The Potent and Selective Histamine H3 Receptor Antagonist E169 Counteracts Cognitive Deficits and Mitigates Disturbances in the PI3K/AKT/GSK-3β Signaling Pathway in MK801-Induced Amnesia in Mice
Abdalla, Sabna, Eissa, Nermin, Jayaprakash, Petrilla, Beiram, Rami, Kuder, Kamil J, Łażewska, Dorota, Kieć-Kononowicz, Katarzyna, Sadek, Bassem
Published in International journal of molecular sciences (01.08.2023)
Published in International journal of molecular sciences (01.08.2023)
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Discovery of Potential, Dual-Active Histamine H3 Receptor Ligands with Combined Antioxidant Properties
Kuder, Kamil J., Kotańska, Magdalena, Szczepańska, Katarzyna, Mika, Kamil, Reiner-Link, David, Stark, Holger, Kieć-Kononowicz, Katarzyna
Published in Molecules (Basel, Switzerland) (15.04.2021)
Published in Molecules (Basel, Switzerland) (15.04.2021)
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AR71, Histamine H3 Receptor Ligand—In Vitro and In Vivo Evaluation (Anti-Inflammatory Activity, Metabolic Stability, Toxicity, and Analgesic Action)
Stasiak, Anna, Honkisz-Orzechowska, Ewelina, Gajda, Zbigniew, Wagner, Waldemar, Popiołek-Barczyk, Katarzyna, Kuder, Kamil J., Latacz, Gniewomir, Juszczak, Michał, Woźniak, Katarzyna, Karcz, Tadeusz, Szczepańska, Katarzyna, Jóźwiak-Bębenista, Marta, Kieć-Kononowicz, Katarzyna, Łażewska, Dorota
Published in International journal of molecular sciences (01.08.2024)
Published in International journal of molecular sciences (01.08.2024)
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Anti-Inflammatory Activities of 8-Benzylaminoxanthines Showing High Adenosine A2A and Dual A1/A2A Receptor Affinity
Załuski, Michał, Łażewska, Dorota, Jaśko, Piotr, Honkisz-Orzechowska, Ewelina, Kuder, Kamil J., Brockmann, Andreas, Latacz, Gniewomir, Zygmunt, Małgorzata, Kaleta, Maria, Greser, Beril Anita, Olejarz-Maciej, Agnieszka, Jastrzębska-Więsek, Magdalena, Vielmuth, Christin, Müller, Christa E., Kieć-Kononowicz, Katarzyna
Published in International journal of molecular sciences (05.09.2023)
Published in International journal of molecular sciences (05.09.2023)
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Benzophenone Derivatives with Histamine H3 Receptor Affinity and Cholinesterase Inhibitory Potency as Multitarget-Directed Ligands for Possible Therapy of Alzheimer’s Disease
Godyń, Justyna, Zaręba, Paula, Stary, Dorota, Kaleta, Maria, Kuder, Kamil J., Latacz, Gniewomir, Mogilski, Szczepan, Reiner-Link, David, Frank, Annika, Doroz-Płonka, Agata, Olejarz-Maciej, Agnieszka, Sudoł-Tałaj, Sylwia, Nolte, Tobias, Handzlik, Jadwiga, Stark, Holger, Więckowska, Anna, Malawska, Barbara, Kieć-Kononowicz, Katarzyna, Łażewska, Dorota, Bajda, Marek
Published in Molecules (Basel, Switzerland) (28.12.2022)
Published in Molecules (Basel, Switzerland) (28.12.2022)
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Histamine H3 Receptor Ligands—KSK-59 and KSK-73—Reduce Body Weight Gain in a Rat Model of Excessive Eating
Mika, Kamil, Szafarz, Małgorzata, Bednarski, Marek, Latacz, Gniewomir, Sudoł, Sylwia, Handzlik, Jadwiga, Pociecha, Krzysztof, Knutelska, Joanna, Nicosia, Noemi, Szczepańska, Katarzyna, Kuder, Kamil J., Kieć-Kononowicz, Katarzyna, Kotańska, Magdalena
Published in Pharmaceuticals (Basel, Switzerland) (25.10.2021)
Published in Pharmaceuticals (Basel, Switzerland) (25.10.2021)
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Metabolic and cardiovascular benefits and risks of 4-hydroxy guanabenz hydrochloride: α2-adrenoceptor and trace amine-associated receptor 1 ligand
Kotańska, Magdalena, Marcinkowska, Monika, Kuder, Kamil J., Walczak, Maria, Bednarski, Marek, Siwek, Agata, Kołaczkowski, Marcin
Published in Pharmacological reports (01.10.2023)
Published in Pharmacological reports (01.10.2023)
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N-Substituted piperazine derivatives as potential multitarget agents acting on histamine H-3 receptor and cancer resistance proteins
Szczepanska, Katarzyna, Kincses, Annamaria, Vincze, Klaudia, Szymanska, Ewa, Latacz, Gniewomir, Kuder, Kamil J., Stark, Holger, Spengler, Gabriella, Handzlik, Jadwiga, Kiec-Kononowicz, Katarzyna
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
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Journal Article
N-Substituted piperazine derivatives as potential multitarget agents acting on histamine H3 receptor and cancer resistance proteins
Szczepańska, Katarzyna, Kincses, Annamária, Vincze, Klaudia, Szymańska, Ewa, Latacz, Gniewomir, Kuder, Kamil J., Stark, Holger, Spengler, Gabriella, Handzlik, Jadwiga, Kieć-Kononowicz, Katarzyna
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
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Journal Article
Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H3R ligands
Szczepańska, Katarzyna, Karcz, Tadeusz, Mogilski, Szczepan, Siwek, Agata, Kuder, Kamil J., Latacz, Gniewomir, Kubacka, Monika, Hagenow, Stefanie, Lubelska, Annamaria, Olejarz, Agnieszka, Kotańska, Magdalena, Sadek, Bassem, Stark, Holger, Kieć-Kononowicz, Katarzyna
Published in European journal of medicinal chemistry (25.05.2018)
Published in European journal of medicinal chemistry (25.05.2018)
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An integrated study of the NE German Basin
Bayer, U., Scheck, M., Rabbel, W., Krawczyk, C.M., Götze, H.-J., Stiller, M., Beilecke, Th, Marotta, A.-M., Barrio-Alvers, L., Kuder, J.
Published in Tectonophysics (10.12.1999)
Published in Tectonophysics (10.12.1999)
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Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent
Szczepańska, Katarzyna, Pockes, Steffen, Podlewska, Sabina, Höring, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata, Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Mönnich, Denise, Seibel, Ulla, Kuder, Kamil J., Kotańska, Magdalena, Stark, Holger, Elz, Sigurd, Kieć-Kononowicz, Katarzyna
Published in European journal of medicinal chemistry (05.03.2021)
Published in European journal of medicinal chemistry (05.03.2021)
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Journal Article
Structural modifications in the distal, regulatory region of histamine H-3 receptor antagonists leading to the identification of a potent anti-obesity agent
Szczepanska, Katarzyna, Pockes, Steffen, Podlewska, Sabina, Horing, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata, Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Monnich, Denise, Seibel, Ulla, Kuder, Kamil J., Kotanska, Magdalena, Stark, Holger, Elz, Sigurd, Kiec-Kononowicz, Katarzyna
Published in European journal of medicinal chemistry (05.03.2021)
Published in European journal of medicinal chemistry (05.03.2021)
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Journal Article
Optimization and preclinical evaluation of novel histamine H-3 receptor ligands: Acetyl and propionyl phenoxyalkyl piperazine derivatives
Szczepanska, Katarzyna, Karcz, Tadeusz, Kotanska, Magdalena, Siwek, Agata, Kuder, Kamil J., Latacz, Gniewomir, Mogilski, Szczepan, Hagenow, Stefanie, Lubelska, Annamaria, Sobolewski, Michal, Stark, Holger, Kiec-Kononowicz, Katarzyna
Published in Bioorganic & medicinal chemistry (15.12.2018)
Published in Bioorganic & medicinal chemistry (15.12.2018)
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