Stereoselective Mukaiyama-Michael/Michael/Aldol Domino Cyclization as the Key Step in the Synthesis of Pentasubstituted Arenes: An Efficient Access to Highly Active Inhibitors of Cholesteryl Ester Transfer Protein (CETP)
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Published in Angewandte Chemie International Edition (15.11.1999)
Published in Angewandte Chemie International Edition (15.11.1999)
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Fluorine-substitution in cholesteryl ester transfer protein inhibitors (CETP-inhibitors) - Biology, chemistry, SAR, and properties
Paulsen, H, Schmeck, C, Brandes, A, Schmidt, G, Stoltefuss, J, Wirtz, SN, Logers, M, Naab, P, Bremm, KD, Bischoff, H, Schmidt, D, Zaiss, S, Antons, S
Published in Chimia (01.03.2004)
Published in Chimia (01.03.2004)
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CRYSTALLINE FORM OF 2-CHLORO-N-CYCLOPROPYL-5-[1-[2,6-DICHLORO-4-[1,2,2,2-TETRAFLUORO-1- (TRIFLUOROMETHYL)ETHYL]PHENYL]PYRAZOL-4-YL]-N-METHYL-PYRIDINE-3-CARBOXAMIDE
OLENIK, Britta, REMBIAK, Andreas, KEIL, Birgit, DOCKNER, Michael, LÖGERS, Michael, MEHL, Benedikt
Year of Publication 25.05.2022
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Year of Publication 25.05.2022
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Mannich Biscyclizations. Total Synthesis of (-)-Ajmalicine
Loegers, Michael, Overman, Larry E, Welmaker, Gregory S
Published in Journal of the American Chemical Society (01.09.1995)
Published in Journal of the American Chemical Society (01.09.1995)
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PROCESS FOR THE PREPARATION OF 4- {4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE,ITS SALTS AND MONOHYDRATE
JOACHIM REHSE, SASKIA WICHMANN, JÜERGEN STIEHL, WERNER HEILMANN, MICHAEL GOTTFRIED, MICHAEL LÖGERS
Year of Publication 15.06.2017
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Year of Publication 15.06.2017
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Process for the preparation of 4-{4-[({[4 chloro-3-(trifluoromethyl)-phenyl]amino}carbonyl)amino]-3-fluorphenoxy-N-ethylpyridie-carboxamide, its salts and monohydrate
Rehse Joachim, Gottfried Michael, Heilmann Werner, Stiehl Juergen, Lögers Michael, Wichmann Saskia
Year of Publication 04.10.2016
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Year of Publication 04.10.2016
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PROCESS FOR THE PREPARATION OF 4-{4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
LÖGERS, MICHAEL, STIEHL, JUERGEN, REHSE, JOACHIM, WICHMANN, SASKIA, HEILMANN, WERNER, GOTTFRIED, MICHAEL
Year of Publication 30.10.2015
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Year of Publication 30.10.2015
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PROCESS FOR THE PREPARATION OF 4- {4-[({[4 -CHLORO-3 -(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
LÖGERS, MICHAEL, REHSE, JOACHIM, STIEHL, JÜRGEN, WICHMANN, SASKIA, HEILMANN, WERNER, GOTTFRIED, MICHAEL
Year of Publication 09.10.2015
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Year of Publication 09.10.2015
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PROCESS FOR THE PREPARATION OF 4-{4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
JUERGEN STIEHL, JOACHIM REHSE, SASKIA WICHMANN, WERNER HEILMANN, MICHAEL GOTTFRIED, MICHAEL LÖGERS
Year of Publication 01.09.2015
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Year of Publication 01.09.2015
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PROCESS FOR THE PREPARATION OF 4-{4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
LÖGERS, MICHAEL, STIEHL, JUERGEN, REHSE, JOACHIM, WICHMANN, SASKIA, HEILMANN, WERNER, GOTTFRIED, MICHAEL
Year of Publication 20.05.2015
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Year of Publication 20.05.2015
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PROCESS FOR THE PREPARATION OF 4- {4-[({[4 -CHLORO-3 -(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
LÖGERS, MICHAEL, STIEHL, JUERGEN, REHSE, JOACHIM, WICHMANN, SASKIA, HEILMANN, WERNER, GOTTFRIED, MICHAEL
Year of Publication 29.04.2015
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Year of Publication 29.04.2015
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Processo para a preparação de 4-{4-[({[4-cloro-3-(trifluorometil)fe-nil]amino}carbonil)amino]fenóxi}nmetilpiridina-2-carboxamida
MATTHÄUS MIKE, KUHN OLIVER, GEHRING REINHOLD, BERWE MATHIAS, LENZ JANA, HEILMANN WERNER, MOHRS KLAUS, STIEHL JÜRGEN, LÖGERS MICHAEL, MÜLLER-GLIEMANN MATTHIAS
Year of Publication 09.11.2021
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Year of Publication 09.11.2021
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Prodrugs of the cytostatic CC-1065 that can be activated in a tumor-selective manner
Tietze, LF, Hannemann, R, Buhr, W, Logers, M, Menningen, P, Lieb, M, Starck, D, Grote, T, Doring, A, Schubert
Published in Angewandte Chemie International Edition (01.12.1996)
Published in Angewandte Chemie International Edition (01.12.1996)
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Process for the preparation of 4-{4[({[4-chloro-3-(trifluoromethyl)-phenyl]amino}carbonyl)amino]-3-fluorophenoxy}-N-methylpyridine-2-carboxamide, its salts and monohydrate
HEILMANN WERNER, REHSE JOACHIM, STIEHL JUERGEN, GOTTFRIED MICHAEL, LÖGERS MICHAEL, WICHMANN SASKIA
Year of Publication 10.06.2014
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Year of Publication 10.06.2014
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