Effect of the myeloperoxidase inhibitor AZD3241 on microglia: a PET study in Parkinson's disease
Jucaite, Aurelija, Svenningsson, Per, Rinne, Juha O, Cselényi, Zsolt, Varnäs, Katarina, Johnström, Peter, Amini, Nahid, Kirjavainen, Anna, Helin, Semi, Minkwitz, Margaret, Kugler, Alan R, Posener, Joel A, Budd, Samantha, Halldin, Christer, Varrone, Andrea, Farde, Lars
Published in Brain (London, England : 1878) (01.09.2015)
Published in Brain (London, England : 1878) (01.09.2015)
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A Phase 3 open-label study of the efficacy, safety and pharmacokinetics of buccally administered midazolam hydrochloride for the treatment of status epilepticus in pediatric Japanese subjects
Yoshinaga, Harumi, Benitez, Arturo, Takeda, Shinichi, Fournier, Martha, Kugler, Alan R.
Published in Epilepsy research (01.08.2021)
Published in Epilepsy research (01.08.2021)
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AZD3293: A Novel, Orally Active BACE1 Inhibitor with High Potency and Permeability and Markedly Slow Off-Rate Kinetics
Eketjäll, Susanna, Janson, Juliette, Kaspersson, Karin, Bogstedt, Anna, Jeppsson, Fredrik, Fälting, Johanna, Haeberlein, Samantha Budd, Kugler, Alan R, Alexander, Robert C, Cebers, Gvido
Published in Journal of Alzheimer's disease (01.01.2016)
Published in Journal of Alzheimer's disease (01.01.2016)
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Pregabalin Add‐on Treatment: A Randomized, Double‐blind, Placebo‐controlled, Dose–Response Study in Adults with Partial Seizures
Arroyo, Santiago, Anhut, Henning, Kugler, Alan R., Lee, Caroline M., Knapp, Lloyd E., Garofalo, Elizabeth A., Messmer, Silke
Published in Epilepsia (Copenhagen) (01.01.2004)
Published in Epilepsia (Copenhagen) (01.01.2004)
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AZD3293: Pharmacokinetic and Pharmacodynamic Effects in Healthy Subjects and Patients with Alzheimer's Disease
Cebers, Gvido, Alexander, Robert C, Haeberlein, Samantha Budd, Han, David, Goldwater, Ronald, Ereshefsky, Larry, Olsson, Tina, Ye, Naidong, Rosen, Laura, Russell, Muir, Maltby, Justine, Eketjäll, Susanna, Kugler, Alan R
Published in Journal of Alzheimer's disease (01.01.2017)
Published in Journal of Alzheimer's disease (01.01.2017)
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Safety and efficacy of two pregabalin regimens for add-on treatment of partial epilepsy
Beydoun, A, Uthman, B M, Kugler, A R, Greiner, M J, Knapp, L E, Garofalo, E A
Published in Neurology (08.02.2005)
Published in Neurology (08.02.2005)
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Dose-response trial of pregabalin adjunctive therapy in patients with partial seizures
French, J A, Kugler, A R, Robbins, J L, Knapp, L E, Garofalo, E A
Published in Neurology (27.05.2003)
Published in Neurology (27.05.2003)
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Virulence and antimicrobial resistance determinants of verotoxigenic Escherichia coli (VTEC) and of multidrug-resistant E. coli from foods of animal origin illegally imported to the EU by flight passengers
Nagy, B., Szmolka, A., Smole Možina, S., Kovač, J., Strauss, A., Schlager, S., Beutlich, J., Appel, B., Lušicky, M., Aprikian, P., Pászti, J., Tóth, I., Kugler, R., Wagner, M.
Published in International journal of food microbiology (16.09.2015)
Published in International journal of food microbiology (16.09.2015)
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Prophylactic efficacy of single dose pulmonary administration of amphotericin B inhalation powder in a guinea pig model of invasive pulmonary aspergillosis
Kirkpatrick, William R., Najvar, Laura K., Vallor, Ana C., Wiederhold, Nathan P., Bocanegra, Rosie, Pfeiffer, Juergen, Perkins, Kimberly, Kugler, Alan R., Sweeney, Theresa D., Patterson, Thomas F.
Published in Journal of antimicrobial chemotherapy (01.04.2012)
Published in Journal of antimicrobial chemotherapy (01.04.2012)
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Evidence of a charge-density threshold for optimum efficiency of biocidal cationic surfaces
Kugler, R, Bouloussa, O, Rondelez, F
Published in Microbiology (Society for General Microbiology) (01.05.2005)
Published in Microbiology (Society for General Microbiology) (01.05.2005)
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A saturable transport mechanism in the intestinal absorption of gabapentin is the underlying cause of the lack of proportionality between increasing dose and drug levels in plasma
Stewart, B H, Kugler, A R, Thompson, P R, Bockbrader, H N
Published in Pharmaceutical research (01.02.1993)
Published in Pharmaceutical research (01.02.1993)
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BACE1 Inhibitor Lanabecestat (AZD3293) in a Phase 1 Study of Healthy Japanese Subjects: Pharmacokinetics and Effects on Plasma and Cerebrospinal Fluid Aβ Peptides
Sakamoto, Kei, Matsuki, Shunji, Matsuguma, Kyoko, Yoshihara, Tatsuya, Uchida, Naoki, Azuma, Fumihiko, Russell, Muir, Hughes, Glen, Haeberlein, Samantha Budd, Alexander, Robert C, Eketjäll, Susanna, Kugler, Alan R
Published in Journal of clinical pharmacology (01.11.2017)
Published in Journal of clinical pharmacology (01.11.2017)
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Failure of Neuroprotection Despite Microglial Suppression by Delayed-Start Myeloperoxidase Inhibition in a Model of Advanced Multiple System Atrophy: Clinical Implications
Kaindlstorfer, Christine, Sommer, Patrick, Georgievska, Biljana, Mather, Robert J., Kugler, Alan R., Poewe, Werner, Wenning, Gregor K., Stefanova, Nadia
Published in Neurotoxicity research (01.10.2015)
Published in Neurotoxicity research (01.10.2015)
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Clinically Negligible Pharmacokinetic and Pharmacodynamic Interactions Between Lanabecestat and Dabigatran Etexilate, a Prototypical P-gp Substrate
Monk, Scott A, Kugler, Alan R, Andersen, Scott W, Ayan-Oshodi, Mosun A, James, Douglas E, Mullen, Jamie, Zimmer, Jennifer A, Willis, Brian A
Published in Journal of clinical pharmacology (01.05.2020)
Published in Journal of clinical pharmacology (01.05.2020)
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Endometrial polyps. A clinical study of 245 cases
Reslová, T, Tosner, J, Resl, M, Kugler, R, Vávrová, I
Published in Archives of gynecology and obstetrics (01.03.1999)
Published in Archives of gynecology and obstetrics (01.03.1999)
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