Pharmacokinetics of Lorlatinib After Single and Multiple Dosing in Patients with Anaplastic Lymphoma Kinase (ALK)-Positive Non-Small Cell Lung Cancer: Results from a Global Phase I/II Study
Chen, Joseph, O’Gorman, Melissa T., James, Lee P., Klamerus, Karen J., Mugundu, Ganesh, Pithavala, Yazdi K.
Published in Clinical pharmacokinetics (01.10.2021)
Published in Clinical pharmacokinetics (01.10.2021)
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Journal Article
Clinical Pharmacology of Axitinib
Chen, Ying, Tortorici, Michael A., Garrett, May, Hee, Brian, Klamerus, Karen J., Pithavala, Yazdi K.
Published in Clinical pharmacokinetics (01.09.2013)
Published in Clinical pharmacokinetics (01.09.2013)
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Journal Article
Dose-ranging evaluation of intravitreal siRNA PF-04523655 for diabetic macular edema (the DEGAS study)
Nguyen, Quan Dong, Schachar, Ronald A, Nduaka, Chudy I, Sperling, Marvin, Basile, Anthony S, Klamerus, Karen J, Chi-Burris, Katherine, Yan, Eric, Paggiarino, Dario A, Rosenblatt, Irit, Aitchison, Roger, Erlich, Shai S
Published in Investigative ophthalmology & visual science (15.11.2012)
Published in Investigative ophthalmology & visual science (15.11.2012)
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Journal Article
Evaluation of the siRNA PF-04523655 versus Ranibizumab for the Treatment of Neovascular Age-related Macular Degeneration (MONET Study)
Nguyen, Quan Dong, MD, MSc, Schachar, Ronald A., MD, PhD, Nduaka, Chudy I., DVM, PhD, Sperling, Marvin, MD, Klamerus, Karen J., PharmD, Chi-Burris, Katherine, MPH, Yan, Eric, PhD, Paggiarino, Dario A., MD, Rosenblatt, Irit, MD, Aitchison, Roger, MS, Erlich, Shai S., PhD
Published in Ophthalmology (Rochester, Minn.) (01.09.2012)
Published in Ophthalmology (Rochester, Minn.) (01.09.2012)
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Journal Article
The effect of tafamidis on the QTc interval in healthy subjects
Klamerus, Karen J., Watsky, Eric, Moller, Robert, Wang, Ronnie, Riley, Steve
Published in British journal of clinical pharmacology (01.06.2015)
Published in British journal of clinical pharmacology (01.06.2015)
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Journal Article
Impact of Acid‐Reducing Agents on the Pharmacokinetics of Palbociclib, a Weak Base With pH‐Dependent Solubility, With Different Food Intake Conditions
Sun, Wan, Klamerus, Karen J., Yuhas, Lisa M., Pawlak, Sylvester, Plotka, Anna, O'Gorman, Melissa, Kirkovsky, Leonid, Kosa, Maha, Wang, Diane
Published in Clinical pharmacology in drug development (01.11.2017)
Published in Clinical pharmacology in drug development (01.11.2017)
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Journal Article
Axitinib inhibits retinal and choroidal neovascularization in in vitro and in vivo models
Giddabasappa, Anand, Lalwani, Kush, Norberg, Rand, Gukasyan, Hovhannes J., Paterson, David, Schachar, Ronald A., Rittenhouse, Kay, Klamerus, Karen, Mosyak, Lydia, Eswaraka, Jeetendra
Published in Experimental eye research (01.04.2016)
Published in Experimental eye research (01.04.2016)
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Journal Article
Pharmacokinetics, metabolism, and excretion of [14C]axitinib, a vascular endothelial growth factor receptor tyrosine kinase inhibitor, in humans
Smith, Bill J, Pithavala, Yazdi, Bu, Hai-Zhi, Kang, Ping, Hee, Brian, Deese, Alan J, Pool, William F, Klamerus, Karen J, Wu, Ellen Y, Dalvie, Deepak K
Published in Drug metabolism and disposition (01.05.2014)
Published in Drug metabolism and disposition (01.05.2014)
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Journal Article
Tofacitinib (CP-690,550), a Janus Kinase Inhibitor for Dry Eye Disease
Liew, Shiao Hui (Melissa), MBBS, MRCOphth, Nichols, Kelly K., OD, PhD, Klamerus, Karen J., PharmD, Li, Jim Z., PhD, Zhang, Min, MS, Foulks, Gary N., MD, FACS
Published in Ophthalmology (Rochester, Minn.) (01.07.2012)
Published in Ophthalmology (Rochester, Minn.) (01.07.2012)
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Journal Article
Effect of food on the pharmacokinetics of sunitinib malate (SU11248), a multi-targeted receptor tyrosine kinase inhibitor: results from a phase I study in healthy subjects
Bello, Carlo L, Sherman, Laurie, Zhou, Jihao, Verkh, Lev, Smeraglia, John, Mount, Janessa, Klamerus, Karen J
Published in Anti-cancer drugs (01.03.2006)
Published in Anti-cancer drugs (01.03.2006)
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Journal Article
Effect of ketoconazole on the pharmacokinetics of axitinib in healthy volunteers
Pithavala, Yazdi K., Tong, Warren, Mount, Janessa, Rahavendran, Sadayappan V., Garrett, May, Hee, Brian, Selaru, Paulina, Sarapa, Nenad, Klamerus, Karen J.
Published in Investigational new drugs (01.02.2012)
Published in Investigational new drugs (01.02.2012)
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Journal Article
Evaluation of the effect of food on the pharmacokinetics of axitinib in healthy volunteers
Pithavala, Yazdi K., Chen, Ying, Toh, Melvin, Selaru, Paulina, LaBadie, Robert R., Garrett, May, Hee, Brian, Mount, Janessa, Ni, Grace, Klamerus, Karen J., Tortorici, Michael A.
Published in Cancer chemotherapy and pharmacology (01.07.2012)
Published in Cancer chemotherapy and pharmacology (01.07.2012)
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Journal Article
Integrating disease progression models, non-clinical pharmacokinetic data and treatment response endpoints to optimize intravitreal dosing regimens
Basile, Anthony S, Johnson, Theodore R, Klamerus, Karen J, Zhou, Duo, Sultan, Marla B, Amantea, Mike, Nickens, Dana J
Published in International journal of clinical pharmacology and therapeutics (01.07.2014)
Published in International journal of clinical pharmacology and therapeutics (01.07.2014)
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Journal Article
Evaluation of the potential interaction between tofacitinib and drugs that undergo renal tubular secretion using metformin, an in vivo marker of renal organic cation transporter 2
Klamerus, Karen J., Alvey, Christine, Li, Lei, Feng, Bo, Wang, Rong, Kaplan, Irina, Shi, Haihong, Dowty, Martin E., Krishnaswami, Sriram
Published in Clinical pharmacology in drug development (01.11.2014)
Published in Clinical pharmacology in drug development (01.11.2014)
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Journal Article
The effect of tafamidis on the QT c interval in healthy subjects
Klamerus, Karen J., Watsky, Eric, Moller, Robert, Wang, Ronnie, Riley, Steve
Published in British journal of clinical pharmacology (01.06.2015)
Published in British journal of clinical pharmacology (01.06.2015)
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Journal Article
Safety and efficacy of lorlatinib (PF-06463922) from the dose-escalation component of a study in patients with advanced ALK+ or ROS1+ non-small cell lung cancer (NSCLC)
Solomon, Benjamin J., Bauer, Todd Michael, Felip, Enriqueta, Besse, Benjamin, James, Leonard Philip, Clancy, Jill S., Klamerus, Karen J., Martini, Jean-Francois, Abbattista, Antonello, Shaw, Alice Tsang
Published in Journal of clinical oncology (20.05.2016)
Published in Journal of clinical oncology (20.05.2016)
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Journal Article
A pharmacokinetic and pharmacodynamic study of the potential drug interaction between tasosartan and atenolol in patients with stage 1 and 2 essential hypertension
Andrawis, N S, Battle, M M, Klamerus, K J, Burghart, P H, Neefe, L, Weinryb, I, Mayer, P, Abernethy, D R
Published in Journal of clinical pharmacology (01.03.2000)
Published in Journal of clinical pharmacology (01.03.2000)
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Journal Article
The use of mycophenolate mofetil suspension in pediatric renal allograft recipients
BUNCHMAN, Timothy, NAVARRO, Mercedes, WALKER, Rowan, ZIMMERHACKL, Lothar B, BLOWEY, Douglas, CLARK, Godfrey, ETTENGER, Robert, ARTERBURN, Sarah, KLAMERUS, Karen, FONG, Alice, TANG, Helen, THOMAS, Susan, BROYER, Michel, RAMOS, Eleanor, SHERBOTIE, Joseph, CHAVERS, Blanche, TÖNSHOFF, Burkhard, BIRK, Patricia, LERNER, Gary, LIRENMAN, David, GREENBAUM, Laurence
Published in Pediatric nephrology (Berlin, West) (01.12.2001)
Published in Pediatric nephrology (Berlin, West) (01.12.2001)
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