Chemical genetics and proteome-wide site mapping reveal cysteine MARylation by PARP-7 on immune-relevant protein targets
Rodriguez, Kelsie M, Buch-Larsen, Sara C, Kirby, Ilsa T, Siordia, Ivan Rodriguez, Hutin, David, Rasmussen, Marit, Grant, Denis M, David, Larry L, Matthews, Jason, Nielsen, Michael L, Cohen, Michael S
Published in eLife (21.01.2021)
Published in eLife (21.01.2021)
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A Novel Agonist of the TRIF Pathway Induces a Cellular State Refractory to Replication of Zika, Chikungunya, and Dengue Viruses
Pryke, Kara M, Abraham, Jinu, Sali, Tina M, Gall, Bryan J, Archer, Iris, Liu, Andrew, Bambina, Shelly, Baird, Jason, Gough, Michael, Chakhtoura, Marita, Haddad, Elias K, Kirby, Ilsa T, Nilsen, Aaron, Streblow, Daniel N, Hirsch, Alec J, Smith, Jessica L, DeFilippis, Victor R
Published in mBio (02.05.2017)
Published in mBio (02.05.2017)
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Journal Article
Reversible ADP-ribosylation of RNA
Munnur, Deeksha, Bartlett, Edward, Mikolčević, Petra, Kirby, Ilsa T, Rack, Johannes Gregor Matthias, Mikoč, Andreja, Cohen, Michael S, Ahel, Ivan
Published in Nucleic Acids Research (20.06.2019)
Published in Nucleic Acids Research (20.06.2019)
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ADP-ribosyl–binding and hydrolase activities of the alphavirus nsP3 macrodomain are critical for initiation of virus replication
Abraham, Rachy, Hauer, Debra, McPherson, Robert Lyle, Utt, Age, Kirby, Ilsa T., Cohen, Michael S., Merits, Andres, Leung, Anthony K. L., Griffin, Diane E.
Published in Proceedings of the National Academy of Sciences - PNAS (30.10.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (30.10.2018)
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Journal Article
A Potent and Selective PARP11 Inhibitor Suggests Coupling between Cellular Localization and Catalytic Activity
Kirby, Ilsa T., Kojic, Ana, Arnold, Moriah R., Thorsell, Ann-Gerd, Karlberg, Tobias, Vermehren-Schmaedick, Anke, Sreenivasan, Raashi, Schultz, Carsten, Schüler, Herwig, Cohen, Michael S.
Published in Cell chemical biology (20.12.2018)
Published in Cell chemical biology (20.12.2018)
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Journal Article
Structure-guided design and characterization of a clickable, covalent PARP16 inhibitor
Bejan, Daniel S, Sundalam, Sunil, Jin, Haihong, Morgan, Rory K, Kirby, Ilsa T, Siordia, Ivan R, Tivon, Barr, London, Nir, Cohen, Michael S
Published in Chemical science (Cambridge) (30.11.2022)
Published in Chemical science (Cambridge) (30.11.2022)
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Allosteric regulation of DNA binding and target residence time drive the cytotoxicity of phthalazinone-based PARP-1 inhibitors
Arnold, Moriah R., Langelier, Marie-France, Gartrell, Jessica, Kirby, Ilsa T., Sanderson, Daniel J., Bejan, Daniel S., Šileikytė, Justina, Sundalam, Sunil K., Nagarajan, Shanthi, Marimuthu, Parthiban, Duell, Anna K., Shelat, Anang A., Pascal, John M., Cohen, Michael S.
Published in Cell chemical biology (15.12.2022)
Published in Cell chemical biology (15.12.2022)
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Journal Article
Rational Design of Cell-Active Inhibitors of PARP10
Morgan, Rory K, Kirby, Ilsa T, Vermehren-Schmaedick, Anke, Rodriguez, Kelsie, Cohen, Michael S
Published in ACS medicinal chemistry letters (10.01.2019)
Published in ACS medicinal chemistry letters (10.01.2019)
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A SARS-CoV-2 protein interaction map reveals targets for drug repurposing
Gordon, David E, Jang, Gwendolyn M, Bouhaddou, Mehdi, Obernier, Kirsten, White, Kris M, O'Meara, Matthew J, Rezelj, Veronica V, Swaney, Danielle L, Tummino, Tia A, Hüttenhain, Ruth, Richards, Alicia L, Tutuncuoglu, Beril, Foussard, Helene, Batra, Jyoti, Haas, Kelsey, Modak, Maya, Kim, Minkyu, Haas, Paige, Polacco, Benjamin J, Braberg, Hannes, Fabius, Jacqueline M, Eckhardt, Manon, Soucheray, Margaret, Bennett, Melanie J, Cakir, Merve, Li, Qiongyu, Meyer, Bjoern, Roesch, Ferdinand, Vallet, Thomas, Mac Kain, Alice, Naing, Zun Zar Chi, Zhou, Yuan, Shi, Ying, Zhang, Ziyang, Shen, Wenqi, Kirby, Ilsa T, Melnyk, James E, Chorba, John S, Lou, Kevin, Barrio-Hernandez, Inigo, Hernandez-Armenta, Claudia, Lyu, Jiankun, Mathy, Christopher J P, Perica, Tina, Pilla, Kala Bharath, Ganesan, Sai J, Saltzberg, Daniel J, Rakesh, Ramachandran, Rosenthal, Sara B, Calviello, Lorenzo, Venkataramanan, Srivats, Lin, Yizhu, Huang, Xi-Ping, Wankowicz, Stephanie A, Bohn, Markus, Safari, Maliheh, Ugur, Fatima S, Koh, Cassandra, Savar, Nastaran Sadat, Tran, Quang Dinh, Shengjuler, Djoshkun, O'Neal, Michael C, Chang, Jason C J, Klippsten, Saker, Sharp, Phillip P, Kuzuoglu-Ozturk, Duygu, Wang, Hao-Yuan, Cavero, Devin A, Rathore, Ujjwal, Subramanian, Advait, Noack, Julia, Stroud, Robert M, Frankel, Alan D, Rosenberg, Oren S, Verba, Kliment A, Agard, David A, Ott, Melanie, Emerman, Michael, Jura, Natalia, von Zastrow, Mark, Verdin, Eric, Ashworth, Alan, Schwartz, Olivier, d'Enfert, Christophe, Jacobson, Matt, Malik, Harmit S, Fujimori, Danica G, Craik, Charles S, Fraser, James S, Gross, John D, Sali, Andrej, Roth, Bryan L, Ruggero, Davide, Taunton, Jack, Kortemme, Tanja, Beltrao, Pedro, García-Sastre, Adolfo, Shokat, Kevan M, Shoichet, Brian K, Krogan, Nevan J
Published in Nature (London) (16.07.2020)
Published in Nature (London) (16.07.2020)
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Host-directed therapies against early-lineage SARS-CoV-2 retain efficacy against B.1.1.7 variant
Reuschl, Ann-Kathrin, Thorne, Lucy G, Zuliani-Alvarez, Lorena, Bouhaddou, Mehdi, Obernier, Kirsten, Hiatt, Joseph, Soucheray, Margaret, Turner, Jane, Fabius, Jacqueline M, Nguyen, Gina T, Swaney, Danielle L, Rosales, Romel, White, Kris M, Avilés, Pablo, Kirby, Ilsa T, Melnyk, James E, Shi, Ying, Zhang, Ziyang, Shokat, Kevan M, García-Sastre, Adolfo, Jolly, Clare, Towers, Gregory J, Krogan, Nevan J
Published in bioRxiv (04.02.2021)
Published in bioRxiv (04.02.2021)
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A SARS-CoV-2-Human Protein-Protein Interaction Map Reveals Drug Targets and Potential Drug-Repurposing
Gordon, David E, Jang, Gwendolyn M, Bouhaddou, Mehdi, Xu, Jiewei, Obernier, Kirsten, O'Meara, Matthew J, Guo, Jeffrey Z, Swaney, Danielle L, Tummino, Tia A, Hüttenhain, Ruth, Kaake, Robyn M, Richards, Alicia L, Tutuncuoglu, Beril, Foussard, Helene, Batra, Jyoti, Haas, Kelsey, Modak, Maya, Kim, Minkyu, Haas, Paige, Polacco, Benjamin J, Braberg, Hannes, Fabius, Jacqueline M, Eckhardt, Manon, Soucheray, Margaret, Bennett, Melanie J, Cakir, Merve, McGregor, Michael J, Li, Qiongyu, Naing, Zun Zar Chi, Zhou, Yuan, Peng, Shiming, Kirby, Ilsa T, Melnyk, James E, Chorba, John S, Lou, Kevin, Dai, Shizhong A, Shen, Wenqi, Shi, Ying, Zhang, Ziyang, Barrio-Hernandez, Inigo, Memon, Danish, Hernandez-Armenta, Claudia, Mathy, Christopher J P, Perica, Tina, Pilla, Kala B, Ganesan, Sai J, Saltzberg, Daniel J, Ramachandran, Rakesh, Liu, Xi, Rosenthal, Sara B, Calviello, Lorenzo, Venkataramanan, Srivats, Lin, Yizhu, Wankowicz, Stephanie A, Bohn, Markus, Trenker, Raphael, Young, Janet M, Cavero, Devin, Hiatt, Joe, Roth, Theo, Rathore, Ujjwal, Subramanian, Advait, Noack, Julia, Hubert, Mathieu, Roesch, Ferdinand, Vallet, Thomas, Meyer, Björn, White, Kris M, Miorin, Lisa, Agard, David, Emerman, Michael, Ruggero, Davide, García-Sastre, Adolfo, Jura, Natalia, von Zastrow, Mark, Taunton, Jack, Schwartz, Olivier, Vignuzzi, Marco, d'Enfert, Christophe, Mukherjee, Shaeri, Jacobson, Matt, Malik, Harmit S, Fujimori, Danica G, Ideker, Trey, Craik, Charles S, Floor, Stephen, Fraser, James S, Gross, John, Sali, Andrej, Kortemme, Tanja, Beltrao, Pedro, Shokat, Kevan, Shoichet, Brian K, Krogan, Nevan J
Published in bioRxiv (27.03.2020)
Published in bioRxiv (27.03.2020)
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