Scalable, One-Pot, Microwave-Accelerated Tandem Synthesis of Unsymmetrical Urea Derivatives
Kulkarni, Abhijit R, Garai, Sumanta, Thakur, Ganesh A
Published in Journal of organic chemistry (20.01.2017)
Published in Journal of organic chemistry (20.01.2017)
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Journal Article
The analgesic-like properties of the alpha7 nAChR silent agonist NS6740 is associated with non-conducting conformations of the receptor
Papke, Roger L., Bagdas, Deniz, Kulkarni, Abhijit R., Gould, Timothy, AlSharari, Shakir D., Thakur, Ganesh A., Damaj, M. Imad
Published in Neuropharmacology (01.04.2015)
Published in Neuropharmacology (01.04.2015)
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Journal Article
Critical Molecular Determinants of α7 Nicotinic Acetylcholine Receptor Allosteric Activation: SEPARATION OF DIRECT ALLOSTERIC ACTIVATION AND POSITIVE ALLOSTERIC MODULATION
Horenstein, Nicole A, Papke, Roger L, Kulkarni, Abhijit R, Chaturbhuj, Ganesh U, Stokes, Clare, Manther, Khan, Thakur, Ganesh A
Published in The Journal of biological chemistry (04.03.2016)
Published in The Journal of biological chemistry (04.03.2016)
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Journal Article
Persistent activation of α7 nicotinic ACh receptors associated with stable induction of different desensitized states
Papke, Roger L, Stokes, Clare, Damaj, M Imad, Thakur, Ganesh A, Manther, Khan, Treinin, Millet, Bagdas, Deniz, Kulkarni, Abhijit R, Horenstein, Nicole A
Published in British journal of pharmacology (01.06.2018)
Published in British journal of pharmacology (01.06.2018)
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Journal Article
Novel Electrophilic and Photoaffinity Covalent Probes for Mapping the Cannabinoid 1 Receptor Allosteric Site(s)
Kulkarni, Pushkar M, Kulkarni, Abhijit R, Korde, Anisha, Tichkule, Ritesh B, Laprairie, Robert B, Denovan-Wright, Eileen M, Zhou, Han, Janero, David R, Zvonok, Nikolai, Makriyannis, Alexandros, Cascio, Maria G, Pertwee, Roger G, Thakur, Ganesh A
Published in Journal of medicinal chemistry (14.01.2016)
Published in Journal of medicinal chemistry (14.01.2016)
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Journal Article
Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant β Subunits Acquire Sensitivity to α7-Selective Positive Allosteric Modulators
Stokes, Clare, Garai, Sumanta, Kulkarni, Abhijit R., Cantwell, Lucas N., Noviello, Colleen M., Hibbs, Ryan E., Horenstein, Nicole A., Abboud, Khalil A., Thakur, Ganesh A., Papke, Roger L.
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
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Journal Article
The interaction between alpha 7 nicotinic acetylcholine receptor and nuclear peroxisome proliferator-activated receptor-α represents a new antinociceptive signaling pathway in mice
Donvito, Giulia, Bagdas, Deniz, Toma, Wisam, Rahimpour, Elnaz, Jackson, Asti, Meade, Julie A., AlSharari, Shakir, Kulkarni, Abhijit R., Ivy Carroll, F., Lichtman, Aron H., Papke, Roger L., Thakur, Ganesh A., Imad Damaj, M.
Published in Experimental neurology (01.09.2017)
Published in Experimental neurology (01.09.2017)
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Journal Article
The Activity of GAT107, an Allosteric Activator and Positive Modulator of α7 Nicotinic Acetylcholine Receptors (nAChR), Is Regulated by Aromatic Amino Acids That Span the Subunit Interface
Papke, Roger L., Horenstein, Nicole A., Kulkarni, Abhijit R., Stokes, Clare, Corrie, Lu W., Maeng, Cheol-Young, Thakur, Ganesh A.
Published in The Journal of biological chemistry (14.02.2014)
Published in The Journal of biological chemistry (14.02.2014)
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Journal Article
RIC3, the cholinergic anti-inflammatory pathway, and neuroinflammation
Ben-David, Yael, Kagan, Sara, Cohen Ben-Ami, Hagit, Rostami, Jinar, Mizrahi, Tehila, Kulkarni, Abhijit R., Thakur, Ganesh A., Vaknin-Dembinsky, Adi, Healy, Luke M., Brenner, Talma, Treinin, Millet
Published in International immunopharmacology (01.06.2020)
Published in International immunopharmacology (01.06.2020)
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Journal Article
Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant β Subunits Acquire Sensitivity to α 7-Selective Positive Allosteric Modulators
Stokes, Clare, Garai, Sumanta, Kulkarni, Abhijit R, Cantwell, Lucas N, Noviello, Colleen M, Hibbs, Ryan E, Horenstein, Nicole A, Abboud, Khalil A, Thakur, Ganesh A, Papke, Roger L
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2019)
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Journal Article
Mapping Cannabinoid 1 Receptor Allosteric Site(s): Critical Molecular Determinant and Signaling Profile of GAT100, a Novel, Potent, and Irreversibly Binding Probe
Laprairie, Robert B, Kulkarni, Abhijit R, Kulkarni, Pushkar M, Hurst, Dow P, Lynch, Diane, Reggio, Patricia H, Janero, David R, Pertwee, Roger G, Stevenson, Lesley A, Kelly, Melanie E. M, Denovan-Wright, Eileen M, Thakur, Ganesh A
Published in ACS chemical neuroscience (15.06.2016)
Published in ACS chemical neuroscience (15.06.2016)
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Expeditious Synthesis, Enantiomeric Resolution, and Enantiomer Functional Characterization of (4-(4-Bromophenyl)-3a,4,5,9b-tetrahydro‑3H‑cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): An Allosteric Agonist-Positive Allosteric Modulator of α7 Nicotinic Acetylcholine Receptors
Thakur, Ganesh A, Kulkarni, Abhijit R, Deschamps, Jeffrey R, Papke, Roger L
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Journal Article
Expeditious Synthesis, Enantiomeric Resolution, and Enantiomer Functional Characterization of (4-(4-Bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): An Allosteric Agonist-Positive Allosteric Modulator of alpha 7 Nicotinic Acetylcholine Receptors
Thakur, Ganesh A., Kulkarni, Abhijit R., Deschamps, Jeffrey R., Papke, Roger L.
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Journal Article
Expeditious Synthesis, Enantiomeric Resolution, and Enantiomer Functional Characterization of (4-(4-Bromophenyl)-3a,4,5,9b-tetrahydro-3 H -cyclopenta[ c ]quinoline-8-sulfonamide (4BP-TQS): An Allosteric Agonist-Positive Allosteric Modulator of α7 Nicotinic Acetylcholine Receptors
Thakur, Ganesh A., Kulkarni, Abhijit R., Deschamps, Jeffrey R., Papke, Roger L.
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Journal Article
Genetic testing in alpha-1 antitrypsin deficiency – to sequence or not
Wan, Ken L., Froomes, Paul, Mazurkijevic, Laura J., Knezovich, Tamaryn, Dennis, Kyle, Bartlett, Essra, Chia, Nicole L.N., Williams, Mark G., Taylor, Peter J., Lu, Zhong X., Wijeratne, Nilika, McNeil, Alan, Lau, Chiyan, Kulkarni, Abhijit R., Mina, Kym D.
Published in Pathology (01.02.2023)
Published in Pathology (01.02.2023)
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Journal Article
Critical Molecular Determinants of α7 Nicotinic Acetylcholine Receptor Allosteric Activation
Horenstein, Nicole A., Papke, Roger L., Kulkarni, Abhijit R., Chaturbhuj, Ganesh U., Stokes, Clare, Manther, Khan, Thakur, Ganesh A.
Published in The Journal of biological chemistry (04.03.2016)
Published in The Journal of biological chemistry (04.03.2016)
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