Synthesis, Pharmacological Characterization, and Molecular Modeling of Heterobicyclic Amino Acids Related to (+)-2-Aminobicyclo[3.1.0]hexane- 2,6-dicarboxylic Acid (LY354740): Identification of Two New Potent, Selective, and Systemically Active Agonists for Group II Metabotropic Glutamate Receptors
Monn, James A, Valli, Matthew J, Massey, Steven M, Hansen, Marvin M, Kress, Thomas J, Wepsiec, James P, Harkness, Allen R, Grutsch, John L, Wright, Rebecca A, Johnson, Bryan G, Andis, Sherri L, Kingston, Ann, Tomlinson, Rosemarie, Lewis, Richard, Griffey, Kelly R, Tizzano, Joseph P, Schoepp, Darryle D
Published in Journal of medicinal chemistry (25.03.1999)
Published in Journal of medicinal chemistry (25.03.1999)
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Synthetic Studies Towards the Partial Ergot Alkaloid LY228729, a Potent 5HT1a Receptor Agonist
Carr, M. A, Creviston, P. E, Hutchison, D. R, Kennedy, J. H, Khau, V. V, Kress, T. J, Leanna, M. R, Marshall, J. D, Martinelli, Michael J, Peterson, B. C, Varie, D. L, Wepsiec, J. P
Published in Journal of organic chemistry (26.06.1998)
Published in Journal of organic chemistry (26.06.1998)
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Aromatase inhibition by 5-substituted pyrimidines and dihydropyrimidines
Taylor, Harold M, Jones, C. David, Davenport, James D, Hirsch, Kenneth S, Kress, T. J, Weaver, Dix
Published in Journal of medicinal chemistry (01.08.1987)
Published in Journal of medicinal chemistry (01.08.1987)
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Synthetic Studies toward the Partial Ergot Alkaloid LY228729, a Potent 5HT1A Receptor Agonist
Carr, M. A, Creviston, P. E, Hutchison, D. R, Kennedy, J. H, Khau, V. V, Kress, T. J, Leanna, M. R, Marshall, J. D, Martinelli, M. J, Peterson, B. C, Varie, D. L, Wepsiec, J. P
Published in Journal of organic chemistry (12.12.1997)
Published in Journal of organic chemistry (12.12.1997)
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The selective dehalogenation of 2,4-dichloro-5(2,4-dichlorodiphenylmethyl)pyrimidine
Campbell, J B, Whitehead, C W, Kress, T J, Moore, L L
Published in Annals of the New York Academy of Sciences (01.06.1973)
Published in Annals of the New York Academy of Sciences (01.06.1973)
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THE SYNTHESIS OF (+) AND (-)-1-BENZOYL-1,2,2A,3,4,5-HEXAHYDRO-BENZ[CD]INDOL-4-AMINE, AND PREPARATION OF LY228729
MARTINELLI, MJ, LEANNA, MR, VARIE, DL, PETERSON, BC, KRESS, TJ, WEPSIEC, JP, KHAU, VV
Published in Tetrahedron letters (01.01.1990)
Published in Tetrahedron letters (01.01.1990)
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Journal Article
Synthetic Studies toward the Partial Ergot Alkaloid LY228729, a Potent 5HT 1A Receptor Agonist
Carr, M. A., Creviston, P. E., Hutchison, D. R., Kennedy, J. H., Khau, V. V., Kress, T. J., Leanna, M. R., Marshall, J. D., Martinelli, M. J., Peterson, B. C., Varie, D. L., Wepsiec, J. P.
Published in Journal of organic chemistry (01.12.1997)
Published in Journal of organic chemistry (01.12.1997)
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Application of Palladium(0)-Catalyzed Processes to the Synthesis of Oxazole-Containing Partial Ergot Alkaloids
Anderson, Benjamin A, Becke, Lisa M, Booher, Richard N, Flaugh, Michael E, Harn, Nancy K, Kress, Thomas J, Varie, David L, Wepsiec, James P
Published in Journal of organic chemistry (12.12.1997)
Published in Journal of organic chemistry (12.12.1997)
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Synthetic studies toward the partial ergot alkaloid LY228729, a potent 5HT(1A) receptor agonist
Carr, MA, Creviston, PE, Hutchison, DR, Kennedy, JH, Khau, VV, Kress, TJ, Leanna, MR, Marshall, JD, Martinelli, MJ, Peterson, BC, Varie, DL, Wepsiec, JP
Published in Journal of organic chemistry (12.12.1997)
Published in Journal of organic chemistry (12.12.1997)
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Journal Article
Resolution of δ-Lactams Provides Access to Nonracemic Benzoquinolinones: The Synthesis of LY300502 and LY300503
Astleford, Bret A, Audia, James E, Deeter, Jack, Heath, Perry C, Janisse, Samantha K, Kress, Thomas J, Wepsiec, James P, Weigel, Leland O
Published in Journal of organic chemistry (26.06.1996)
Published in Journal of organic chemistry (26.06.1996)
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