Delivery of an ectonucleotidase inhibitor with ROS-responsive nanoparticles overcomes adenosine-mediated cancer immunosuppression
Mao, Chengqiong, Yeh, Stacy, Fu, Juan, Porosnicu, Mercedes, Thomas, Alexandra, Kucera, Gregory L, Votanopoulos, Konstantinos I, Tian, Shaomin, Ming, Xin
Published in Science translational medicine (08.06.2022)
Published in Science translational medicine (08.06.2022)
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Intrapleural nano-immunotherapy promotes innate and adaptive immune responses to enhance anti-PD-L1 therapy for malignant pleural effusion
Liu, Yang, Wang, Lulu, Song, Qianqian, Ali, Muhammad, Crowe, William N., Kucera, Gregory L., Hawkins, Gregory A., Soker, Shay, Thomas, Karl W., Miller, Lance D., Lu, Yong, Bellinger, Christina R., Zhang, Wei, Habib, Amyn A., Petty, W. Jeffrey, Zhao, Dawen
Published in Nature nanotechnology (01.02.2022)
Published in Nature nanotechnology (01.02.2022)
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Modulation of oxidative phosphorylation and mitochondrial biogenesis by cigarette smoke influence the response to immune therapy in NSCLC patients
Wang, Yuezhu, Smith, Margaret, Ruiz, Jimmy, Liu, Yin, Kucera, Gregory L., Topaloglu, Umit, Chan, Michael D., Li, Wencheng, Su, Jing, Xing, Fei
Published in Lung cancer (Amsterdam, Netherlands) (01.04.2023)
Published in Lung cancer (Amsterdam, Netherlands) (01.04.2023)
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Journal Article
Diet Alters Entero-Mammary Signaling to Regulate the Breast Microbiome and Tumorigenesis
Soto-Pantoja, David R, Gaber, Mohamed, Arnone, Alana A, Bronson, Steven M, Cruz-Diaz, Nildris, Wilson, Adam S, Clear, Kenysha Y J, Ramirez, Manuel U, Kucera, Gregory L, Levine, Edward A, Lelièvre, Sophie A, Chaboub, Lesley, Chiba, Akiko, Yadav, Hariom, Vidi, Pierre-Alexandre, Cook, Katherine L
Published in Cancer research (Chicago, Ill.) (15.07.2021)
Published in Cancer research (Chicago, Ill.) (15.07.2021)
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c-Met Mediated Cytokine Network Promotes Brain Metastasis of Breast Cancer by Remodeling Neutrophil Activities
Liu, Yin, Smith, Margaret R, Wang, Yuezhu, D'Agostino, Jr, Ralph, Ruiz, Jimmy, Lycan, Thomas, Kucera, Gregory L, Miller, Lance D, Li, Wencheng, Chan, Michael D, Farris, Michael, Su, Jing, Song, Qianqian, Zhao, Dawen, Chandrasekaran, Arvind, Xing, Fei
Published in Cancers (05.05.2023)
Published in Cancers (05.05.2023)
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Design of Enzymatically Cleavable Prodrugs of a Potent Platinum-Containing Anticancer Agent
Ding, Song, Pickard, Amanda J., Kucera, Gregory L., Bierbach, Ulrich
Published in Chemistry : a European journal (01.12.2014)
Published in Chemistry : a European journal (01.12.2014)
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Redesigning the DNA-Targeted Chromophore in Platinum-Acridine Anticancer Agents: A Structure-Activity Relationship Study
Pickard, Amanda J., Liu, Fang, Bartenstein, Thomas F., Haines, Laura G., Levine, Keith E., Kucera, Gregory L., Bierbach, Ulrich
Published in Chemistry : a European journal (01.12.2014)
Published in Chemistry : a European journal (01.12.2014)
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Journal Article
The novel phospholipid mimetic KPC34 is highly active against preclinical models of Philadelphia chromosome positive acute lymphoblastic leukemia
Alexander, Peter M, Caudell, David L, Kucera, Gregory L, Pladna, Kristin M, Pardee, Timothy S
Published in PloS one (23.06.2017)
Published in PloS one (23.06.2017)
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Synthesis, Aqueous Reactivity, and Biological Evaluation of Carboxylic Acid Ester-Functionalized Platinum–Acridine Hybrid Anticancer Agents
Graham, Leigh A, Suryadi, Jimmy, West, Tiffany K, Kucera, Gregory L, Bierbach, Ulrich
Published in Journal of medicinal chemistry (13.09.2012)
Published in Journal of medicinal chemistry (13.09.2012)
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Dissecting intratumoral myeloid cell plasticity by single cell RNA‐seq
Song, Qianqian, Hawkins, Gregory A., Wudel, Leonard, Chou, Ping‐Chieh, Forbes, Elizabeth, Pullikuth, Ashok K., Liu, Liang, Jin, Guangxu, Craddock, Lou, Topaloglu, Umit, Kucera, Gregory, O’Neill, Stacey, Levine, Edward A., Sun, Peiqing, Watabe, Kounosuke, Lu, Yong, Alexander‐Miller, Martha A., Pasche, Boris, Miller, Lance D., Zhang, Wei
Published in Cancer medicine (Malden, MA) (01.06.2019)
Published in Cancer medicine (Malden, MA) (01.06.2019)
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Journal Article
Improving nucleoside analogs via lipid conjugation: Is fatter any better?
Alexander, Peter, Kucera, Gregory, Pardee, Timothy S
Published in Critical reviews in oncology/hematology (01.04.2016)
Published in Critical reviews in oncology/hematology (01.04.2016)
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A Non-Cross-Linking Platinum−Acridine Agent with Potent Activity in Non-Small-Cell Lung Cancer
Ma, Zhidong, Choudhury, Jayati Roy, Wright, Marcus W, Day, Cynthia S, Saluta, Gilda, Kucera, Gregory L, Bierbach, Ulrich
Published in Journal of medicinal chemistry (11.12.2008)
Published in Journal of medicinal chemistry (11.12.2008)
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Synthesis, Reactivity, and Biological Activity of Gold(I) Complexes Modified with Thiourea-Functionalized Tyrosine Kinase Inhibitors
Yang, Mu, Pickard, Amanda J, Qiao, Xin, Gueble, Matthew J, Day, Cynthia S, Kucera, Gregory L, Bierbach, Ulrich
Published in Inorganic chemistry (06.04.2015)
Published in Inorganic chemistry (06.04.2015)
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Journal Article
Phosphorylation of PDHA by AMPK Drives TCA Cycle to Promote Cancer Metastasis
Cai, Zhen, Li, Chien-Feng, Han, Fei, Liu, Chunfang, Zhang, Anmei, Hsu, Che-Chia, Peng, Danni, Zhang, Xian, Jin, Guoxiang, Rezaeian, Abdol-Hossein, Wang, Guihua, Zhang, Weina, Pan, Bo-Syong, Wang, Chi-Yun, Wang, Yu-Hui, Wu, Shih-Ying, Yang, Shun-Chin, Hsu, Fang-Chi, D’Agostino, Ralph B., Furdui, Christina M., Kucera, Gregory L., Parks, John S., Chilton, Floyd H., Huang, Chih-Yang, Tsai, Fuu-Jen, Pasche, Boris, Watabe, Kounosuke, Lin, Hui-Kuan
Published in Molecular cell (15.10.2020)
Published in Molecular cell (15.10.2020)
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Gold(I) Analogues of a Platinum−Acridine Antitumor Agent Are Only Moderately Cytotoxic but Show Potent Activity against Mycobacterium tuberculosis
Eiter, Lauren C, Hall, Nathan W, Day, Cynthia S, Saluta, Gilda, Kucera, Gregory L, Bierbach, Ulrich
Published in Journal of medicinal chemistry (12.11.2009)
Published in Journal of medicinal chemistry (12.11.2009)
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