Resiniferatoxin‐type phorboid vanilloids display capsaicin‐like selectivity at native vanilloid receptors on rat DRG neurons and at the cloned vanilloid receptor VR1
Szallasi, A, Szabó, T, Bíró, T, Modarres, S, Blumberg, P M, Krause, J E, Cortright, D N, Appendino, G
Published in British journal of pharmacology (01.09.1999)
Published in British journal of pharmacology (01.09.1999)
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A non‐pungent triprenyl phenol of fungal origin, scutigeral, stimulates rat dorsal root ganglion neurons via interaction at vanilloid receptors
Szallasi, A, Bíró, T, Szabó, T, Modarres, S, Petersen, M, Klusch, A, Blumberg, P M, Krause, J E, Sterner, O
Published in British journal of pharmacology (01.03.1999)
Published in British journal of pharmacology (01.03.1999)
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Nerve growth factor induces mechanical allodynia associated with novel A fibre-evoked spinal reflex activity and enhanced neurokinin-1 receptor activation in the rat
Thompson, S.W.N., Dray, A., McCarson, K.E., Krause, J.E., Urban, L.
Published in Pain (Amsterdam) (01.08.1995)
Published in Pain (Amsterdam) (01.08.1995)
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Effects of systemic resiniferatoxin treatment on substance P mRNA in rat dorsal root ganglia and substance P receptor mRNA in the spinal dorsal horn
Szallasi, Arpad, Farkas-Szallasi, Tünde, Tucker, Joseph B, Lundberg, Jan M, Hökfelt, Tomas, Krause, James E
Published in Brain research (09.01.1999)
Published in Brain research (09.01.1999)
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Structure, Functions, and Mechanisms of Substance P Receptor Action
Krause, James E, Takeda, Yasuo, Hershey, Andrew D
Published in Journal of investigative dermatology (01.06.1992)
Published in Journal of investigative dermatology (01.06.1992)
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Conference Proceeding
C5L2, a Nonsignaling C5A Binding Protein
Okinaga, Shoji, Slattery, Dubhfeasa, Humbles, Alison, Zsengeller, Zsusanna, Morteau, Olivier, Kinrade, Michele Bennett, Brodbeck, Robbin M, Krause, James E, Choe, Hye-Ryun, Gerard, Norma P, Gerard, Craig
Published in Biochemistry (Easton) (12.08.2003)
Published in Biochemistry (Easton) (12.08.2003)
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Distribution of mRNA for Vanilloid Receptor Subtype 1 (VR1), and VR1-Like Immunoreactivity, in the Central Nervous System of the Rat and Human
Mezey, Eva, Toth, Zsuzsanna E., Cortright, Daniel N., Arzubi, Michelle K., Krause, James E., Elde, Robert, Guo, Athena, Blumberg, Peter M., Szallasi, Arpad
Published in Proceedings of the National Academy of Sciences - PNAS (28.03.2000)
Published in Proceedings of the National Academy of Sciences - PNAS (28.03.2000)
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Regulation of the responses to gonadotropin-releasing hormone, muscarine and substance P in sympathetic neurons by changes in cellular constituents and intracellular application of peptide fragments of the substance P receptor
Simmons, M A, Schneider, C R, Krause, J E
Published in The Journal of pharmacology and experimental therapeutics (01.11.1994)
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Published in The Journal of pharmacology and experimental therapeutics (01.11.1994)
Journal Article
Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists
Blum, Charles A, Caldwell, Timothy, Zheng, Xiaozhang, Bakthavatchalam, Rajagopal, Capitosti, Scott, Brielmann, Harry, De Lombaert, Stéphane, Kershaw, Mark T, Matson, David, Krause, James E, Cortright, Daniel, Crandall, Marci, Martin, William J, Murphy, Beth Ann, Boyce, Susan, Jones, A. Brian, Mason, Glenn, Rycroft, Wayne, Perrett, Helen, Conley, Rachael, Burnaby-Davies, Nicola, Chenard, Bertrand L, Hodgetts, Kevin J
Published in Journal of medicinal chemistry (22.04.2010)
Published in Journal of medicinal chemistry (22.04.2010)
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Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites
Hodgetts, Kevin J., Blum, Charles A., Caldwell, Timothy, Bakthavatchalam, Rajagopal, Zheng, Xiaozhang, Capitosti, Scott, Krause, James E., Cortright, Daniel, Crandall, Marci, Murphy, Beth Ann, Boyce, Susan, Brian Jones, A., Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Substance P and its receptor neurokinin 1 expression in asthmatic airways
Chu, Hong Wei, Kraft, Monica, Krause, James E., Rex, Michael D., Martin, Richard J.
Published in Journal of allergy and clinical immunology (01.10.2000)
Published in Journal of allergy and clinical immunology (01.10.2000)
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