Discovery, synthesis and SAR of 2-acyl-1-biarylmethyl pyrazolidines, dual orexin receptor antagonists designed as fast and short-acting sleeping drugs
Surivet, Jean-Philippe, Kessler, Melanie, Vaillant, Catherine, Aissaoui, Hamed, Bezençon, Olivier, Busch, Louise, Kiry, Manon, Lüthi, Urs, Marck, Nicolas, Masse, Florence, Peters, Jens-Uwe, Sweatman, Catherine, Weigel, Aude, Kohl, Christopher
Published in Bioorganic & medicinal chemistry (01.10.2024)
Published in Bioorganic & medicinal chemistry (01.10.2024)
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