In Situ Selection of Lead Compounds by Click Chemistry: Target-Guided Optimization of Acetylcholinesterase Inhibitors
Krasiński, Antoni, Radić, Zoran, Manetsch, Roman, Raushel, Jessica, Taylor, Palmer, Sharpless, K. Barry, Kolb, Hartmuth C.
Published in Journal of the American Chemical Society (11.05.2005)
Published in Journal of the American Chemical Society (11.05.2005)
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CCR2 antagonist CCX140-B provides renal and glycemic benefits in diabetic transgenic human CCR2 knockin mice
Sullivan, Timothy, Miao, Zhenhua, Dairaghi, Daniel J, Krasinski, Antoni, Wang, Yu, Zhao, Bin N, Baumgart, Trageen, Ertl, Linda S, Pennell, Andrew, Seitz, Lisa, Powers, Jay, Zhao, Ruiping, Ungashe, Solomon, Wei, Zheng, Boring, Landin, Tsou, Chia-Lin, Charo, Israel, Berahovich, Robert D, Schall, Thomas J, Jaen, Juan C
Published in American journal of physiology. Renal physiology (01.11.2013)
Published in American journal of physiology. Renal physiology (01.11.2013)
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CCR2 antagonism leads to marked reduction in proteinuria and glomerular injury in murine models of focal segmental glomerulosclerosis (FSGS)
Miao, Zhenhua, Ertl, Linda S, Newland, Dale, Zhao, Bin, Wang, Yu, Zang, Xiaoping, Campbell, James J, Liu, Xiaoli, Dang, Ton, Miao, Shichang, Krasinski, Antoni, Punna, Sreenivas, Zeng, Yibin, McMahon, Jeffrey, Zhang, Penglie, Charo, Israel F, Schall, Thomas J, Singh, Rajinder
Published in PloS one (21.03.2018)
Published in PloS one (21.03.2018)
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Experimental evidence for the use of CCR2 antagonists in the treatment of type 2 diabetes
Sullivan, Timothy J, Miao, Zhenhua, Zhao, Bin N, Ertl, Linda S, Wang, Yu, Krasinski, Antoni, Walters, Matthew J, Powers, Jay P, Dairaghi, Daniel J, Baumgart, Trageen, Seitz, Lisa C, Berahovich, Robert D, Schall, Thomas J, Jaen, Juan C
Published in Metabolism, clinical and experimental (01.11.2013)
Published in Metabolism, clinical and experimental (01.11.2013)
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Immunosuppressive Myeloid Cells Induced by Chemotherapy Attenuate Antitumor CD4+ T-Cell Responses through the PD-1-PD-L1 Axis
DING, Zhi-Chun, XIAOYUN LU, BLAZAR, Bruce R, MELLOR, Andrew L, MUNN, David H, GANG ZHOU, MIAO YU, LEMOS, Henrique, LEI HUANG, CHANDLER, Phillip, KEBIN LIU, WALTERS, Matthew, KRASINSKI, Antoni, MACK, Matthias
Published in Cancer research (Chicago, Ill.) (01.07.2014)
Published in Cancer research (Chicago, Ill.) (01.07.2014)
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CCR2-Mediated Uptake of Constitutively Produced CCL2: A Mechanism for Regulating Chemokine Levels in the Blood
Zhao, Bin N, Campbell, James J, Salanga, Catherina L, Ertl, Linda S, Wang, Yu, Yau, Simon, Dang, Ton, Zeng, Yibin, McMahon, Jeffrey P, Krasinski, Antoni, Zhang, Penglie, Kufareva, Irina, Handel, Tracy M, Charo, Israel F, Singh, Rajinder, Schall, Thomas J
Published in The Journal of immunology (1950) (15.12.2019)
Published in The Journal of immunology (1950) (15.12.2019)
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Journal Article
Molecular basis of interactions of cholinesterases with tight binding inhibitors
Radić, Zoran, Manetsch, Roman, Krasiński, Antoni, Raushel, Jessica, Yamauchi, John, Garcia, Cindy, Kolb, Hartmuth, Sharpless, K. Barry, Taylor, Palmer
Published in Chemico-biological interactions (15.12.2005)
Published in Chemico-biological interactions (15.12.2005)
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Journal Article
FP240CCR2 INHIBITION IMPROVES RENAL FUNCTION IN MURINE MODELS OF CHRONIC KIDNEY DISEASE
Miao, Zhenhua, Ertl, Linda, Wang, Yu, Zhao, Bin, Zang, Xiaoping, Newland, Dale, Zeng, Yibin, Krasinski, Antoni, Mcmahon, Jeffrey, Liu, Xiaoli, Dang, Ton, Yau, Simon, Campbell, James, Miao, Shichang, Zhang, Penglie, Charo, Israel, Schall, Thomas, Singh, Rajinder
Published in Nephrology, dialysis, transplantation (01.06.2019)
Published in Nephrology, dialysis, transplantation (01.06.2019)
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Abstract 5655: Inhibition of CCR2 potentiates checkpoint inhibitor immunotherapy in murine model of pancreatic cancer
Janson, Christine, Jung, Heiyoun, Ertl, Linda, Liu, Shirley, Dang, Ton, Zeng, Yibin, Krasinski, Antoni, McMahon, Jeff, Zhang, Penglie, Charo, Israel, Singh, Rajinder, Schall, Thomas J.
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Tu1499 Efficacy of a Small Molecule CCR2 Antagonist in Experimental Model of Chronic Pancreatitis
Xue, Jing, Zhao, Qinglan, Sharma, Vishal, Kalisiak, Jaroslav, Zeng, Yibin, Krasinski, Antoni, Zhang, Penglie, McMahon, Jeff, Campbell, James J, Charo, Israel, Schall, Thomas, Habtezion, Aida
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
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Abstract 1745: Inhibition of chemokine receptor 2 (CCR2) with a small molecule antagonist enhances the effectiveness of checkpoint inhibition by altering the tumor microenvironment in mouse colorectal tumors: Reducing tumor size and increasing long term survival
Campbell, James J., Janson, Christine, Ertl, Linda, Li, Chris, Miao, Zhenhua, Krasinski, Antoni, Lui, Rebecca, Mali, Venkat, McMahon, Jeffrey, Zheng, Yibin, Wang, Yu, Zang, Xiaoping, Chhina, Vicky, Vilalta, Marta, Kumamoto, Alice, Dang, Ton, Liu, Shirley, Yao, Simon, Zhang, Penglie, Schall, Thomas J., Singh, Rajinder
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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