Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U‑Shaped Binding Mode
Lu, Jun, Patel, Sangita, Sharma, Nandini, Soisson, Stephen M, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Lumb, Kevin J, Singh, Sheo B
Published in ACS chemical biology (19.09.2014)
Published in ACS chemical biology (19.09.2014)
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Journal Article
Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent
Singh, Sheo B, Dayananth, Priya, Balibar, Carl J, Garlisi, Charles G, Lu, Jun, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Ha, Sookhee, Young, Katherine
Published in Antimicrobial agents and chemotherapy (01.06.2015)
Published in Antimicrobial agents and chemotherapy (01.06.2015)
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Journal Article
Structural and Functional Studies of the HAMP Domain of EnvZ, an Osmosensing Transmembrane Histidine Kinase in Escherichia coli
Kishii, Ryuta, Falzon, Liliana, Yoshida, Takeshi, Kobayashi, Hiroshi, Inouye, Masayori
Published in The Journal of biological chemistry (07.09.2007)
Published in The Journal of biological chemistry (07.09.2007)
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Journal Article
Contributions of the 8-Methoxy Group of Gatifloxacin to Resistance Selectivity, Target Preference, and Antibacterial Activity against Streptococcus pneumoniae
FUKUDA, Hideyuki, KISHII, Ryuta, TAKEI, Masaya, HOSAKA, Masaki
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
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Journal Article
In Vitro Activities and Spectrum of the Novel Fluoroquinolone Lascufloxacin (KRP-AM1977)
Kishii, Ryuta, Yamaguchi, Yuko, Takei, Masaya
Published in Antimicrobial agents and chemotherapy (01.06.2017)
Published in Antimicrobial agents and chemotherapy (01.06.2017)
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Journal Article
Contribution of the 8-Methoxy Group to the Activity of Gatifloxacin against Type II Topoisomerases of Streptococcus pneumoniae
KISHII, Ryuta, TAKEI, Masaya, FUKUDA, Hideyuki, HAYASHI, Katsuhiko, HOSAKA, Masaki
Published in Antimicrobial Agents and Chemotherapy (01.01.2003)
Published in Antimicrobial Agents and Chemotherapy (01.01.2003)
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Journal Article
The effect of pharmacokinetic/pharmacodynamic (PK/PD) parameters of gatifloxacin on its bactericidal activity and resistance selectivity against clinical isolates of Streptococcus pneumoniae
Ebisu, Hiroyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Hideyuki
Published in Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy (01.09.2003)
Published in Journal of infection and chemotherapy : official journal of the Japan Society of Chemotherapy (01.09.2003)
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Journal Article
Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-9)
Singh, Sheo B., Tan, Christopher M., Kaelin, David, Meinke, Peter T., Miesel, Lynn, Olsen, David B., Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Ohata, Kohei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Journal Article
LpxC Inhibitors: Design, Synthesis, and Biological Evaluation of Oxazolidinones as Gram-negative Antibacterial Agents
Kurasaki, Haruaki, Tsuda, Kosuke, Shinoyama, Mariko, Takaya, Noriko, Yamaguchi, Yuko, Kishii, Ryuta, Iwase, Kazuhiko, Ando, Naoki, Nomura, Masahiro, Kohno, Yasushi
Published in ACS medicinal chemistry letters (09.06.2016)
Published in ACS medicinal chemistry letters (09.06.2016)
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Journal Article
In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase
Tan, Christopher M, Gill, Charles J, Wu, Jin, Toussaint, Nathalie, Yin, Jingjun, Tsuchiya, Takayuki, Garlisi, Charles G, Kaelin, David, Meinke, Peter T, Miesel, Lynn, Olsen, David B, Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Oohata, Kouhei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi, Singh, Sheo B
Published in Antimicrobial agents and chemotherapy (01.08.2016)
Published in Antimicrobial agents and chemotherapy (01.08.2016)
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Journal Article
Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents
Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Meinke, Peter T, Olsen, David, Lagrutta, Armando, Bradley, Prudence, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Wei, Changqing, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi
Published in ACS medicinal chemistry letters (08.05.2014)
Published in ACS medicinal chemistry letters (08.05.2014)
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Journal Article
Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Lu, Jun, Patel, Sangita, Rickert, Keith W., Smith, Robert F., Soisson, Stephen, Sherer, Edward, Joyce, Leo A., Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takano, Hisashi, Shibasaki, Mitsuhito, Yajima, Masanobu, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
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Journal Article
Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Gill, Charles, Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Shibue, Taku, Ohata, Kohei, Takano, Hisashi, Ban, Shizuka, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
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Journal Article
Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5)
Singh, Sheo B., Kaelin, David E., Meinke, Peter T., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Olsen, David B., Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Takano, Hisashi, Ohata, Kohei, Kurasaki, Haruaki, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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Journal Article
Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Yajima, Masanobu, Shibue, Taku, Shibata, Takeshi, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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