Search Results - "Konkel, Michael J" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Anxiolytic- and Antidepressant-like Profiles of the Galanin-3 Receptor ($Gal_3$) Antagonists SNAP 37889 and SNAP 398299

Anxiolytic- and Antidepressant-like Profiles of the Galanin-3 Receptor ($Gal_3$) Antagonists SNAP 37889 and SNAP 398299

by Chad J. Swanson, Thomas P. Blackburn, Xuexiang Zhang, Zheng, Kang, Xu, Zhi-Qing David, Hökfelt, Tomas, Toni D. Wolinsky, Michael J. Konkel, Heidi Chen, Huailing Zhong, Mary W. Walker, Craig, Douglas A., Christophe P. G. Gerald, Branchek, Theresa A.
Published in Proceedings of the National Academy of Sciences - PNAS (29.11.2005)

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Journal Article

3-Arylimino-2-indolones Are Potent and Selective Galanin GAL3 Receptor Antagonists

3-Arylimino-2-indolones Are Potent and Selective Galanin GAL3 Receptor Antagonists

by Konkel, Michael J, Lagu, Bharat, Boteju, Lakmal W, Jimenez, Hermogenes, Noble, Stewart, Walker, Mary W, Chandrasena, Gamini, Blackburn, Thomas P, Nikam, Sham S, Wright, Jon L, Kornberg, Brian E, Gregory, Tracy, Pugsley, Thomas A, Akunne, Hyacinth, Zoski, Kim, Wise, Lawrence D
Published in Journal of medicinal chemistry (29.06.2006)

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Journal Article

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal3 receptor binding affinity and improved solubility

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal3 receptor binding affinity and improved solubility

by KONKEL, Michael J, PACKIARAJAN, Mathivanan, HEIDI CHEN, TOPIWALA, Upendra P, JIMENEZ, Hermogenes, TALISMAN, Ian Jamie, COATE, Heather, WALKER, Mary W
Published in Bioorganic & medicinal chemistry letters (01.08.2006)

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Journal Article

Synthesis and Structure−Activity Relationship of Fluoro Analogues of 8-{2-[4-(4-Methoxyphenyl)piperazin-1yl]ethyl}-8-azaspiro[4.5]decane-7,9-dione as Selective α1d-Adrenergic Receptor Antagonists

Synthesis and Structure−Activity Relationship of Fluoro Analogues of 8-{2-[4-(4-Methoxyphenyl)piperazin-1yl]ethyl}-8-azaspiro[4.5]decane-7,9-dione as Selective α1d-Adrenergic Receptor Antagonists

by Konkel, Michael J, Wetzel, John M, Cahir, Marie, Craig, Douglas A, Noble, Stewart A, Gluchowski, Charles
Published in Journal of medicinal chemistry (21.04.2005)

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Palladium-Catalyzed Allylic Coupling of 1,2,3-Triazolo[4,5-d]pyrimidines (8-Azapurines)

Palladium-Catalyzed Allylic Coupling of 1,2,3-Triazolo[4,5-d]pyrimidines (8-Azapurines)

by Konkel, Michael J, Vince, Robert
Published in Journal of organic chemistry (06.09.1996)

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Journal Article

Structure Determination of the Products from the Acid-Catalyzed Condensation of Indole with Acetone

Structure Determination of the Products from the Acid-Catalyzed Condensation of Indole with Acetone

by Noland, Wayland E, Konkel, Michael J, Konkel, Lisa M. C, Pearce, Bradley C, Barnes, Charles L, Schlemper, Elmer O
Published in Journal of organic chemistry (26.01.1996)

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Journal Article

3-arylimino-2-indolones are potent and selective galanin GAL(3) receptor antagonists

3-arylimino-2-indolones are potent and selective galanin GAL(3) receptor antagonists

by Konkel, Michael J., Lagu, Bharat, Boteju, Lakmal W., Jimenez, Hermogenes, Noble, Stewart, Walker, Mary W., Chandrasena, Gamini, Blackburn, Thomas P., Nikam, Sham S., Wright, Jon L., Kornberg, Brian E., Gregory, Tracy, Pugsley, Thomas A., Akunne, Hyacinth, Zoski, Kim, Wise, Lawrence D.
Published in Journal of medicinal chemistry (29.06.2006)

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Journal Article

Synthesis and Structure−Activity Relationship of Fluoro Analogues of 8-{2-[4-(4-Methoxyphenyl)piperazin-1yl]ethyl}-8-azaspiro[4.5]decane-7,9-dione as Selective α 1d -Adrenergic Receptor Antagonists

Synthesis and Structure−Activity Relationship of Fluoro Analogues of 8-{2-[4-(4-Methoxyphenyl)piperazin-1yl]ethyl}-8-azaspiro[4.5]decane-7,9-dione as Selective α 1d -Adrenergic Receptor Antagonists

by Konkel, Michael J., Wetzel, John M., Cahir, Marie, Craig, Douglas A., Noble, Stewart A., Gluchowski, Charles
Published in Journal of medicinal chemistry (01.04.2005)

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Journal Article

Synthesis and structure-activity relationship of fluoro analogues of 8-{2-[4-(4-methoxyphenyl)piperazin-lyllethyl}-8-azaspiro[4.5]decane-7,9-dione as selective alpha(1d)-adrenergic receptor antagonists

Synthesis and structure-activity relationship of fluoro analogues of 8-{2-[4-(4-methoxyphenyl)piperazin-lyllethyl}-8-azaspiro[4.5]decane-7,9-dione as selective alpha(1d)-adrenergic receptor antagonists

by Konkel, MJ, Wetzel, JM, Cahir, M, Craig, DA, Noble, SA, Gluchowski, C
Published in Journal of medicinal chemistry (21.04.2005)

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Journal Article

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal 3 receptor binding affinity and improved solubility

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal 3 receptor binding affinity and improved solubility

by Konkel, Michael J., Packiarajan, Mathivanan, Chen, Heidi, Topiwala, Upendra P., Jimenez, Hermogenes, Talisman, Ian Jamie, Coate, Heather, Walker, Mary W.
Published in Bioorganic & medicinal chemistry letters (2006)

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Journal Article

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal sub(3) receptor binding affinity and improved solubility

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal sub(3) receptor binding affinity and improved solubility

by Konkel, Michael J, Packiarajan, Mathivanan, Chen, Heidi, Topiwala, Upendra P, Jimenez, Hermogenes, Talisman, Ian Jamie, Coate, Heather, Walker, Mary W
Published in Bioorganic & medicinal chemistry letters (01.01.2006)

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Journal Article

3-Arylimino-2-indolones Are Potent and Selective Galanin GAL 3 Receptor Antagonists

3-Arylimino-2-indolones Are Potent and Selective Galanin GAL 3 Receptor Antagonists

by Konkel, Michael J., Lagu, Bharat, Boteju, Lakmal W., Jimenez, Hermogenes, Noble, Stewart, Walker, Mary W., Chandrasena, Gamini, Blackburn, Thomas P., Nikam, Sham S., Wright, Jon L., Kornberg, Brian E., Gregory, Tracy, Pugsley, Thomas A., Akunne, Hyacinth, Zoski, Kim, Wise, Lawrence D.
Published in Journal of medicinal chemistry (01.06.2006)

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Journal Article

3-arylimino-2-indolones are potent and selective galanin GAL3receptor antagonists

3-arylimino-2-indolones are potent and selective galanin GAL3receptor antagonists

by KONKEL, Michael J, LAGU, Bharat, KORNBERG, Brian E, GREGORY, Tracy, PUGSLEY, Thomas A, AKUNNE, Hyacinth, ZOSKI, Kim, WISE, Lawrence D, BOTEJU, Lakmal W, JIMENEZ, Hermogenes, NOBLE, Stewart, WALKER, Mary W, CHANDRASENA, Gamini, BLACKBURN, Thomas P, NIKAM, Sham S, WRIGHT, Jon L
Published in Journal of medicinal chemistry (2006)

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Journal Article

Anxiolytic- and antidepressant-like profiles of the galanin-3 receptor (Gal 3 ) antagonists SNAP 37889 and SNAP 398299 (vol 102, pg 14789, 2005)

Anxiolytic- and antidepressant-like profiles of the galanin-3 receptor (Gal 3 ) antagonists SNAP 37889 and SNAP 398299 (vol 102, pg 14789, 2005)

by Swanson, CJ, Blackburn, TP, Zhang, XX, Zheng, K, Xu, ZQD, Hokfelt, T, Wolinsky, TD, Konkel, MJ, Chen, HD, Zhong, HL, Walker, MW, Craig, DA, Gerald, CPG, Branchek, TA
Published in Proceedings of the National Academy of Sciences - PNAS (03.10.2006)

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Journal Article

Cyclohexenyl nucleosides: Synthesis of cis-4-(9 H-purin-9-yl)-2-cyclohexenylcarbinols

Cyclohexenyl nucleosides: Synthesis of cis-4-(9 H-purin-9-yl)-2-cyclohexenylcarbinols

by Konkel, Michael J., Vince, Robert
Published in Tetrahedron (15.01.1996)

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Journal Article

Cyclohexenyl nucleosides: Synthesis and biological activity of trans-3-(purin-9-yl)-4-cyclohexenylcarbinols

Cyclohexenyl nucleosides: Synthesis and biological activity of trans-3-(purin-9-yl)-4-cyclohexenylcarbinols

by Konkel, Michael J., Vince, Robert
Published in Tetrahedron (01.07.1996)

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Journal Article

In situ vinylindole synthesis. Diels-Alder reactions with maleic anhydride and maleic acid to give tetrahydrocarbazoles and carbazoles

In situ vinylindole synthesis. Diels-Alder reactions with maleic anhydride and maleic acid to give tetrahydrocarbazoles and carbazoles

by Noland, Wayland E., Xia, Guang-Ming, Gee, Kyle R., Konkel, Michael J., Wahlstrom, Mary J., Condoluci, John J., Rieger, Dale L.
Published in Tetrahedron (25.03.1996)

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Journal Article

The crystal structure of a novel product from the acid-catalyzed condensation of 1-benzylindole with acetone

The crystal structure of a novel product from the acid-catalyzed condensation of 1-benzylindole with acetone

by NOLAND, W. E, KONKEL, M. J, FANBURG, S. J, VENKATRAMAN, S, BRITTON, D
Published in Journal of chemical crystallography (1999)

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Journal Article

USE OF GAL3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF DEPRESSION AND/OR ANXIETY AND COMPOUNDS USEFUL IN SUCH METHODS

USE OF GAL3 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF DEPRESSION AND/OR ANXIETY AND COMPOUNDS USEFUL IN SUCH METHODS

by PACKIARAJAN, MATHIVANAN, CHEN, HEIDI, JIMENEZ, HERMO, LAGU, BHARAT, BLACKBURN, THOMAS P, BOTEJU, LAKMAL, WETZEL, JOHN M, NOBLE, STEWART, KONKEL, MICHAEL J, LIM, KITAE, TALISMAN, IAN JAMIE
Year of Publication 26.06.2012

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Patent

Amino Substituted Analogues of 1-Phenyl-3-phenylimino-2-indolones with Potent Galanin GaI3 Receptor Binding Affinity and Improved Solubility

Amino Substituted Analogues of 1-Phenyl-3-phenylimino-2-indolones with Potent Galanin GaI3 Receptor Binding Affinity and Improved Solubility

by Konkel, Michael J., Packiarajan, Mathivanan, Chen, Heidi, Topiwala, Upendra P., Jimenez, Hermogenes, Talisman, Ian Jamie, Coate, Heather, Walker, Mary W.
Published in ChemInform (07.11.2006)

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Journal Article