Correction to: Identification and characterization of deschloro-chlorothricin obtained from a large natural product library targeting aurora A kinase in multiple myeloma
Özenver, Nadire, Abdelfatah, Sara, Klinger, Anette, Fleischer, Edmond, Efferth, Thomas
Published in Investigational new drugs (01.04.2022)
Published in Investigational new drugs (01.04.2022)
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A novel ligand of the translationally controlled tumor protein (TCTP) identified by virtual drug screening for cancer differentiation therapy
Fischer, Nicolas, Seo, Ean-Jeong, Abdelfatah, Sara, Fleischer, Edmond, Klinger, Anette, Efferth, Thomas
Published in Investigational new drugs (01.08.2021)
Published in Investigational new drugs (01.08.2021)
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Journal Article
Identification and characterization of deschloro-chlorothricin obtained from a large natural product library targeting aurora A kinase in multiple myeloma
Özenver, Nadire, Abdelfatah, Sara, Klinger, Anette, Fleischer, Edmond, Efferth, Thomas
Published in Investigational new drugs (01.04.2021)
Published in Investigational new drugs (01.04.2021)
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Putative molecular determinants mediating sensitivity or resistance towards carnosic acid tumor cell responses
Mahmoud, Nuha, Saeed, Mohamed E.M., Sugimoto, Yoshikazu, Klinger, Anette, Fleischer, Edmond, Efferth, Thomas
Published in Phytomedicine (Stuttgart) (01.10.2020)
Published in Phytomedicine (Stuttgart) (01.10.2020)
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Vitamin K3 thio-derivative: a novel specific apoptotic inducer in the doxorubicin-sensitive and -resistant cancer cells
Hegazy, Mohamed-Elamir F., Fukaya, Masashi, Dawood, Mona, Yan, Ge, Klinger, Anette, Fleischer, Edmond, Zaglool, Asmaa W., Efferth, Thomas
Published in Investigational new drugs (01.06.2020)
Published in Investigational new drugs (01.06.2020)
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MCC1019, a selective inhibitor of the Polo-box domain of Polo-like kinase 1 as novel, potent anticancer candidate
Abdelfatah, Sara, Berg, Angela, Huang, Qi, Yang, Li Jun, Hamdoun, Sami, Klinger, Anette, Greten, Henry J., Fleischer, Edmond, Berg, Thorsten, Wong, Vincent K.W., Efferth, Thomas
Published in Acta pharmaceutica Sinica. B (01.09.2019)
Published in Acta pharmaceutica Sinica. B (01.09.2019)
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Novel 3,4-Dihydroisocoumarins Inhibit Human P-gp and BCRP in Multidrug Resistant Tumors and Demonstrate Substrate Inhibition of Yeast Pdr5
Sachs, Julia, Döhl, Katja, Weber, Anja, Bonus, Michele, Ehlers, Ferdinand, Fleischer, Edmond, Klinger, Anette, Gohlke, Holger, Pietruszka, Jörg, Schmitt, Lutz, Teusch, Nicole
Published in Frontiers in pharmacology (16.04.2019)
Published in Frontiers in pharmacology (16.04.2019)
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Isopetasin and S-isopetasin as novel P-glycoprotein inhibitors against multidrug-resistant cancer cells
Abdelfatah, Sara, Böckers, Madeleine, Asensio, Maitane, Kadioglu, Onat, Klinger, Anette, Fleischer, Edmond, Efferth, Thomas
Published in Phytomedicine (Stuttgart) (01.06.2021)
Published in Phytomedicine (Stuttgart) (01.06.2021)
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AMG900 as novel inhibitor of the translationally controlled tumor protein
Fischer, Nicolas, Seo, Ean-Jeong, Klinger, Anette, Fleischer, Edmond, Efferth, Thomas
Published in Chemico-biological interactions (25.01.2021)
Published in Chemico-biological interactions (25.01.2021)
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Cytotoxicity of 4-hydroxy-N-(naphthalen-1-yl)-2-oxo-2H-chromene-3-carboxamide in multidrug-resistant cancer cells through activation of PERK/eIF2α/ATF4 pathway
Lu, Xiaohua, Yan, Ge, Klauck, Sabine M., Fleischer, Edmond, Klinger, Anette, Sugimoto, Yoshikazu, Shan, Letian, Efferth, Thomas
Published in Biochemical pharmacology (01.11.2021)
Published in Biochemical pharmacology (01.11.2021)
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A novel moniliformin derivative as pan-inhibitor of histone deacetylases triggering apoptosis of leukemia cells
Lu, Xiaohua, Yan, Ge, Dawood, Mona, Klauck, Sabine M., Sugimoto, Yoshikazu, Klinger, Anette, Fleischer, Edmond, Shan, Letian, Efferth, Thomas
Published in Biochemical pharmacology (01.12.2021)
Published in Biochemical pharmacology (01.12.2021)
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Vitamin K 3 chloro derivative (VKT-2) inhibits HDAC6, activates autophagy and apoptosis, and inhibits aggresome formation in hepatocellular carcinoma cells
Dawood, Mona, Hegazy, Mohamed-Elamir F, Elbadawi, Mohamed, Fleischer, Edmond, Klinger, Anette, Bringmann, Gerhard, Kuntner, Claudia, Shan, Letian, Efferth, Thomas
Published in Biochemical pharmacology (01.10.2020)
Published in Biochemical pharmacology (01.10.2020)
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Naphthoquinone derivatives as P-glycoprotein inducers in inflammatory bowel disease: 2D monolayers, 3D spheroids, and in vivo models
Mahmoud, Nuha, Hegazy, Mohamed-Elamir F., Wadie, Walaa, Elbadawi, Mohamed, Fleischer, Edmond, Klinger, Anette, Bringmann, Gerhard, Khayyal, Mohamed T., Efferth, Thomas
Published in Pharmacological research (01.05.2022)
Published in Pharmacological research (01.05.2022)
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Journal Article
Vitamin K3 chloro derivative (VKT-2) inhibits HDAC6, activates autophagy and apoptosis, and inhibits aggresome formation in hepatocellular carcinoma cells
Dawood, Mona, Hegazy, Mohamed-Elamir F., Elbadawi, Mohamed, Fleischer, Edmond, Klinger, Anette, Bringmann, Gerhard, Kuntner, Claudia, Shan, Letian, Efferth, Thomas
Published in Biochemical pharmacology (01.10.2020)
Published in Biochemical pharmacology (01.10.2020)
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