Johnson, Kevin, Brooks, Marjory, Stablein, Alyssa, Beaumier, Francis, Constantineau-Forget, Léa, Grand-Maître, Chantal, Lépissier, Luce, Ciblat, Stéphane, Sturino, Claudio, Chen, Yong, Hu, Baihua, Elstrott, Justin, Gandham, Vineela, Joseph, Victory, Booler, Helen, Cain, Gary, Chou, Carolina, Fullerton, Aaron, Lepherd, Michelle, Stainton, Shannon, Torres, Elizabeth, Urban, Konnie, Yu, Lanlan, Zhong, Yu, Bao, Linda, Chou, Kang-Jye, Lin, Jessica, Zhang, Wei, La, Hank, Liu, Liling, Mulder, Teresa, Chen, Jun, Chernov-Rogan, Tania, Johnson, Adam R., Hackos, David H., Leahey, Rebecca, Shields, Shannon D., Balestrini, Alessia, Riol-Blanco, Lorena, Safina, Brian S., Volgraf, Matthew, Magnuson, Steven, Kakiuchi-Kiyota, Satoko
Published in Journal of medicinal chemistry (14.03.2024)

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Journal Article

Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2‑a]pyridine Series of Autotaxin Inhibitors

Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2‑a]pyridine Series of Autotaxin Inhibitors

by Joncour, Agnès, Desroy, Nicolas, Housseman, Christopher, Bock, Xavier, Bienvenu, Natacha, Cherel, Laëtitia, Labeguere, Virginie, Peixoto, Christophe, Annoot, Denis, Lepissier, Luce, Heiermann, Jörg, Hengeveld, Willem Jan, Pilzak, Gregor, Monjardet, Alain, Wakselman, Emanuelle, Roncoroni, Veronique, Le Tallec, Sandrine, Galien, René, David, Christelle, Vandervoort, Nele, Christophe, Thierry, Conrath, Katja, Jans, Mia, Wohlkonig, Alexandre, Soror, Sameh, Steyaert, Jan, Touitou, Robert, Fleury, Damien, Vercheval, Lionel, Mollat, Patrick, Triballeau, Nicolas, van der Aar, Ellen, Brys, Reginald, Heckmann, Bertrand
Published in Journal of medicinal chemistry (14.09.2017)

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Journal Article

Correction to Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2‑a]pyridine Series of Autotaxin Inhibitors

Correction to Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2‑a]pyridine Series of Autotaxin Inhibitors

by Joncour, Agnès, Desroy, Nicolas, Housseman, Christopher, Bock, Xavier, Bienvenu, Natacha, Cherel, Laëtitia, Labeguere, Virginie, Peixoto, Christophe, Annoot, Denis, Lepissier, Luce, Heiermann, Jörg, Hengeveld, Willem Jan, Pilzak, Gregor, Monjardet, Alain, Wakselman, Emanuelle, Roncoroni, Veronique, Le Tallec, Sandrine, Galien, René, David, Christelle, Vandervoort, Nele, Christophe, Thierry, Conrath, Katja, Jans, Mia, Wohlkonig, Alexandre, Soror, Sameh, Steyaert, Jan, Touitou, Robert, Fleury, Damien, Vercheval, Lionel, Mollat, Patrick, Triballeau, Nicolas, van der Aar, Ellen, Brys, Reginald, Heckmann, Bertrand
Published in Journal of medicinal chemistry (10.05.2018)

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Journal Article

Compounds for the modulation of Myc activity

Compounds for the modulation of Myc activity

by Sow, Boubacar, Beaumier, Francis, Marineau, Jason J, Berstler, Lauren, Lépissier, Luce, Rahl, Peter B, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 12.09.2023

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Patent

FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY

FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY

by DELIGNY, Michaël Louis Robert, KEYAERTS, Jean, LÉPISSIER, Luce Elsa, HEER, Jag Paul, LOWE, Martin Alexander
Year of Publication 18.08.2021

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Patent

Oxadiazole transient receptor potential channel inhibitors

Oxadiazole transient receptor potential channel inhibitors

by Chen, Huifen, Déry, Martin, Volgraf, Matthew, Sturino, Claudio, Beaumier, Francis, Villemure, Elisia, Lépissier, Luce, Constantineau-Forget, Lea, Larouche-Gauthier, Robin, Grand-Maître, Chantal, Terrett, Jack Alexander
Year of Publication 23.05.2023

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Patent

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

by Sow, Boubacar, Beaumier, Francis, Marineau, Jason J, Berstler, Lauren, Lépissier, Luce, Rahl, Peter B, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 11.05.2023

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Patent

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

by VILLEMURE, Elisia, CHEN, Huifen, TERRETT, Jack Alexander, Larouche-Gauthier, Robin, BEAUMIER, Francis, VOLGRAF, Matthew, CONSTANTINEAU-FORGET, Lea, GRAND-MAÎTRE, Chantal, LÉPISSIER, Luce, DÉRY, Martin, STURINO, Claudio
Year of Publication 20.04.2023

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Patent

Compounds for the modulation of MYC activity

Compounds for the modulation of MYC activity

by Beaumier, Francis, Sow, Boubacar, Rahi, Peter B, Marineau, Jason J, Lépissier, Luce, Berstler, Lauren, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 15.03.2022

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Patent

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

by Sow, Boubacar, Beaumier, Francis, Marineau, Jason J, Berstler, Lauren, Lépissier, Luce, Rahl, Peter B, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 17.02.2022

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Patent

Compounds for the modulation of Myc activity

Compounds for the modulation of Myc activity

by Sow, Boubacar, Beaumier, Francis, Marineau, Jason J, Berstler, Lauren, Lépissier, Luce, Rahl, Peter B, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 21.09.2021

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Patent

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

by Beaumier, Francis, Sow, Boubacar, Marineau, Jason J, Lépissier, Luce, Berstler, Lauren, Zhang, Yi, Rahl, Peter B, Larouche-Gauther, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 22.07.2021

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Patent

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

COMPOUNDS FOR THE MODULATION OF MYC ACTIVITY

by Sow, Boubacar, Beaumier, Francis, Marineau, Jason J, Berstler, Lauren, Lépissier, Luce, Rahl, Peter B, Zhang, Yi, Larouche-Gauthier, Robin, Sprott, Kevin, Ciblat, Stephane, Roberts, Christopher
Year of Publication 24.06.2021

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Patent

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

by VILLEMURE, Elisia, CHEN, Huifen, LAROUCHE-GAUTHIER, Robin, TERRETT, Jack Alexander, BEAUMIER, Francis, VOLGRAF, Matthew, CONSTANTINEAU-FORGET, Lea, GRAND-MAÎTRE, Chantal, LÉPISSIER, Luce, DÉRY, Martin, STURINO, Claudio
Year of Publication 27.01.2021

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Patent

INHIBITEURS DE CANAL À POTENTIEL DE RÉCEPTEUR TRANSITOIRE À BASE D'OXADIAZOLE

INHIBITEURS DE CANAL À POTENTIEL DE RÉCEPTEUR TRANSITOIRE À BASE D'OXADIAZOLE

by VILLEMURE, Elisia, CHEN, Huifen, LAROUCHE-GAUTHIER, Robin, TERRETT, Jack Alexander, BEAUMIER, Francis, VOLGRAF, Matthew, CONSTANTINEAU-FORGET, Lea, GRAND-MAÎTRE, Chantal, LÉPISSIER, Luce, DÉRY, Martin, STURINO, Claudio
Year of Publication 27.01.2021

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Patent

FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY

FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY

by DELIGNY, Michaël Louis Robert, KEYAERTS, Jean, LÉPISSIER, Luce Elsa, HEER, Jag Paul, LOWE, Martin Alexander
Year of Publication 06.02.2019

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Patent

Inhibidores de canal de potencial de receptor transitorio de oxadiazol

Inhibidores de canal de potencial de receptor transitorio de oxadiazol

by VILLEMURE, Elisia, CHEN, Huifen, LAROUCHE-GAUTHIER, Robin, TERRETT, Jack Alexander, VOLGRAF, Matthew, BEAUMIER, Francis, CONSTANTINEAU-FORGET, Lea, GRAND-MAÎTRE, Chantal, LÉPISSIER, Luce, DÉRY, Martin, STURINO, Claudio
Year of Publication 18.12.2020

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Patent

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

by VILLEMURE, Elisia, CHEN, Huifen, LAROUCHE-GAUTHIER, Robin, TERRETT, Jack Alexander, BEAUMIER, Francis, VOLGRAF, Matthew, CONSTANTINEAU-FORGET, Lea, GRAND-MAÎTRE, Chantal, LÉPISSIER, Luce, DÉRY, Martin, STURINO, Claudio
Year of Publication 29.10.2020

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Patent

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS

by Chen, Huifen, Déry, Martin, Volgraf, Matthew, Sturino, Claudio, Beaumier, Francis, Villemure, Elisia, Lépissier, Luce, Constantineau-Forget, Lea, Larouche-Gauthier, Robin, Grand-Maître, Chantal, Terrett, Jack Alexander
Year of Publication 01.10.2020

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Patent