Active-state model of a dopamine D2 receptor-Gαi complex stabilized by aripiprazole-type partial agonists
Kling, Ralf C, Tschammer, Nuska, Lanig, Harald, Clark, Timothy, Gmeiner, Peter
Published in PloS one (16.06.2014)
Published in PloS one (16.06.2014)
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Journal Article
Development of Covalent Ligand–Receptor Pairs to Study the Binding Properties of Nonpeptidic Neurotensin Receptor 1 Antagonists
Kling, Ralf C, Plomer, Manuel, Lang, Christopher, Banerjee, Ashutosh, Hübner, Harald, Gmeiner, Peter
Published in ACS chemical biology (15.04.2016)
Published in ACS chemical biology (15.04.2016)
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Journal Article
GPCR crystal structures: Medicinal chemistry in the pocket
Shonberg, Jeremy, Kling, Ralf C., Gmeiner, Peter, Löber, Stefan
Published in Bioorganic & medicinal chemistry (15.07.2015)
Published in Bioorganic & medicinal chemistry (15.07.2015)
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Journal Article
Structural insights into µ-opioid receptor activation
Huang, Weijiao, Manglik, Aashish, Venkatakrishnan, A J, Laeremans, Toon, Feinberg, Evan N, Sanborn, Adrian L, Kato, Hideaki E, Livingston, Kathryn E, Thorsen, Thor S, Kling, Ralf C, Granier, Sébastien, Gmeiner, Peter, Husbands, Stephen M, Traynor, John R, Weis, William I, Steyaert, Jan, Dror, Ron O, Kobilka, Brian K
Published in Nature (London) (20.08.2015)
Published in Nature (London) (20.08.2015)
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Journal Article
Structure-based discovery of opioid analgesics with reduced side effects
Manglik, Aashish, Lin, Henry, Aryal, Dipendra K, McCorvy, John D, Dengler, Daniela, Corder, Gregory, Levit, Anat, Kling, Ralf C, Bernat, Viachaslau, Hübner, Harald, Huang, Xi-Ping, Sassano, Maria F, Giguère, Patrick M, Löber, Stefan, Da Duan, Scherrer, Grégory, Kobilka, Brian K, Gmeiner, Peter, Roth, Bryan L, Shoichet, Brian K
Published in Nature (London) (08.09.2016)
Published in Nature (London) (08.09.2016)
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Journal Article
Identification of Two Distinct Sites for Antagonist and Biased Agonist Binding to the Human Chemokine Receptor CXCR3
Milanos, Lampros, Saleh, Noureldin, Kling, Ralf C., Kaindl, Jonas, Tschammer, Nuska, Clark, Timothy
Published in Angewandte Chemie (International ed.) (05.12.2016)
Published in Angewandte Chemie (International ed.) (05.12.2016)
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Journal Article
Functionally Selective Dopamine D2, D3 Receptor Partial Agonists
Möller, Dorothee, Kling, Ralf C, Skultety, Marika, Leuner, Kristina, Hübner, Harald, Gmeiner, Peter
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
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Journal Article
Basal Histamine H4 Receptor Activation: Agonist Mimicry by the Diphenylalanine Motif
Wifling, David, Pfleger, Christopher, Kaindl, Jonas, Ibrahim, Passainte, Kling, Ralf C., Buschauer, Armin, Gohlke, Holger, Clark, Timothy
Published in Chemistry : a European journal (18.11.2019)
Published in Chemistry : a European journal (18.11.2019)
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Journal Article
Molecular Determinants of Biased Agonism at the Dopamine D2 Receptor
Weichert, Dietmar, Banerjee, Ashutosh, Hiller, Christine, Kling, Ralf C, Hübner, Harald, Gmeiner, Peter
Published in Journal of medicinal chemistry (26.03.2015)
Published in Journal of medicinal chemistry (26.03.2015)
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Journal Article
Basal Histamine H 4 Receptor Activation: Agonist Mimicry by the Diphenylalanine Motif
Wifling, David, Pfleger, Christopher, Kaindl, Jonas, Ibrahim, Passainte, Kling, Ralf C, Buschauer, Armin, Gohlke, Holger, Clark, Timothy
Published in Chemistry : a European journal (18.11.2019)
Published in Chemistry : a European journal (18.11.2019)
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Journal Article
1,4-Disubstituted aromatic piperazines with high 5-HT2A/D2 selectivity: Quantitative structure-selectivity investigations, docking, synthesis and biological evaluation
Möller, Dorothee, Salama, Ismail, Kling, Ralf C., Hübner, Harald, Gmeiner, Peter
Published in Bioorganic & medicinal chemistry (15.09.2015)
Published in Bioorganic & medicinal chemistry (15.09.2015)
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Journal Article
Functionally Selective Dopamine D2/D3 Receptor Agonists Comprising an Enyne Moiety
Hiller, Christine, Kling, Ralf C, Heinemann, Frank W, Meyer, Karsten, Hübner, Harald, Gmeiner, Peter
Published in Journal of medicinal chemistry (27.06.2013)
Published in Journal of medicinal chemistry (27.06.2013)
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Journal Article
Author Correction: Structural insights into μ-opioid receptor activation
Huang, Weijiao, Manglik, Aashish, Venkatakrishnan, A J, Laeremans, Toon, Feinberg, Evan N, Sanborn, Adrian L, Kato, Hideaki E, Livingston, Kathryn E, Thorsen, Thor S, Kling, Ralf C, Granier, Sébastien, Gmeiner, Peter, Husbands, Stephen M, Traynor, John R, Weis, William I, Steyaert, Jan, Dror, Ron O, Kobilka, Brian K
Published in Nature (London) (13.08.2020)
Published in Nature (London) (13.08.2020)
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Journal Article
NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids
Simeth, Nadja A., Bause, Manuel, Dobmeier, Michael, Kling, Ralf C., Lachmann, Daniel, Hübner, Harald, Einsiedel, Jürgen, Gmeiner, Peter, König, Burkhard
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Structural insights into [micro]-opioid receptor activation
Huang, Weijiao, Manglik, Aashish, Venkatakrishnan, A. J, Laeremans, Toon, Feinberg, Evan N, Sanborn, Adrian L, Kato, Hideaki E
Published in Nature (London) (20.08.2015)
Published in Nature (London) (20.08.2015)
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Journal Article
1,4-Disubstituted aromatic piperazines with high 5-HT2A/D-2 selectivity: Quantitative structure-selectivity investigations, docking, synthesis and biological evaluation
Moeller, Dorothee, Salama, Ismail, Kling, Ralf C., Huebner, Harald, Gmeiner, Peter
Published in Bioorganic & medicinal chemistry (15.09.2015)
Published in Bioorganic & medicinal chemistry (15.09.2015)
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Journal Article