Discovery and evaluation of novel Mycobacterium tuberculosis ketol-acid reductoisomerase inhibitors as therapeutic drug leads
Krishna, Vagolu Siva, Zheng, Shan, Rekha, Estharla Madhu, Guddat, Luke W., Sriram, Dharmarajan
Published in Journal of computer-aided molecular design (01.03.2019)
Published in Journal of computer-aided molecular design (01.03.2019)
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Journal Article
Synthesis, antitubercular evaluation and molecular docking studies of phthalimide bearing 1,2,3-triazoles
Phatak, Pramod S., Bakale, Rajubai D., Dhumal, Sambhaji T., Dahiwade, Lalita K., Choudhari, Prafulla B., Siva Krishna, Vagolu, Sriram, Dharmarajan, Haval, Kishan P.
Published in Synthetic communications (18.08.2019)
Published in Synthetic communications (18.08.2019)
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Journal Article
The design and green synthesis of novel benzotriazoloquinolinyl spirooxindolopyrrolizidines: antimycobacterial and antiproliferative studies
Pogaku, Vinay, Krishna, Vagolu Siva, Balachandran, Chandrasekar, Rangan, Krishnan, Sriram, Dharmarajan, Aoki, Shin, Basavoju, Srinivas
Published in New journal of chemistry (2019)
Published in New journal of chemistry (2019)
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Journal Article
Isoniazid Linked to Sulfonate Esters via Hydrazone Functionality: Design, Synthesis, and Evaluation of Antitubercular Activity
Koçak Aslan, Ebru, Han, Muhammed İhsan, Krishna, Vagolu Siva, Tamhaev, Rasoul, Dengiz, Cagatay, Doğan, Şengül Dilem, Lherbet, Christian, Mourey, Lionel, Tønjum, Tone, Gündüz, Miyase Gözde
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2022)
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2022)
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Journal Article
Design, synthesis, and in vitro biological evaluation of dehydroaripiprazole derivatives as antituberculosis agents and molecular docking study
Raja Sekhara Reddy, B., Pratap Reddy Gajulapalli, V., Madhu Rekha, Estharla, Siva Krishna, Vagolu, Sriram, Dharmarajan, Sudakar Babu, K, Kim, Eunha
Published in Results in Chemistry (01.01.2022)
Published in Results in Chemistry (01.01.2022)
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Journal Article
Ultrasonication-ionic liquid synergy for the synthesis of new potent anti-tuberculosis 1,2,4-triazol-1-yl-pyrazole based spirooxindolopyrrolizidines
Pogaku, Vinay, Krishna, Vagolu Siva, Sriram, Dharmarajan, Rangan, Krishnan, Basavoju, Srinivas
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
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Journal Article
Synthesis of novel morpholine, thiomorpholine and N-substituted piperazine coupled 2-(thiophen-2-yl)dihydroquinolines as potent inhibitors of Mycobacterium tuberculosis
Marvadi, Sandeep Kumar, Krishna, Vagolu Siva, Sriram, Dharmarajan, Kantevari, Srinivas
Published in European journal of medicinal chemistry (15.02.2019)
Published in European journal of medicinal chemistry (15.02.2019)
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Journal Article
Pyrazole–coumarin and pyrazole–quinoline chalcones as potential antitubercular agents
Kumar, Gautam, Siva Krishna, Vagolu, Sriram, Dharmarajan, Jachak, Sanjay M.
Published in Archiv der Pharmazie (Weinheim) (01.08.2020)
Published in Archiv der Pharmazie (Weinheim) (01.08.2020)
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Journal Article
Stereoselective synthesis and discovery of novel spirooxindolopyrrolidine engrafted indandione heterocyclic hybrids as antimycobacterial agents
Arumugam, Natarajan, Almansour, Abdulrahman I., Kumar, Raju Suresh, Siva Krishna, Vagolu, Sriram, Dharmarajan, Dege, Necmi
Published in Bioorganic chemistry (01.05.2021)
Published in Bioorganic chemistry (01.05.2021)
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Journal Article
Synthesis and biological evaluation of 1H-pyrrolo[2,3-d]pyrimidine-1,2,3-triazole derivatives as novel anti-tubercular agents
Shiva Raju, Kasa, AnkiReddy, Sandeep, Sabitha, Gowravaram, Siva Krishna, Vagolu, Sriram, Dharmarajan, Bharathi Reddy, Kunduru, Rao Sagurthi, Someswar
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
Published in Bioorganic & medicinal chemistry letters (15.01.2019)
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Journal Article
Identification and development of benzoxazole derivatives as novel bacterial glutamate racemase inhibitors
Malapati, Prasanthi, Krishna, Vagolu Siva, Nallangi, Radhika, Srilakshmi, Rudraraju Reshma, Sriram, Dharmarajan
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
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Journal Article
1,2,3-Triazole-fused spirochromenes as potential anti-tubercular agents: synthesis and biological evaluation
Ashok, Dongamanti, Chiranjeevi, Pamula, Kumar, Aamate Vikas, Sarasija, Madderla, Krishna, Vagolu Siva, Sriram, Dharmarajan, Balasubramanian, Sridhar
Published in RSC advances (01.01.2018)
Published in RSC advances (01.01.2018)
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Journal Article
Anti-tubercular activity of novel class of spiropyrrolidine tethered indenoquinoxaline heterocyclic hybrids
Arumugam, Natarajan, Almansour, Abdulrahman I., Suresh Kumar, Raju, Ibrahim Alaqeel, Shatha, Siva Krishna, Vagolu, Sriram, Dharmarajan
Published in Bioorganic chemistry (01.06.2020)
Published in Bioorganic chemistry (01.06.2020)
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Journal Article
Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities
Keleş Atıcı, Rüveyde, Doğan, Şengül Dilem, Gündüz, Miyase Gözde, Krishna, Vagolu Siva, Chebaiki, Melina, Homberset, Håvard, Lherbet, Christian, Mourey, Lionel, Tønjum, Tone
Published in Drug development research (01.09.2022)
Published in Drug development research (01.09.2022)
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Journal Article
Regio- and diastereoselective synthesis of spiropyrroloquinoxaline grafted indole heterocyclic hybrids and evaluation of their anti- Mycobacterium tuberculosis activity
Arumugam, Natarajan, Almansour, Abdulrahman I, Kumar, Raju Suresh, Mohammad Ali Al-Aizari, Abdul Jaleel, Alaqeel, Shatha Ibrahim, Kansız, Sevgi, Krishna, Vagolu Siva, Sriram, Dharmarajan, Dege, Necmi
Published in RSC advances (19.06.2020)
Published in RSC advances (19.06.2020)
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Journal Article