Medicinal Chemistry and Therapeutic Potential of Agonists, Antagonists and Allosteric Modulators of A1 Adenosine Receptor: Current Status and Perspectives
Deb, Pran Kishore, Deka, Satyendra, Borah, Pobitra, Abed, Sara N, Klotz, Karl-Norbert
Published in Current pharmaceutical design (2019)
Published in Current pharmaceutical design (2019)
Get more information
Journal Article
Pharmacological characterisation of novel adenosine A3 receptor antagonists
Barkan, Kerry, Lagarias, Panagiotis, Stampelou, Margarita, Stamatis, Dimitrios, Hoare, Sam, Safitri, Dewi, Klotz, Karl-Norbert, Vrontaki, Eleni, Kolocouris, Antonios, Ladds, Graham
Published in Scientific reports (27.11.2020)
Published in Scientific reports (27.11.2020)
Get full text
Journal Article
7‐Amino‐2‐aryl/hetero‐aryl‐5‐oxo‐5,8‐dihydro[1,2,4]triazolo[1,5‐a]pyridine‐6‐carbonitriles: Synthesis and adenosine receptor binding studies
Shaik, Khasim, Deb, Pran Kishore, Mailavaram, Raghu Prasad, Chandrasekaran, Balakumar, Kachler, Sonja, Klotz, Karl‐Norbert, Jaber, Abdul Muttaleb Yousef
Published in Chemical biology & drug design (01.08.2019)
Published in Chemical biology & drug design (01.08.2019)
Get full text
Journal Article
Neuroprotective potential of adenosine A 1 receptor partial agonists in experimental models of cerebral ischemia
Martire, Alberto, Lambertucci, Catia, Pepponi, Rita, Ferrante, Antonella, Benati, Nicholas, Buccioni, Michela, Dal Ben, Diego, Marucci, Gabriella, Klotz, Karl-Norbert, Volpini, Rosaria, Popoli, Patrizia
Published in Journal of neurochemistry (01.04.2019)
Published in Journal of neurochemistry (01.04.2019)
Get full text
Journal Article
Synthesis, adenosine receptor binding and molecular modelling studies of novel thieno[2,3‐d]pyrimidine derivatives
Deb, Pran Kishore, Mailavaram, Raghuprasad, Chandrasekaran, Balakumar, Kaki, Venkata Rao, Kaur, Rajwinder, Kachler, Sonja, Klotz, Karl‐Norbert, Akkinepally, Raghuram Rao
Published in Chemical biology & drug design (01.04.2018)
Published in Chemical biology & drug design (01.04.2018)
Get full text
Journal Article
Analysis of receptor oligomerization by FRAP microscopy
Bünemann, Moritz, Engelhardt, Stefan, Klotz, Karl-Norbert, Lohse, Martin J, Dorsch, Sandra
Published in Nature methods (01.03.2009)
Published in Nature methods (01.03.2009)
Get full text
Journal Article
Targeting G Protein‐Coupled Receptors with Magnetic Carbon Nanotubes: The Case of the A3 Adenosine Receptor
Pineux, Florent, Federico, Stephanie, Klotz, Karl‐Norbert, Kachler, Sonja, Michiels, Carine, Sturlese, Mattia, Prato, Maurizio, Spalluto, Giampiero, Moro, Stefano, Bonifazi, Davide
Published in ChemMedChem (19.10.2020)
Published in ChemMedChem (19.10.2020)
Get full text
Journal Article
Adenosine Receptor Ligands: Coumarin–Chalcone Hybrids as Modulating Agents on the Activity of hARs
Vazquez-Rodriguez, Saleta, Vilar, Santiago, Kachler, Sonja, Klotz, Karl-Norbert, Uriarte, Eugenio, Borges, Fernanda, Matos, Maria João
Published in Molecules (Basel, Switzerland) (19.09.2020)
Published in Molecules (Basel, Switzerland) (19.09.2020)
Get full text
Journal Article
Discovery of Novel Adenosine Receptor Antagonists through a Combined Structure- and Ligand-Based Approach Followed by Molecular Dynamics Investigation of Ligand Binding Mode
Lagarias, Panagiotis, Vrontaki, Eleni, Lambrinidis, George, Stamatis, Dimitrios, Convertino, Marino, Ortore, Gabriella, Mavromoustakos, Thomas, Klotz, Karl-Norbert, Kolocouris, Antonios
Published in Journal of chemical information and modeling (23.04.2018)
Published in Journal of chemical information and modeling (23.04.2018)
Get full text
Journal Article
A2A Adenosine Receptor Antagonists: Are Triazolotriazine and Purine Scaffolds Interchangeable?
Spinaci, Andrea, Lambertucci, Catia, Buccioni, Michela, Dal Ben, Diego, Graiff, Claudia, Barbalace, Maria Cristina, Hrelia, Silvana, Angeloni, Cristina, Tayebati, Seyed Khosrow, Ubaldi, Massimo, Masi, Alessio, Klotz, Karl-Norbert, Volpini, Rosaria, Marucci, Gabriella
Published in Molecules (Basel, Switzerland) (07.04.2022)
Published in Molecules (Basel, Switzerland) (07.04.2022)
Get full text
Journal Article
Discovery of indolylpiperazinylpyrimidines with dual-target profiles at adenosine A2A and dopamine D2 receptors for Parkinson's disease treatment
Shao, Yi-Ming, Ma, Xiaohua, Paira, Priyankar, Tan, Aaron, Herr, Deron Raymond, Lim, Kah Leong, Ng, Chee Hoe, Venkatesan, Gopalakrishnan, Klotz, Karl-Norbert, Federico, Stephanie, Spalluto, Giampiero, Cheong, Siew Lee, Chen, Yu Zong, Pastorin, Giorgia
Published in PloS one (01.01.2018)
Published in PloS one (01.01.2018)
Get full text
Journal Article
Neuroprotective potential of adenosine A1 receptor partial agonists in experimental models of cerebral ischemia
Martire, Alberto, Lambertucci, Catia, Pepponi, Rita, Ferrante, Antonella, Benati, Nicholas, Buccioni, Michela, Dal Ben, Diego, Marucci, Gabriella, Klotz, Karl‐Norbert, Volpini, Rosaria, Popoli, Patrizia
Published in Journal of neurochemistry (01.04.2019)
Published in Journal of neurochemistry (01.04.2019)
Get full text
Journal Article
Pyrazolo-triazolo-pyrimidine Scaffold as a Molecular Passepartout for the Pan-Recognition of Human Adenosine Receptors
Salmaso, Veronica, Persico, Margherita, Da Ros, Tatiana, Spalluto, Giampiero, Kachler, Sonja, Klotz, Karl-Norbert, Moro, Stefano, Federico, Stephanie
Published in Biomolecules (Basel, Switzerland) (01.11.2023)
Published in Biomolecules (Basel, Switzerland) (01.11.2023)
Get full text
Journal Article
Chalcone-based derivatives as new scaffolds for hA3 adenosine receptor antagonists
Vazquez-Rodriguez, Saleta, Matos, Maria João, Santana, Lourdes, Uriarte, Eugenio, Borges, Fernanda, Kachler, Sonja, Klotz, Karl-Norbert
Published in Journal of pharmacy and pharmacology (01.05.2013)
Published in Journal of pharmacy and pharmacology (01.05.2013)
Get more information
Journal Article
Organoruthenium Antagonists of Human A3 Adenosine Receptors
Paira, Priyankar, Chow, Mun Juinn, Venkatesan, Gopalakrishnan, Kosaraju, Vamsi Krishna, Cheong, Siew Lee, Klotz, Karl-Norbert, Ang, Wee Han, Pastorin, Giorgia
Published in Chemistry : a European journal (17.06.2013)
Published in Chemistry : a European journal (17.06.2013)
Get full text
Journal Article
The Influence of the 1-(3-Trifluoromethyl-Benzyl)-1H-Pyrazole-4-yl Moiety on the Adenosine Receptors Affinity Profile of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidine Derivatives
Federico, Stephanie, Redenti, Sara, Sturlese, Mattia, Ciancetta, Antonella, Kachler, Sonja, Klotz, Karl-Norbert, Cacciari, Barbara, Moro, Stefano, Spalluto, Giampiero
Published in PloS one (01.12.2015)
Published in PloS one (01.12.2015)
Get full text
Journal Article
Synthesis and adenosine receptors binding affinities of a series of 3-arylcoumarins
Matos, Maria João, Hogger, Veronika, Gaspar, Alexandra, Kachler, Sonja, Borges, Fernanda, Uriarte, Eugenio, Santana, Lourdes, Klotz, Karl-Norbert
Published in Journal of pharmacy and pharmacology (01.11.2013)
Published in Journal of pharmacy and pharmacology (01.11.2013)
Get more information
Journal Article