Pharmacological classification of histamine H3 receptor agents across species is attributable to transmembrane 3 sequence differences
Esbenshade, T A, Estvander, B R, Miller, T R, Baranowski, J L, Sharma, R, Hancock, A A, Krueger, K M
Published in Inflammation research (01.04.2007)
Published in Inflammation research (01.04.2007)
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Journal Article
Structure-activity relationships of A-331440: a new histamine-3 antagonist with anti-obesity properties
Faghih, R, Esbenshade, T A, Krueger, K M, Yao, B B, Witte, D G, Miller, T M, Kang, C H, Fox, G B, Cowart, M, Bennani, Y L, Hancock, A A
Published in Inflammation research (01.03.2004)
Published in Inflammation research (01.03.2004)
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Journal Article
Clathrin-mediated Endocytosis of the β-Adrenergic Receptor Is Regulated by Phosphorylation/Dephosphorylation of β-Arrestin1
Lin, Fang-Tsyr, Krueger, Kathleen M., Kendall, Humphrey E., Daaka, Yehia, Fredericks, Zoey L., Pitcher, Julie A., Lefkowitz, Robert J.
Published in The Journal of biological chemistry (05.12.1997)
Published in The Journal of biological chemistry (05.12.1997)
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Journal Article
The carboxyl terminus of the S1 subunit of pertussis toxin confers high affinity binding to transducin
CORTINA, G, KRUEGER, K. M, BARBIERI, T
Published in The Journal of biological chemistry (15.12.1991)
Published in The Journal of biological chemistry (15.12.1991)
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Journal Article
Protease treatment of pertussis toxin identifies the preferential cleavage of the S1 subunit
KRUEGER, K. M, MENDE-MUELLER, L. M, BARBIERI, J. T
Published in The Journal of biological chemistry (05.05.1991)
Published in The Journal of biological chemistry (05.05.1991)
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Journal Article
A new family of histamine H3 receptor antagonists based on a natural product: discovery, SAR, and properties of the series
Cowart, M, Sun, M, Zhao, C, Witte, D G, Miller, T R, Krueger, K M, Browman, K, Fox, G B, Bennani, Y L, Esbenshade, T A, Hancock, A A
Published in Inflammation research (01.04.2007)
Published in Inflammation research (01.04.2007)
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Journal Article
Antiobesity evaluation of histamine H3 receptor (H3R) antagonist analogs of A-331440 with improved safety and efficacy
Hancock, A A, Diehl, M S, Fey, T A, Bush, E N, Faghih, R, Miller, T R, Krueger, K M, Pratt, J K, Cowart, M D, Dickinson, R W, Shapiro, R, Knourek-Segel, V E, Droz, B A, McDowell, C A, Krishna, G, Brune, M E, Esbenshade, T A, Jacobson, P B
Published in Inflammation research (01.04.2005)
Published in Inflammation research (01.04.2005)
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Journal Article
Differences in pharmacological properties of histamine H3 receptor agonists and antagonists revealed at two human H3 receptor isoforms
Esbenshade, T. A., Krueger, K. M., Yao, B. B., Witte, D. G., Estvander, B. R., Baranowski, J. L., Miller, T. R., Hancock, A. A.
Published in Inflammation research (01.04.2006)
Published in Inflammation research (01.04.2006)
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Journal Article
Selective H3 receptor (H3R) blockade: broad efficacy in cognition and schizophrenia
Fox, G B, Esbenshade, T A, Pan, J B, Browman, K E, Zhang, M, Ballard, M E, Radek, R J, Miner, H, Bitner, R S, Krueger, K M, Yao, B B, Faghih, R, Rueter, L E, Komater, V A, Drescher, K U, Buckley, M J, Sullivan, J P, Cowart, M D, Decker, M W, Hancock, A A
Published in Inflammation research (01.04.2005)
Published in Inflammation research (01.04.2005)
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Journal Article
Use of novel, non-imidazole inverse agonist radioligands to define histamine H3 receptor pharmacology
Esbenshade, T A, Yao, B B, Witte, D G, Carr, T L, Sharma, R, Baranowski, J L, Krueger, K M, Miller, T R, Surber, B W, Faghih, R, Hancock, A A
Published in Inflammation research (01.04.2005)
Published in Inflammation research (01.04.2005)
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Journal Article
Distinctions and contradistinctions between antiobesity histamine H3 receptor (H3R) antagonists compared to cognition-enhancing H3 receptor antagonists
Esbenshade, T. A., Hancock, A. A., Bitner, R. S., Krueger, K. M., Otte, S., Nikkel, A. L., Fey, T. A., Bush, E. N., Dickinson, R. W., Shapiro, R., Knourek-Segel, V., Droz, B. A., Brune, M. E., Jacobson, P. B., Cowart, M. D.
Published in Inflammation research (01.04.2006)
Published in Inflammation research (01.04.2006)
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Journal Article
D-alanine piperazine-amides: novel non-imidazole antagonists of the histamine H3 receptor
Faghih, R, Phelan, K, Esbenshade, T A, Miller, T R, Kang, C H, Krueger, K M, Yao, B B, Fox, G B, Bennani, Y L, Hancock, A A
Published in Inflammation research (01.04.2003)
Published in Inflammation research (01.04.2003)
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Journal Article
2. Histaminergic mechanisms in the CNS: Selective H3 receptor (H3R) blockade: broad efficacy in cognition and schizophrenia
Fox, G. B., Esbenshade, T. A., Pan, J. B., Browman, K. E., Zhang, M., Ballard, M. E., Radek, R. J., Miner, H., Bitner, R. S., Krueger, K. M., Yao, B. B., Faghih, R., Rueter, L. E., Komater, V. A., Drescher, K. U., Buckley, M. J., Sullivan, J. P., Cowart, M. D., Decker, M. W., Hancock, A. A.
Published in Inflammation research (01.04.2005)
Published in Inflammation research (01.04.2005)
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Journal Article
In vitro pharmacological properties of two novel non-imidazole H3 receptor (H3R) antagonists
Yao, B B, Witte, D G, Miller, T R, Krueger, K M, Carr, T L, Kang, C H, Faghih, R, Bennani, Y L, Esbenshade, T A, Hancock, A A
Published in Inflammation research (01.04.2003)
Published in Inflammation research (01.04.2003)
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Journal Article
D-alanine piperazine-amides: novel non-imidazole antagonists of the histamine H 3 receptor
Faghih, R., Phelan, K., Esbenshade, T. A., Miller, T. R., Kang, C-H., Krueger, K. M., Yao, B. B., Fox, G. B., Bennani, Y. L., Hancock, A. A.
Published in Inflammation research (01.04.2003)
Published in Inflammation research (01.04.2003)
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Journal Article
In vitro pharmacological properties of two novel non-imidazole H 3 receptor (H 3 R) antagonists
Witte, D. G., Miller, T. R., Faghih, R., Yao, B. B., Esbenshade, T. A., Krueger, K. M., Carr, T. L., Kang, C. H., Hancock, A. A., Bennani, Y. L.
Published in Inflammation research (01.04.2003)
Published in Inflammation research (01.04.2003)
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Journal Article