Novel potent and selective inhibitors of inducible nitric oxide synthase
Nakane, M, Klinghofer, V, Kuk, J E, Donnelly, J L, Budzik, G P, Pollock, J S, Basha, F, Carter, G W
Published in Molecular pharmacology (01.04.1995)
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Published in Molecular pharmacology (01.04.1995)
Journal Article
Species Specificity of Amidine-Based Urokinase Inhibitors
Klinghofer, Vered, Stewart, Kent, McGonigal, Tom, Smith, Richard, Sarthy, Aparna, Nienaber, Vicki, Butler, Chris, Dorwin, Sarah, Richardson, Paul, Weitzberg, Moshe, Wendt, Mike, Rockway, Todd, Zhao, Xumiao, Hulkower, Keren I, Giranda, Vincent L
Published in Biochemistry (Easton) (07.08.2001)
Published in Biochemistry (Easton) (07.08.2001)
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Journal Article
Immunochemical detection of inducible NO synthase in human lung
Tracey, W R, Xue, C, Klinghofer, V, Barlow, J, Pollock, J S, Förstermann, U, Johns, R A
Published in The American journal of physiology (01.06.1994)
Published in The American journal of physiology (01.06.1994)
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Journal Article
Functional Expression of Three Isoforms of Human Nitric Oxide Synthase in Baculovirus-Infected Insect Cells
Nakane, M., Pollock, J.S., Klinghofer, V., Basha, F., Marsden, P.A., Hokari, A., Ogura, T., Esumi, H., Carter, G.W.
Published in Biochemical and biophysical research communications (17.01.1995)
Published in Biochemical and biophysical research communications (17.01.1995)
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Journal Article
The nitric oxide synthase inhibitor, L-NG-monomethylarginine, reduces carrageenan-induced pleurisy in the rat
Tracey, W R, Nakane, M, Kuk, J, Budzik, G, Klinghofer, V, Harris, R, Carter, G
Published in The Journal of pharmacology and experimental therapeutics (01.06.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1995)
Journal Article
Syntheses of Potent, Selective, and Orally Bioavailable Indazole-Pyridine Series of Protein Kinase B/Akt Inhibitors with Reduced Hypotension
Zhu, Gui-Dong, Gandhi, Viraj B, Gong, Jianchun, Thomas, Sheela, Woods, Keith W, Song, Xiaohong, Li, Tongmei, Diebold, R. Bruce, Luo, Yan, Liu, Xuesong, Guan, Ran, Klinghofer, Vered, Johnson, Eric F, Bouska, Jennifer, Olson, Amanda, Marsh, Kennan C, Stoll, Vincent S, Mamo, Mulugeta, Polakowski, James, Campbell, Thomas J, Martin, Ruth L, Gintant, Gary A, Penning, Thomas D, Li, Qun, Rosenberg, Saul H, Giranda, Vincent L
Published in Journal of medicinal chemistry (28.06.2007)
Published in Journal of medicinal chemistry (28.06.2007)
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Journal Article
Structure-directed discovery of potent non-peptidic inhibitors of human urokinase that access a novel binding subsite
Nienaber, Vicki L, Davidson, Donald, Edalji, Rohinton, Giranda, Vincent L, Klinghofer, Vered, Henkin, Jack, Magdalinos, Peter, Mantei, Robert, Merrick, Sean, Severin, Jean M, Smith, Richard A, Stewart, Kent, Walter, Karl, Wang, Jieyi, Wendt, Michael, Weitzberg, Moshe, Zhao, Xumiao, Rockway, Todd
Published in Structure (London) (15.05.2000)
Published in Structure (London) (15.05.2000)
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Journal Article
Endothelial nitric oxide synthase is myristylated
Pollock, Jennifer S., Klinghofer, Vered, Förstermann, Ulrich, Murad, Ferid
Published in FEBS letters (14.09.1992)
Published in FEBS letters (14.09.1992)
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Journal Article
Discovery of a Peptide-Based Renin Inhibitor with Oral Bioavailability and Efficacy
Kleinert, Hollis D., Rosenberg, Saul H., Baker, William R., Stein, Herman H., Klinghofer, Vered, Barlow, Jennifer, Spina, Kenneth, Polakowski, James, Kovar, Peter, Cohen, Jerome, Denissen, Jon
Published in Science (American Association for the Advancement of Science) (25.09.1992)
Published in Science (American Association for the Advancement of Science) (25.09.1992)
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Journal Article
Discovery of a new cyclooxygenase-2 lead compound through 3-D database searching and combinatorial chemistry
Stewart, Kent D., Loren, Stefan, Frey, Lisa, Otis, Ellen, Klinghofer, Vered, Hulkower, Keren I.
Published in Bioorganic & medicinal chemistry letters (03.03.1998)
Published in Bioorganic & medicinal chemistry letters (03.03.1998)
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Journal Article
Studies directed toward the design of orally active renin inhibitors. 2. Development of the efficacious, bioavailable renin inhibitor (2S)-2-benzyl-3-[[(1-methylpiperazin-4-yl)sulfonyl]propionyl]-3-thiazol-4-yl-L-alanine amide of (2S,3R,4S)-2-amino-1-cyclohexyl-3,4-dihydroxy-6-methylheptane (A-72517)
Rosenberg, Saul H, Spina, Kenneth P, Condon, Stephen L, Polakowski, Jim, Yao, Zhengli, Kovar, Peter, Stein, Herman H, Cohen, Jerome, Barlow, Jennifer L
Published in Journal of medicinal chemistry (19.02.1993)
Published in Journal of medicinal chemistry (19.02.1993)
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Journal Article
C-Terminal modifications of nonpeptide renin inhibitors: improved oral bioavailability via modification of physicochemical properties
Boyd, Steven A, Fung, Anthony K. L, Baker, William R, Mantei, Robert A, Armiger, Yoek Lin, Stein, Herman H, Cohen, Jerome, Egan, David A, Barlow, Jennifer L
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Journal Article
Discovery of a Well-Absorbed, Efficacious Renin Inhibitor, A-74273
Kleinert, Hollis D, Stein, Herman H, Boyd, Steven, Fung, Anthony K.L, Baker, William R, Verburg, Kenneth M, Polakowski, James S, Kovar, Peter, Barlow, Jennifer, Cohen, Jerome, Klinghofer, Vered, Mantei, Robert, Cepa, Steven, Rosenberg, Saul, Denissen, Jon F
Published in Hypertension (Dallas, Tex. 1979) (01.12.1992)
Published in Hypertension (Dallas, Tex. 1979) (01.12.1992)
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Journal Article
Studies directed toward the design of orally active renin inhibitors. II: Development of the efficacious, bioavailable renin inhibitor (2S)-2-benzyl-3-[[(1-methylpiperazin-4-yl)sulfonyl]propionyl]-3-thiazol-4-yl-L-alanine amide of (2S,3R,4S)-2-amino-1-cyclohexyl-3,4-dihydroxy-6-methylheptane (A-72517)
ROSENBERG, S. H, SPINA, K. P, EGAN, D. A, TRICARICO, K. A, PERUN, T. J, BAKER, W. R, KLEINERT, H. D, CONDON, S. L, POLAKOWSKI, J, ZHENGLI YAO, KOVAR, P, STEIN, H. H, COHEN, J, BARLOW, J. L, KLINGHOFER, V
Published in Journal of medicinal chemistry (1993)
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Published in Journal of medicinal chemistry (1993)
Journal Article
Cardiovascular effects and hemodynamic mechanism of action of the novel, nonpeptidic renin inhibitor A-74273 in dogs
Wessale, J L, Calzadilla, S V, Boyd, S A, Baker, W R, Stein, H H, Kovar, P J, Barlow, J, Klinghofer, V, Mantei, R, Kleinert, H D
Published in Journal of cardiovascular pharmacology (01.10.1993)
Published in Journal of cardiovascular pharmacology (01.10.1993)
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Journal Article
Effects of high doses of A-74273, a novel nonpeptidic and orally bioavailable renin inhibitor
Verburg, K M, Polakowski, J S, Kovar, P J, Klinghofer, V, Barlow, J L, Stein, H H, Mantei, R A, Fung, A K, Boyd, S A, Baker, W R
Published in Journal of cardiovascular pharmacology (01.01.1993)
Published in Journal of cardiovascular pharmacology (01.01.1993)
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