The 5‐lipoxygenase inhibitor, zileuton, suppresses prostaglandin biosynthesis by inhibition of arachidonic acid release in macrophages
Rossi, A, Pergola, C, Koeberle, A, Hoffmann, M, Dehm, F, Bramanti, P, Cuzzocrea, S, Werz, O, Sautebin, L
Published in British journal of pharmacology (01.10.2010)
Published in British journal of pharmacology (01.10.2010)
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Journal Article
Docosahexaenoic acid in the treatment of rheumatoid arthritis: A double-blind, placebo-controlled, randomized cross-over study with microalgae vs . sunflower oil
Dawczynski, C, Dittrich, M, Neumann, T, Goetze, K, Welzel, A, Oelzner, P, Völker, S, Schaible, A.M, Troisi, F, Thomas, L, Pace, S, Koeberle, A, Werz, O, Schlattmann, P, Lorkowski, S, Jahreis, G
Published in Clinical nutrition (Edinburgh, Scotland) (01.04.2018)
Published in Clinical nutrition (Edinburgh, Scotland) (01.04.2018)
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Journal Article
Myrtucommulone, a natural acylphloroglucinol, inhibits microsomal prostaglandin E 2 synthase‐1
Koeberle, A, Pollastro, F, Northoff, H, Werz, O
Published in British journal of pharmacology (01.03.2009)
Published in British journal of pharmacology (01.03.2009)
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Journal Article
Inhibition of microsomal prostaglandin E 2 synthase‐1 as a molecular basis for the anti‐inflammatory actions of boswellic acids from frankincense
Siemoneit, U, Koeberle, A, Rossi, A, Dehm, F, Verhoff, M, Reckel, S, Maier, TJ, Jauch, J, Northoff, H, Bernhard, F, Doetsch, V, Sautebin, L, Werz, O
Published in British journal of pharmacology (01.01.2011)
Published in British journal of pharmacology (01.01.2011)
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Journal Article
High capacity for leukotriene biosynthesis in peripheral blood during pregnancy
Schaible, A.M, Koeberle, A, Northoff, H, Lawrenz, B, Weinigel, C, Barz, D, Werz, O, Pergola, C
Published in Prostaglandins, leukotrienes and essential fatty acids (01.09.2013)
Published in Prostaglandins, leukotrienes and essential fatty acids (01.09.2013)
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Journal Article
Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4‐benzoquinone that inhibits 5‐lipoxygenase
Schaible, A M, Filosa, R, Temml, V, Krauth, V, Matteis, M, Peduto, A, Bruno, F, Luderer, S, Roviezzo, F, Di Mola, A, Rosa, M, D'Agostino, B, Weinigel, C, Barz, D, Koeberle, A, Pergola, C, Schuster, D, Werz, O
Published in British journal of pharmacology (01.05.2014)
Published in British journal of pharmacology (01.05.2014)
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Journal Article
Myrtucommulone, a natural acylphloroglucinol, inhibits microsomal prostaglandin E2 synthase‐1
Koeberle, A, Pollastro, F, Northoff, H, Werz, O
Published in British journal of pharmacology (01.03.2009)
Published in British journal of pharmacology (01.03.2009)
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Journal Article
Targeting biosynthetic networks of the proinflammatory and proresolving lipid metabolome
Werner, Markus, Jordan, Paul M, Romp, Erik, Czapka, Anna, Rao, Zhigang, Kretzer, Christian, Koeberle, Andreas, Garscha, Ulrike, Pace, Simona, Claesson, Hans-Erik, Serhan, Charles N, Werz, Oliver, Gerstmeier, Jana
Published in The FASEB journal (01.05.2019)
Published in The FASEB journal (01.05.2019)
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Journal Article
599 Amelioration of symptoms of dry and eczema-prone skin by an oil-in-water emulsion containing a combination of a zingiber officinale root extract and cbd with antioxidative and anti-inflammatory activity in vitro
Soeberdt, M., Neubauer, C., Kragl, M., Mähler, N., Moritz, K., Hoch, S., Steindl, H., Filipek, P., Bonyadirad, E., Jakschitz, T., Koeberle, A., Bonn, G., Abels, C.
Published in Journal of investigative dermatology (01.05.2023)
Published in Journal of investigative dermatology (01.05.2023)
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Journal Article
262 Canephron® N reduces pain in experimental cystitis and prostatitis putatively by inhibition of PGE2 production
Nausch, B, Koeberle, A, Werz, O, Ammendola, A, Künstle, G
Published in European urology supplements : official journal of the European Association of Urology (01.03.2016)
Published in European urology supplements : official journal of the European Association of Urology (01.03.2016)
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Journal Article
Androgen-mediated sex bias impairs efficiency of leukotriene biosynthesis inhibitors in males
Pace, Simona, Pergola, Carlo, Dehm, Friederike, Rossi, Antonietta, Gerstmeier, Jana, Troisi, Fabiana, Pein, Helmut, Schaible, Anja M, Weinigel, Christina, Rummler, Silke, Northoff, Hinnak, Laufer, Stefan, Maier, Thorsten J, Rådmark, Olof, Samuelsson, Bengt, Koeberle, Andreas, Sautebin, Lidia, Werz, Oliver
Published in The Journal of clinical investigation (01.08.2017)
Published in The Journal of clinical investigation (01.08.2017)
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Journal Article
P068 Polyunsaturated fatty acid excess fuels pro-inflammatory transcriptional networks in GPX4 deficient intestinal epithelial cells
Meyer, M, Grabherr, F, Schwärzler, J, Mayr, L, Jukic, A, Rao, Z, Rieder, D, Zollner, A, Grander, C, Trajanoski, Z, Koeberle, A, Tilg, H, Adolph, T E
Published in Journal of Crohn's and colitis (30.01.2023)
Published in Journal of Crohn's and colitis (30.01.2023)
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Journal Article
Lipophilic extracts of Leucas zeylanica, a multi-purpose medicinal plant in the tropics, inhibit key enzymes involved in inflammation and gout
Napagoda, Mayuri, Gerstmeier, Jana, Butschek, Hannah, Lorenz, Sybille, Kanatiwela, Dinusha, Qader, Mallique, Nagahawatte, Ajith, De Soyza, Sudhara, Wijayaratne, Gaya Bandara, Svatoš, Aleš, Jayasinghe, Lalith, Koeberle, Andreas, Werz, Oliver
Published in Journal of ethnopharmacology (05.10.2018)
Published in Journal of ethnopharmacology (05.10.2018)
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Journal Article
Otolith shape as a classification tool for Chinook salmon (Oncorhynchus tshawytscha) discrimination in native and introduced systems
Koeberle, Alexander L, Arismendi, Ivan, Crittenden, Whitney, Di Prinzio, Cecilia, Gomez-Uchida, Daniel, Noakes, David L.G, Richardson, Shannon
Published in Canadian journal of fisheries and aquatic sciences (01.07.2020)
Published in Canadian journal of fisheries and aquatic sciences (01.07.2020)
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Journal Article
Triterpene Acids from Frankincense and Semi-Synthetic Derivatives That Inhibit 5-Lipoxygenase and Cathepsin G
Koeberle, Andreas, Henkel, Arne, Verhoff, Moritz, Tausch, Lars, König, Stefanie, Fischer, Dagmar, Kather, Nicole, Seitz, Stefanie, Paul, Michael, Jauch, Johann, Werz, Oliver
Published in Molecules (Basel, Switzerland) (24.02.2018)
Published in Molecules (Basel, Switzerland) (24.02.2018)
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Journal Article
OP0151 Docosahexaenoic acid treatment of rheumatoid arthritis: a randomized, double-blind, placebo-controlled, cross-over study
Neumann, T, Dawczynski, C, Dittrich, M, Goetze, K, Welzel, A, Oelzner, P, Voelker, S, Schaible, AM, Troisi, F, Thomas, L, Pace, S, Koeberle, A, Werz, O, Schlattmann, P, Lorkowski, S, Jahreis, G
Published in Annals of the rheumatic diseases (01.06.2017)
Published in Annals of the rheumatic diseases (01.06.2017)
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Journal Article
Hyperforin is a novel type of 5-lipoxygenase inhibitor with high efficacy in vivo
Feißt, Christian, Pergola, Carlo, Rakonjac, Marija, Rossi, Antonietta, Koeberle, Andreas, Dodt, Gabriele, Hoffmann, Marika, Hoernig, Christina, Fischer, Lutz, Steinhilber, Dieter, Franke, Lutz, Schneider, Gisbert, Rådmark, Olof, Sautebin, Lidia, Werz, Oliver
Published in Cellular and molecular life sciences : CMLS (01.08.2009)
Published in Cellular and molecular life sciences : CMLS (01.08.2009)
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Journal Article
Computational investigation of multi-target effects in the arachidonic acid cascade on the example of potent natural 5-LO inhibitor garcinoic acid
Temml, V, Pein, H, Pace, S, Garscha, U, Waltenberger, B, Roviezzo, F, Helesbeux, JJ, Séraphin, D, Rossi, A, Lorkowski, S, Richomme, P, Werz, O, Koeberle, A, Schuster, D, Stuppner, H
Published in Planta Medica (01.12.2019)
Published in Planta Medica (01.12.2019)
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Conference Proceeding
Green tea epigallocatechin-3-gallate inhibits microsomal prostaglandin E sub(2) synthase-1
Koeberle, A, Bauer, J, Verhoff, M, Hoffmann, M, Northoff, H, Werz, O
Published in Biochemical and biophysical research communications (16.10.2009)
Published in Biochemical and biophysical research communications (16.10.2009)
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