Late‐Stage Functionalization of Histidine in Unprotected Peptides
Noisier, Anaïs F. M., Johansson, Magnus J., Knerr, Laurent, Hayes, Martin A., Drury, William J., Valeur, Eric, Malins, Lara R., Gopalakrishnan, Ranganath
Published in Angewandte Chemie International Edition (19.12.2019)
Published in Angewandte Chemie International Edition (19.12.2019)
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Glucagon Like Peptide 1 Receptor Agonists for Targeted Delivery of Antisense Oligonucleotides to Pancreatic Beta Cell
Knerr, Laurent, Prakash, Thazha P, Lee, Richard, Drury III, William J, Nikan, Mehran, Fu, Wuxia, Pirie, Elaine, Maria, Leonardo De, Valeur, Eric, Hayen, Ahlke, Ölwegård-Halvarsson, Maria, Broddefalk, Johan, Ämmälä, Carina, Østergaard, Michael E, Meuller, Johan, Sundström, Linda, Andersson, Patrik, Janzén, David, Jansson-Löfmark, Rasmus, Seth, Punit P, Andersson, Shalini
Published in Journal of the American Chemical Society (10.03.2021)
Published in Journal of the American Chemical Society (10.03.2021)
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IA-Lab: A MATLAB framework for efficient microscopy image analysis development, applied to quantifying intracellular transport of internalized peptide-drug conjugate
Corrigan, Adam M, Karlsson, Johan, Wildenhain, Jan, Knerr, Laurent, Ölwegård-Halvarsson, Maria, Karlsson, Maria, Lünse, Svenja, Wang, Yinhai
Published in PloS one (01.08.2019)
Published in PloS one (01.08.2019)
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Discovery of AZD2716: A Novel Secreted Phospholipase A2 (sPLA2) Inhibitor for the Treatment of Coronary Artery Disease
Giordanetto, Fabrizio, Pettersen, Daniel, Starke, Ingemar, Nordberg, Peter, Dahlström, Mikael, Knerr, Laurent, Selmi, Nidhal, Rosengren, Birgitta, Larsson, Lars-Olof, Sandmark, Jenny, Castaldo, Marie, Dekker, Niek, Karlsson, Ulla, Hurt-Camejo, Eva
Published in ACS medicinal chemistry letters (13.10.2016)
Published in ACS medicinal chemistry letters (13.10.2016)
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Stapled Vasoactive Intestinal Peptide (VIP) Derivatives Improve VPAC2 Agonism and Glucose-Dependent Insulin Secretion
Giordanetto, Fabrizio, Revell, Jefferson D, Knerr, Laurent, Hostettler, Marie, Paunovic, Amalia, Priest, Claire, Janefeldt, Annika, Gill, Adrian
Published in ACS medicinal chemistry letters (12.12.2013)
Published in ACS medicinal chemistry letters (12.12.2013)
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Exploring physicochemical space via a bioisostere of the trifluoromethyl and ethyl groups (BITE): attenuating lipophilicity in fluorinated analogues of Gilenya (R) for multiple sclerosis
Erdeljac, Nathalie, Kehr, Gerald, Ahlqvist, Marie, Knerr, Laurent, Gilmour, Ryan
Published in Chemical communications (Cambridge, England) (23.10.2018)
Published in Chemical communications (Cambridge, England) (23.10.2018)
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The Conundrum of GSK3 Inhibitors: Is it the Dawn of a New Beginning?
Bhat, Ratan V, Andersson, Ulf, Andersson, Shalini, Knerr, Laurent, Bauer, Udo, Sundgren-Andersson, Anna K
Published in Journal of Alzheimer's disease (01.01.2018)
Published in Journal of Alzheimer's disease (01.01.2018)
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Exploring physicochemical space via a bioisostere of the trifluoromethyl and ethyl groups (BITE): attenuating lipophilicity in fluorinated analogues of Gilenya® for multiple sclerosisElectronic supplementary information (ESI) available. See DOI: 10.1039/c8cc05643a
Erdeljac, Nathalie, Kehr, Gerald, Ahlqvist, Marie, Knerr, Laurent, Gilmour, Ryan
Year of Publication 23.10.2018
Year of Publication 23.10.2018
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Journal Article
Late-Stage Functionalization with Cysteine Staples Generates Potent and Selective Melanocortin Receptor‑1 Agonists
White, Andrew M., Dellsén, Anita, Larsson, Niklas, Kaas, Quentin, Jansen, Frank, Plowright, Alleyn T., Knerr, Laurent, Durek, Thomas, Craik, David J.
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Stereocontrolled Synthesis of Tetrafluoropentanols: Multivicinal Fluorinated Alkane Units for Drug Discovery
Bentler, Patrick, Erdeljac, Nathalie, Bussmann, Kathrin, Ahlqvist, Marie, Knerr, Laurent, Bergander, Klaus, Daniliuc, Constantin G, Gilmour, Ryan
Published in Organic letters (04.10.2019)
Published in Organic letters (04.10.2019)
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A structure-specific small molecule inhibits a miRNA-200 family member precursor and reverses a type 2 diabetes phenotype
Haniff, Hafeez S., Liu, Xiaohui, Tong, Yuquan, Meyer, Samantha M., Knerr, Laurent, Lemurell, Malin, Abegg, Daniel, Aikawa, Haruo, Adibekian, Alexander, Disney, Matthew D.
Published in Cell chemical biology (17.02.2022)
Published in Cell chemical biology (17.02.2022)
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Incorporation of Intracellular NanoSIMS Tracers to Oligonucleotide Conjugates via Strain Promoted Sydnone–Alkyne Cycloaddition
Lincy-Bianchi, Loujahine, Häfner, Maximilian, Becquart, Cécile, Tängemo, Carolina, Kurczy, Michael E., Munier, Claire C., Knerr, Laurent
Published in Bioconjugate chemistry (17.07.2024)
Published in Bioconjugate chemistry (17.07.2024)
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Design of a small molecule that stimulates vascular endothelial growth factor A enabled by screening RNA fold-small molecule interactions
Haniff, Hafeez S, Knerr, Laurent, Liu, Xiaohui, Crynen, Gogce, Boström, Jonas, Abegg, Daniel, Adibekian, Alexander, Lekah, Elizabeth, Wang, Kye Won, Cameron, Michael D, Yildirim, Ilyas, Lemurell, Malin, Disney, Matthew D
Published in Nature chemistry (01.10.2020)
Published in Nature chemistry (01.10.2020)
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Fluorine‐Directed Glycosylation Enables the Stereocontrolled Synthesis of Selective SGLT2 Inhibitors for Type II Diabetes
Sadurní, Anna, Kehr, Gerald, Ahlqvist, Marie, Wernevik, Johan, Sjögren, Helena Peilot, Kankkonen, Cecilia, Knerr, Laurent, Gilmour, Ryan
Published in Chemistry : a European journal (26.02.2018)
Published in Chemistry : a European journal (26.02.2018)
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