Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader
Carmona, Angelica V, Jonnalagadda, Shirisha, Case, Alfie M, Maddeboina, Krishnaiah, Jonnalagadda, Sravan K, Dow, Louise F, Duan, Ling, Penning, Trevor M, Trippier, Paul C
Published in Communications chemistry (29.04.2024)
Published in Communications chemistry (29.04.2024)
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Journal Article
Highly regioselective ring opening of epoxides and aziridines using (bromodimethyl)sulfonium bromide
Das, Biswanath, Krishnaiah, Maddeboina, Venkateswarlu, Katta
Published in Tetrahedron letters (26.06.2006)
Published in Tetrahedron letters (26.06.2006)
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Journal Article
1425 The novel small molecule multitarget inhibitor LCI133 sensitizes endometrial carcinoma to TRAIL-mediated apoptosis
McHale, Cody C, Delara, Ritchie, Pal, Dhananjaya, Maddeboina, Krishnaiah, Dryden, Hailey, Arditti, Page Mangum, Yada, Bharath, Wendel Naumnn, R, Crane, Erin, Brown, Jubilee, Durden, Donald
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
Combinatorial inhibition of BTK, PI3K-AKT and BRD4-MYC as a strategy for treatment of mantle cell lymphoma
Vann, Kendra R., Pal, Dhananjaya, Smith, Audrey L., Sahar, Namood-e, Krishnaiah, Maddeboina, El-Gamal, Dalia, Kutateladze, Tatiana G.
Published in Molecular biomedicine (15.01.2022)
Published in Molecular biomedicine (15.01.2022)
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Journal Article
Regio- and stereoselective ring opening of epoxides and aziridines using zirconyl chloride: An efficient approach for the synthesis of beta-chlorohydrins and beta-chloroamines
Das, Biswanath, Krishnaiah, Maddeboina, Venkateswarlu, Katta
Published in Chemistry letters (05.01.2007)
Published in Chemistry letters (05.01.2007)
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Journal Article
Hypervalent iodine-mediated efficient synthesis of imidazoles
Das, Biswanath, Srinivas, Yallamalla, Holla, Harish, Krishnaiah, Maddeboina, Narender, Ravirala
Published in Chemistry letters (05.10.2007)
Published in Chemistry letters (05.10.2007)
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Journal Article
Protecting Groups in Peptide Synthesis
Conda-Sheridan, Martin, Krishnaiah, Maddeboina
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
Published in Methods in molecular biology (Clifton, N.J.) (01.01.2020)
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Journal Article
Recent advances in multitarget-directed ligands via in silico drug discovery
Maddeboina, Krishnaiah, Yada, Bharath, Kumari, Shikha, McHale, Cody, Pal, Dhananjaya, Durden, Donald L.
Published in Drug discovery today (01.03.2024)
Published in Drug discovery today (01.03.2024)
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Journal Article
A Rapid and Efficient Stereoselective Synthesis of (Z)- and (E)-Allyl Bromides fromBaylis–Hillman Adducts Using Bromo(dimethyl)sulfonium Bromide
Das, Biswanath, Venkateswarlu, Katta, Krishnaiah, Maddeboina, Holla, Harish, Majhi, Anjoy
Published in Helvetica chimica acta (01.07.2006)
Published in Helvetica chimica acta (01.07.2006)
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Journal Article
Pivotal role of nitrogen heterocycles in Alzheimer’s disease drug discovery
Kumari, Shikha, Maddeboina, Krishnaiah, Bachu, Rinda Devi, Boddu, Sai H.S., Trippier, Paul C., Tiwari, Amit K.
Published in Drug discovery today (01.10.2022)
Published in Drug discovery today (01.10.2022)
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Journal Article
The Novel CDK9/CDK4/6/PI3K Triple Inhibitor LCI139 for the Treatment of MYC -Driven Mantle Cell Lymphoma
Pal, Dhananjaya, Arditti, Page Mangum, Maddeboina, Krishnaiah, McHale, Cody C., Yang, Hsih-Te, Yada, Bharath, Dryden, Hailey Lynn, Foureau, David M, Durden, Donald L.
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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Journal Article
Novel multitarget small molecule inhibitor LCI133 and synthetic lethality in endometrial carcinoma via CDK9/PI3K axis
Delara, Ritchie, Pal, Dhananjaya, Maddeboina, Krishnaiah, Naumann, R. Wendel, Crane, Erin, Brown, Jubilee, Mangum Arditti, Page, Dryden, Hailey L., Yada, Bharath, Sha, Wei, Durden, Donald, McHale, Cody
Published in Journal of clinical oncology (01.06.2023)
Published in Journal of clinical oncology (01.06.2023)
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Journal Article
Aldo-Keto Reductase 1C3 Inhibitor Prodrug Improves Pharmacokinetic Profile and Demonstrates In Vivo Efficacy in a Prostate Cancer Xenograft Model
Maddeboina, Krishnaiah, Jonnalagadda, Sravan K., Morsy, Ahmed, Duan, Ling, Chhonker, Yashpal S., Murry, Daryl J., Penning, Trevor M., Trippier, Paul C.
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Journal Article
Discovery of N‑((4-([1,2,4]Triazolo[1,5‑a]pyridin-6-yl)-5-(6-methylpyridin-2-yl)‑1H‑imidazol-2-yl)methyl)-2-fluoroaniline (EW-7197): A Highly Potent, Selective, and Orally Bioavailable Inhibitor of TGF‑β Type I Receptor Kinase as Cancer Immunotherapeutic/Antifibrotic Agent
Jin, Cheng Hua, Krishnaiah, Maddeboina, Sreenu, Domalapally, Subrahmanyam, Vura B, Rao, Kota S, Lee, Hwa Jeong, Park, So-Jung, Park, Hyun-Ju, Lee, Kiho, Sheen, Yhun Yhong, Kim, Dae-Kee
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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Journal Article
A remarkably simple N-formylation of anilines using polyethylene glycol
Das, Biswanath, Krishnaiah, Maddeboina, Balasubramanyam, P., Veeranjaneyulu, Boyapati, Nandan Kumar, D.
Published in Tetrahedron letters (31.03.2008)
Published in Tetrahedron letters (31.03.2008)
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Journal Article
Synthesis, biological evaluation, and metabolic stability of phenazine derivatives as antibacterial agents
Krishnaiah, Maddeboina, de Almeida, Nathalia Rodrigues, Udumula, Venkatareddy, Song, Zhongcheng, Chhonker, Yashpal Singh, Abdelmoaty, Mai M., do Nascimento, Valter Aragao, Murry, Daryl J., Conda-Sheridan, Martin
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
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