High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C‑Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling
Kuhn, Kilian K, Ertl, Thomas, Dukorn, Stefanie, Keller, Max, Bernhardt, Günther, Reiser, Oliver, Buschauer, Armin
Published in Journal of medicinal chemistry (14.07.2016)
Published in Journal of medicinal chemistry (14.07.2016)
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Journal Article
In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d‑Amino Acids into Oligopeptides Derived from the C‑Termini of the Endogenous Agonists
Kuhn, Kilian K, Littmann, Timo, Dukorn, Stefanie, Tanaka, Miho, Keller, Max, Ozawa, Takeaki, Bernhardt, Günther, Buschauer, Armin
Published in ACS omega (31.07.2017)
Published in ACS omega (31.07.2017)
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Journal Article
Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples
Keller, Max, Kuhn, Kilian K, Einsiedel, Jürgen, Hübner, Harald, Biselli, Sabrina, Mollereau, Catherine, Wifling, David, Svobodová, Jaroslava, Bernhardt, Günther, Cabrele, Chiara, Vanderheyden, Patrick M L, Gmeiner, Peter, Buschauer, Armin
Published in Journal of medicinal chemistry (10.03.2016)
Published in Journal of medicinal chemistry (10.03.2016)
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Journal Article
Mimicking of Arginine by Functionalized N ω‑Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples
Keller, Max, Kuhn, Kilian K, Einsiedel, Jürgen, Hübner, Harald, Biselli, Sabrina, Mollereau, Catherine, Wifling, David, Svobodová, Jaroslava, Bernhardt, Günther, Cabrele, Chiara, Vanderheyden, Patrick M. L, Gmeiner, Peter, Buschauer, Armin
Published in Journal of medicinal chemistry (10.03.2016)
Published in Journal of medicinal chemistry (10.03.2016)
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Journal Article
In Search of NPY Y 4 R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists
Kuhn, Kilian K, Littmann, Timo, Dukorn, Stefanie, Tanaka, Miho, Keller, Max, Ozawa, Takeaki, Bernhardt, Günther, Buschauer, Armin
Published in ACS omega (31.07.2017)
Published in ACS omega (31.07.2017)
Get full text
Journal Article
High Affinity Agonists of the Neuropeptide Y (NPY) Y-4 Receptor Derived from the C-Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling
Kuhn, Kilian K., Ertl, Thomas, Dukorn, Stefanie, Keller, Max, Bernhardt, Guenther, Reiser, Oliver, Buschauer, Armin
Published in Journal of medicinal chemistry (14.07.2016)
Published in Journal of medicinal chemistry (14.07.2016)
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Journal Article
N-omega-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y-1 Receptor Antagonists and a Radio labeled Selective High-Affinity Molecular Tool ([H-3]UR-MK299) with Extended Residence Time
Keller, Max, Weiss, Stefan, Hutzler, Christoph, Kuhn, Kilian K., Mollereau, Catherine, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Gunther, Konig, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (26.11.2015)
Published in Journal of medicinal chemistry (26.11.2015)
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Journal Article
N ω -Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y 1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([ 3 H]UR-MK299) with Extended Residence Time
Keller, Max, Weiss, Stefan, Hutzler, Christoph, Kuhn, Kilian K., Mollereau, Catherine, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (25.11.2015)
Published in Journal of medicinal chemistry (25.11.2015)
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Journal Article
N(ω)-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([(3)H]UR-MK299) with Extended Residence Time
Keller, Max, Weiss, Stefan, Hutzler, Christoph, Kuhn, Kilian K, Mollereau, Catherine, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (25.11.2015)
Published in Journal of medicinal chemistry (25.11.2015)
Get full text
Journal Article
Nω‑Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y1 Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([3H]UR-MK299) with Extended Residence Time
Keller, Max, Weiss, Stefan, Hutzler, Christoph, Kuhn, Kilian K, Mollereau, Catherine, Dukorn, Stefanie, Schindler, Lisa, Bernhardt, Günther, König, Burkhard, Buschauer, Armin
Published in Journal of medicinal chemistry (25.11.2015)
Published in Journal of medicinal chemistry (25.11.2015)
Get full text
Journal Article