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Tatake, Revati J., O’Neill, Margaret M., Kennedy, Charles A., Wayne, Anita L., Jakes, Scott, Wu, Di, Kugler, Stanley Z., Kashem, Mohammed A., Kaplita, Paul, Snow, Roger J.
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Published in Biochemical and biophysical research communications (05.12.2008)
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Discovery of potent inhibitors of interleukin-2 inducible T-cell kinase (ITK) through structure-based drug design
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Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Published in Bioorganic & medicinal chemistry letters (15.03.2009)
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
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Mitigation of off-target adrenergic binding and effects on cardiovascular function in the discovery of novel ribosomal S6 kinase 2 inhibitors
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Published in The Journal of pharmacology and experimental therapeutics (01.03.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2012)
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2-Aminobenzimidazoles as potent ITK antagonists: trans-stilbene-like moieties targeting the kinase specificity pocket
Lo, Ho Yin, Bentzien, Jörg, Fleck, Roman W, Pullen, Steven S, Khine, Hnin Hnin, Woska, Jr, Joseph R, Kugler, Stanley Z, Kashem, Mohammed A, Takahashi, Hidenori
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
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2-Aminobenzimidazoles as potent 1TK antagonists : trans-stilbene-like moieties targeting the kinase specificity pocket
HO YIN LO, BENTZIEN, Jörg, FLECK, Roman W, PULLEN, Steven S, HNIN HNIN KHINE, WOSKA, Joseph R, KUGLER, Stanley Z, KASHEM, Mohammed A, TAKAHASHI, Hidenori
Published in Bioorganic & medicinal chemistry letters (2008)
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Published in Bioorganic & medicinal chemistry letters (2008)
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