Rapid and Robust Multi-Phenotypic Assay System for ALS Using Human iPS Cells with Mutations in Causative Genes
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Published in International journal of molecular sciences (01.04.2023)
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Differential Effects of 2-Hydroxypropyl-Cyclodextrins on Lipid Accumulation in Npc1 -Null Cells
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Published in International journal of molecular sciences (30.01.2020)
Published in International journal of molecular sciences (30.01.2020)
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Discovery of a 1‑Methyl-3,4-dihydronaphthalene-Based Sphingosine-1-Phosphate (S1P) Receptor Agonist Ceralifimod (ONO-4641). A S1P1 and S1P5 Selective Agonist for the Treatment of Autoimmune Diseases
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Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Sphingosine 1-phosphate receptor modulator ONO-4641 stimulates CD11b + Gr-1 + cell expansion and inhibits lymphocyte infiltration in the lungs to ameliorate murine pulmonary emphysema
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Published in Mucosal immunology (01.11.2018)
Published in Mucosal immunology (01.11.2018)
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A sphingosine 1-phosphate receptor agonist ameliorates animal model of vasculitis
Miyabe, Chie, Miyabe, Yoshishige, Komiya, Takaki, Shioya, Hiroki, Miura, Noriko N., Takahashi, Kei, Ohno, Naohito, Tsuboi, Ryoji, Luster, Andrew D., Kawai, Shinichi, Miyasaka, Nobuyuki, Nanki, Toshihiro
Published in Inflammation research (01.04.2017)
Published in Inflammation research (01.04.2017)
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Sphingosine 1-Phosphate Receptor Modulator ONO-4641 Regulates Trafficking of T Lymphocytes and Hematopoietic Stem Cells and Alleviates Immune-Mediated Aplastic Anemia in a Mouse Model
Komiya, Takaki, Gohda, Masashi, Shioya, Hiroki, Katsumata, Seishi
Published in The Journal of pharmacology and experimental therapeutics (01.02.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2021)
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Discovery of a 1-Methyl-3,4-dihydronaphthalene-Based Sphingosine-1-Phosphate (S1P) Receptor Agonist Ceralifimod (ONO-4641). A S1P(1) and S1P(5) Selective Agonist for the Treatment of Autoimmune Diseases
Kurata, Haruto, Kusumi, Kensuke, Otsuki, Kazuhiro, Suzuki, Ryo, Kurono, Masakuni, Komiya, Takaki, Hagiya, Hiroshi, Mizuno, Hirotaka, Shioya, Hiroki, Ono, Takeji, Takada, Yuka, Maeda, Tatsuo, Matsunaga, Norikazu, Kondo, Tetsu, Tominaga, Sachiko, Nunoya, Ken-Ici, Kiyoshi, Hidekazu, Komeno, Masaharu, Nakade, Shinji, Habashita, Hiromu
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Journal Article
Discovery of a 1-Methyl-3,4-dihydronaphthalene-Based Sphingosine-1-Phosphate (S1P) Receptor Agonist Ceralifimod (ONO-4641). A S1P 1 and S1P 5 Selective Agonist for the Treatment of Autoimmune Diseases
Kurata, Haruto, Kusumi, Kensuke, Otsuki, Kazuhiro, Suzuki, Ryo, Kurono, Masakuni, Komiya, Takaki, Hagiya, Hiroshi, Mizuno, Hirotaka, Shioya, Hiroki, Ono, Takeji, Takada, Yuka, Maeda, Tatsuo, Matsunaga, Norikazu, Kondo, Tetsu, Tominaga, Sachiko, Nunoya, Ken-Ici, Kiyoshi, Hidekazu, Komeno, Masaharu, Nakade, Shinji, Habashita, Hiromu
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR S1P5-MEDIATED DISEASES
KOMIYA TAKAKI, WATANABE TOSHIHIDE, TSUBURAYA NAOMI, KUSUMI KENSUKE, IMAIDE SATOMI, ENDO TOSHIMITSU
Year of Publication 04.03.2021
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Year of Publication 04.03.2021
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S1P5 수용체 작동 활성을 갖는 화합물
KOMIYA TAKAKI, WATANABE TOSHIHIDE, TSUBURAYA NAOMI, KUSUMI KENSUKE, IMAIDE SATOMI, ENDO TOSHIMITSU
Year of Publication 03.11.2020
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Year of Publication 03.11.2020
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Suppressive effects of a novel CC chemokine receptor 4 antagonist on Th2 cell trafficking in ligand- and antigen-induced mouse models
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Published in European journal of pharmacology (15.11.2013)
Published in European journal of pharmacology (15.11.2013)
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COMPOUND HAVING S1P5 RECEPTOR AGONIST ACTIVITY
KUSUMI, Kensuke, TSUBURAYA, Naomi, IMAIDE, Satomi, ENDO, Toshimitsu, KOMIYA, Takaki, WATANABE, Toshihide
Year of Publication 29.08.2019
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Year of Publication 29.08.2019
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Structure–activity relationship studies of S1P agonists with a dihydronaphthalene scaffold
Kurata, Haruto, Kusumi, Kensuke, Otsuki, Kazuhiro, Suzuki, Ryo, Kurono, Masakuni, Tokuda, Natsuko, Takada, Yuka, Shioya, Hiroki, Mizuno, Hirotaka, Komiya, Takaki, Ono, Takeji, Hagiya, Hiroshi, Minami, Masashi, Nakade, Shinji, Habashita, Hiromu
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Discovery of S1P agonists with a dihydronaphthalene scaffold
Kurata, Haruto, Kusumi, Kensuke, Otsuki, Kazuhiro, Suzuki, Ryo, Kurono, Masakuni, Takada, Yuka, Shioya, Hiroki, Komiya, Takaki, Mizuno, Hirotaka, Ono, Takeji, Hagiya, Hiroshi, Minami, Masashi, Nakade, Shinji, Habashita, Hiromu
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
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S1P RECEPTOR BINDING-ABILITY POSSESSING COMPOUND AND MEDICAL USE THEREOF
KURATA HARUTO, HABASHITA HIROSHI, MIZUNO HIROKI, ONO TAKEJI, KOMIYA TAKAKI, SAGA HIROSHI, NAKADE SHINJI, OTSUKI KAZUHIRO, KUSUMI KENSUKE, MINAMI SHINJI, HAGIYA HIROSHI
Year of Publication 25.12.2014
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Year of Publication 25.12.2014
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1-[[(3S)-3-METHYL-6-(4(4,4-TRIFLUOROBUTOXY)-3,4-DIHYDRONAPHTHALEN-2YL]METHYL]AZETIDINE-3-CARBOXYLIC ACID HAVING S1P5 RECEPTOR AGONIST ACTIVITY FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS AND CANCER
KUSUMI, Kensuke, TSUBURAYA, Naomi, IMAIDE, Satomi, ENDO, Toshimitsu, KOMIYA, Takaki, WATANABE, Toshihide
Year of Publication 28.08.2024
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Year of Publication 28.08.2024
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Compounds having S1P5 receptor agonistic activity
Watanabe, Toshihide, Kusumi, Kensuke, Tsuburaya, Naomi, Endo, Toshimitsu, Imaide, Satomi, Komiya, Takaki
Year of Publication 30.07.2024
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Year of Publication 30.07.2024
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Compound having S1P5 receptor agonist activity
KUSUMI, Kensuke, TSUBURAYA, Naomi, IMAIDE, Satomi, ENDO, Toshimitsu, KOMIYA, Takaki, WATANABE, Toshihide
Year of Publication 27.06.2024
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Year of Publication 27.06.2024
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