Discovery, Chemistry, and Preclinical Development of Pritelivir, a Novel Treatment Option for Acyclovir-Resistant Herpes Simplex Virus Infections
Birkmann, Alexander, Bonsmann, Susanne, Kropeit, Dirk, Pfaff, Tamara, Rangaraju, Manickam, Sumner, Melanie, Timmler, Burkhard, Zimmermann, Holger, Buschmann, Helmut, Ruebsamen-Schaeff, Helga
Published in Journal of medicinal chemistry (27.10.2022)
Published in Journal of medicinal chemistry (27.10.2022)
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Journal Article
Evaluation of the Clinical Drug‐Drug Interaction Potential of Pritelivir on Transporters and CYP450 Enzymes Using a Cocktail Approach
Vries, Michiel, Bonsmann, Susanne, Pausch, Jörg, Sumner, Melanie, Birkmann, Alexander, Zimmermann, Holger, Kropeit, Dirk
Published in Clinical pharmacology in drug development (01.07.2024)
Published in Clinical pharmacology in drug development (01.07.2024)
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Journal Article
Pharmacokinetics and Safety of Letermovir Coadministered With Cyclosporine A or Tacrolimus in Healthy Subjects
Kropeit, Dirk, Richter, Oliver, Stobernack, Hans‐Peter, Rübsamen‐Schaeff, Helga, Zimmermann, Holger
Published in Clinical pharmacology in drug development (01.01.2018)
Published in Clinical pharmacology in drug development (01.01.2018)
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Journal Article
Mass Balance and Metabolite Profile after Single and Multiple Oral Doses of Pritelivir in Healthy Subjects
Bonsmann, Susanne, McCormick, David, Pausch, Jörg, Vries, Michiel, Sumner, Melanie, Birkmann, Alexander, Zimmermann, Holger, Kropeit, Dirk
Published in Clinical pharmacology in drug development (01.04.2024)
Published in Clinical pharmacology in drug development (01.04.2024)
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Journal Article
Pharmacokinetics and safety of letermovir, a novel anti‐human cytomegalovirus drug, in patients with renal impairment
Kropeit, Dirk, Scheuenpflug, Jürgen, Erb‐Zohar, Katharina, Halabi, Atef, Stobernack, Hans‐Peter, Hulskotte, Ellen G. J., Schanke, Arne, Zimmermann, Holger, Rübsamen‐Schaeff, Helga
Published in British journal of clinical pharmacology (01.09.2017)
Published in British journal of clinical pharmacology (01.09.2017)
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Journal Article
Pharmacokinetics and safety of the anti‐human cytomegalovirus drug letermovir in subjects with hepatic impairment
Kropeit, Dirk, McCormick, David, Erb‐Zohar, Katharina, Moiseev, Valentin S., Kobalava, Zhanna D., Stobernack, Hans‐Peter, Zimmermann, Holger, Rübsamen‐Schaeff, Helga
Published in British journal of clinical pharmacology (01.12.2017)
Published in British journal of clinical pharmacology (01.12.2017)
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Journal Article
FRI-199-First in Human, single ascending dose clinical trial of AIC649 in patients with chronic hepatitis
Addy, Ibironke, Jambrecina, Alen, Berg, Thomas, Bömmel, Florian van, Kropeit, Dirk, Vank, Christiane, Bigge, Alexandra, Nedoschinsky, Katja, Stobernack, Hans-Peter, Rangaraju, Manickam, Kummer, Silke, Matschl, Urte, Gehring, Adam, Eberhard, Johanna, Altfeld, Marcus, Wiesch, Julian Schulze zur, Zimmermann, Holger, Paulsen, Daniela
Published in Journal of hepatology (01.04.2019)
Published in Journal of hepatology (01.04.2019)
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First‐in‐Human, Single‐ and Multiple‐Ascending‐Dose, Food‐Effect, and Absolute Bioavailability Trials to Assess the Pharmacokinetics, Safety, and Tolerability of Pritelivir, a Nonnucleoside Helicase‐Primase Inhibitor Against Herpes Simplex Virus in Healthy Subjects
Kropeit, Dirk, Bonsmann, Susanne, Richter, Oliver, McCormick, David, Pausch, Jörg, Sumner, Melanie, Birkmann, Alexander, Zimmermann, Holger, Rübsamen‐Schaeff, Helga
Published in Clinical pharmacology in drug development (01.07.2023)
Published in Clinical pharmacology in drug development (01.07.2023)
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Journal Article
Pharmacokinetics and Safety of Letermovir and Midazolam Coadministration in Healthy Subjects
Kropeit, Dirk, McCormick, David, Erb‐Zohar, Katharina, Stobernack, Hans‐Peter, Zimmermann, Holger, Rübsamen‐Schaeff, Helga
Published in Clinical pharmacology in drug development (01.01.2022)
Published in Clinical pharmacology in drug development (01.01.2022)
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Journal Article
The Effect of Oral Letermovir Administration on the Pharmacokinetics of a Single Oral Dose of P‐Glycoprotein Substrate Digoxin in Healthy Volunteers
Scheuenpflug, Jürgen, Kropeit, Dirk, Erb‐Zohar, Katharina, Theis, Jochen G.W., Stobernack, Hans‐Peter, McCormick, David, Zimmermann, Holger, Rübsamen‐Schaeff, Helga
Published in Clinical pharmacology in drug development (01.01.2022)
Published in Clinical pharmacology in drug development (01.01.2022)
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Journal Article
Pharmacokinetics-Pharmacodynamics of the Helicase-Primase Inhibitor Pritelivir following Treatment of Wild-Type or Pritelivir-Resistant Virus Infection in a Murine Herpes Simplex Virus 1 Infection Model
BISWAS, Subhajit, SUKLA, Soumi, GOLDNER, Thomas, FIELD, Hugh J, KROPEIT, Dirk, PAULSEN, Daniela, WELBERS, André, RUEBSAMEN-SCHAEFF, Helga, ZIMMERMANN, Holger, BIRKMANN, Alexander
Published in Antimicrobial agents and chemotherapy (01.07.2014)
Published in Antimicrobial agents and chemotherapy (01.07.2014)
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