Correction to Discovery of the Hemifumarate and (α‑l‑Alanyloxy)methyl Ether as Prodrugs of an Antirheumatic Oxindole: Prodrugs for the Enolic OH Group
Robinson, Ralph P, Reiter, Lawrence A, Barth, Wayne E, Campeta, Anthony M, Cooper, Kelvin, Cronin, Brian J, Destito, Rosalina, Donahue, Kathleen M, Falkner, Fred C, Fiese, Eugene F, Johnson, Diane L, Kuperman, Alexander V, Liston, Theodore E, Malloy, Deborah, Martin, John J, Mitchell, David Y, Rusek, Frank W, Shamblin, Sheri L, Wright, Charles F
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Pharmacokinetics and Metabolism of a Cysteinyl Leukotriene-1 Receptor Antagonist from the Heterocyclic Chromanol Series in Rats: In Vitro-In Vivo Correlation, Gender-Related Differences, Isoform Identification, and Comparison with Metabolism in Human Hepatic Tissue
KUPERMAN, Alexander V, KALGUTKAR, Amit S, MARFAT, Anthony, CHAMBERS, Robert J, LISTON, Theodore E
Published in Drug metabolism and disposition (01.11.2001)
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Published in Drug metabolism and disposition (01.11.2001)
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Structure–activity relationships of triazolopyridine oxazole p38 inhibitors: Identification of candidates for clinical development
McClure, Kim F., Letavic, Michael A., Kalgutkar, Amit S., Gabel, Christopher A., Audoly, Laurent, Barberia, John T., Braganza, John F., Carter, Demetrius, Carty, Thomas J., Cortina, Santo R., Dombroski, Mark A., Donahue, Kathleen M., Elliott, Nancy C., Gibbons, Colleen P., Jordan, Crystal K., Kuperman, Alexander V., Labasi, Jeff M., LaLiberte, Ronald E., McCoy, Jennifer M., Naiman, Brian M., Nelson, Kendra L., Nguyen, Hang T., Peese, Kevin M., Sweeney, Francis J., Taylor, Timothy J., Trebino, Catherine E., Abramov, Yuriy A., Laird, Ellen R., Volberg, Walter A., Zhou, Jun, Bach, Justin, Lombardo, Franco
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Journal Article
Discovery of the Hemifumarate and (α-l-Alanyloxy)methyl Ether as Prodrugs of an Antirheumatic Oxindole: Prodrugs for the Enolic OH Group
Robinson, Ralph P, Reiter, Lawrence A, Barth, Wayne E, Campeta, Anthony M, Cooper, Kelvin, Cronin, Brian J, Destito, Rosalina, Donahue, Kathleen M, Falkner, Fred C, Fiese, Eugene F, Johnson, Diane L, Kuperman, Alexander V, Liston, Theodore E, Malloy, Deborah, Martin, John J, Mitchell, David Y, Rusek, Frank W, Shamblin, Sheri L, Wright, Charles F
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyridine, a novel and selective p38α inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S., Hatch, Heather L., Kosea, Frederick, Nguyen, Hang T., Choo, Edna F., McClure, Kim F., Taylor, Timothy J., Henne, Kirk R., Kuperman, Alexander V., Dombroski, Mark A., Letavic, Michael A.
Published in Biopharmaceutics & drug disposition (01.11.2006)
Published in Biopharmaceutics & drug disposition (01.11.2006)
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Journal Article
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyridine, a novel and selective p38alpha inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S, Hatch, Heather L, Kosea, Frederick, Nguyen, Hang T, Choo, Edna F, McClure, Kim F, Taylor, Timothy J, Henne, Kirk R, Kuperman, Alexander V, Dombroski, Mark A, Letavic, Michael A
Published in Biopharmaceutics & drug disposition (01.11.2006)
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Published in Biopharmaceutics & drug disposition (01.11.2006)
Journal Article
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3 -isopropyl -[1,2,4 ] -triazolo [4,3-a] pyridine, a novel and selective p38a inhibitor : Identification of an active metabolite in preclinical species and human liver microsomes
KALGUTKAR, Amit S, HATCH, Heather L, LETAVIC, Michael A, KOSEA, Frederick, NGUYEN, Hang T, CHOO, Edna F, MCCLURE, Kim F, TAYLOR, Timothy J, HENNE, Kirk R, KUPERMAN, Alexander V, DOMBROSKI, Mark A
Published in Biopharmaceutics & drug disposition (2006)
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Published in Biopharmaceutics & drug disposition (2006)
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Preclinical pharmacokinetics and metabolism of 6-(4-(2,5- difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyr idine , a novel and selective p38 alpha inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S, Hatch, Heather L, Kosea, Frederick, Nguyen, Hang T, Choo, Edna F, McClure, Kim F, Taylor, Timothy J, Henne, Kirk R, Kuperman, Alexander V, Dombroski, Mark A, Letavic, Michael A
Published in Biopharmaceutics & drug disposition (01.01.2006)
Published in Biopharmaceutics & drug disposition (01.01.2006)
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