Identification of 2-[2-(4-tert-butylphenyl)ethyl]-N-(4-fluorophenyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide (29) as an orally available MGAT2 inhibitor
Busujima, Tsuyoshi, Tanaka, Hiroaki, Shirasaki, Yoshihisa, Munetomo, Eiji, Saito, Masako, Kitano, Kiyokazu, Minagawa, Toshiya, Yoshida, Koji, Osaki, Naoto, Sato, Nagaaki
Published in Bioorganic & medicinal chemistry (01.09.2015)
Published in Bioorganic & medicinal chemistry (01.09.2015)
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Identification of 2-[2-(4-tert-Butylphenyl)ethyl]-N-[4-(3-cyclopentylpropyl)-2-fluorophenyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide as an Orally Active MGAT2 Inhibitor
Busujima, Tsuyoshi, Tanaka, Hiroaki, Iwakiri, Kanako, Shirasaki, Yoshihisa, Munetomo, Eiji, Saito, Masako, Masuko, Aiko, Kitano, Kiyokazu, Io, Fusayo, Kato, Koji, Kamigaso, Shunsuke, Nozoe, Akiko, Sato, Nagaaki
Published in Chemical & pharmaceutical bulletin (01.03.2016)
Published in Chemical & pharmaceutical bulletin (01.03.2016)
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Synthesis and structure–activity relationships of potent 3- or 4-substituted-2-cyanopyrrolidine dipeptidyl peptidase IV inhibitors
Fukushima, Hiroshi, Hiratate, Akira, Takahashi, Masato, Saito, Masako, Munetomo, Eiji, Kitano, Kiyokazu, Saito, Hidetaka, Takaoka, Yuji, Yamamoto, Koji
Published in Bioorganic & medicinal chemistry (01.12.2004)
Published in Bioorganic & medicinal chemistry (01.12.2004)
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Synthesis and Structure–Activity Relationships of Potent 1-(2-Substituted-aminoacetyl)-4-fluoro-2-cyanopyrrolidine Dipeptidyl Peptidase IV Inhibitors
Fukushima, Hiroshi, Hiratate, Akira, Takahashi, Masato, Saito-Hori, Masako, Munetomo, Eiji, Kitano, Kiyokazu, Saito, Hidetaka, Takaoka, Yuji, Yamamoto, Koji
Published in Chemical & Pharmaceutical Bulletin (01.08.2008)
Published in Chemical & Pharmaceutical Bulletin (01.08.2008)
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(2 S,4 S)-4-Fluoro-1-{[(2-hydroxy-1,1-dimethylethyl)amino]acetyl}-pyrrolidine-2-carbonitrile monobenzenesulfonate (TS-021) is a selective and reversible dipeptidyl peptidase IV inhibitor
Tajima, Atsushi, Yamamoto, Koji, Kozakai, Akinori, Okumura-Kitajima, Lisa, Mita, Yasuo, Kitano, Kiyokazu, Jingu, Shigeji, Nakaike, Shiro
Published in European journal of pharmacology (25.03.2011)
Published in European journal of pharmacology (25.03.2011)
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Purification of a novel muscle cell growth factor S-myotrophin from porcine skeletal muscle
Hayashi, Toshiya, Takeshita, Keisuke, Tsuchida, Nobuyuki, Kitano, Kiyokazu, Kawabata, Shun-Ichiro, Iwanaga, Sadaaki, Ito, Tatsumi
Published in The international journal of biochemistry & cell biology (01.08.1998)
Published in The international journal of biochemistry & cell biology (01.08.1998)
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ChemInform Abstract: Synthesis and Structure-Activity Relationships of Potent 1-(2-Substituted-aminoacetyl)-4-fluoro-2-cyanopyrrolidine Dipeptidyl Peptidase IV Inhibitors
Fukushima, Hiroshi, Hiratate, Akira, Takahashi, Masato, Saito-Hori, Masako, Munetomo, Eiji, Kitano, Kiyokazu, Saito, Hidetaka, Takaoka, Yuji, Yamamoto, Koji
Published in ChemInform (20.01.2009)
Published in ChemInform (20.01.2009)
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Involvement of 5-HT4 receptors in regulation of defecation
Ito, Chika, Kawamura, Reiko, Kitano, Kiyokazu, Isobe, Yoshihiko, Fukushima, Kiyomi
Published in Japanese journal of pharmacology (1999)
Published in Japanese journal of pharmacology (1999)
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