Anti-steatotic effects in conjunction with lowering of PNPLA3 mRNA exerted by LXR inverse agonists in human hepatocytes and in rodent models of non-alcoholic fatty liver disease
Kremoser, C, Hambruch, E, Gege, C, Deuschle, U, Kinzel, O, Krol, D.H, Albers, M, Birkel, M
Published in Journal of hepatology (2017)
Published in Journal of hepatology (2017)
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99 NOVEL FXR AGONISTS WITH POTENT LIPID LOWERING, INSULIN SENSITISING, ANTI-INFLAMMATORY AND ANTI-FIBROTISATION EFFECTS IN MOUSE MODELS OF METABOLIC SYNDROME AND NASH
Kremoser, C, Hambruch, E, Deuschle, U, Kinzel, O, Burnet, M, Yoneyama, H
Published in Journal of hepatology (01.03.2011)
Published in Journal of hepatology (01.03.2011)
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THU-495 - LXR inverse agonists inhibit de novo lipogenesis and reduce intestinal lipid and cholesterol absorption in a NAFLD mouse model
Kremoser, C., Deuschle, U., Gege, C., Kinzel, O., Krol, H.D., Albers, M., Birkel, M., Hambruch, E.
Published in Journal of hepatology (01.04.2018)
Published in Journal of hepatology (01.04.2018)
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THU-382 - Anti-steatotic effects in conjunction with lowering of PNPLA3 mRNA exerted by LXR inverse agonists in human hepatocytes and in rodent models of non-alcoholic fatty liver disease
Kremoser, C., Hambruch, E., Gege, C., Deuschle, U., Kinzel, O., Krol, D.H., Albers, M., Birkel, M.
Published in Journal of hepatology (2017)
Published in Journal of hepatology (2017)
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FRI-288 - From Mice to Men – Changes in FGF15/19 Expression and Bile Acid Levels as Sensitive Markers of Pharmacological FXR Activation; Results from Human Phase I and Animal Studies Using the Potent and Selective FXR Agonist Px-102
Hambruch, E., Krol, H., Perović-Ottstadt, S., Hornberger, M., Steeneck, C., Kinzel, O., Deuschle, U., Birkel, M., Kremoser, C.
Published in Journal of hepatology (2016)
Published in Journal of hepatology (2016)
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Journal Article
LXR inverse agonists inhibit de novo lipogenesis and reduce intestinal lipid and cholesterol absorption in a NAFLD mouse model
Kremoser, C., Deuschle, U., Gege, C., Kinzel, O., Krol, H.D., Albers, M., Birkel, M., Hambruch, E.
Published in Journal of hepatology (01.04.2018)
Published in Journal of hepatology (01.04.2018)
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A practical approach to the synthesis of hairpin polyamide-peptide conjugates through the use of a safety-catch linker
FATTORI, Daniela, KINZEL, Olaf, INGALLINELLA, Paolo, BIANCHI, Elisabetta, PESSI, Antonello
Published in Bioorganic & medicinal chemistry letters (22.04.2002)
Published in Bioorganic & medicinal chemistry letters (22.04.2002)
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Tetrazole thioacetanilides: Potent non-nucleoside inhibitors of WT HIV reverse transcriptase and its K103N mutant
Muraglia, Ester, Kinzel, Olaf D., Laufer, Ralph, Miller, Michael D., Moyer, Gregory, Munshi, Vandna, Orvieto, Federica, Palumbi, Maria Cecilia, Pescatore, Giovanna, Rowley, Michael, Williams, Peter D., Summa, Vincenzo
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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Synthesis of a functionalized high affinity mannose receptor ligand and its application in the construction of peptide-, polyamide- and PNA-conjugates
Kinzel, Olaf, Fattori, Daniela, Ingallinella, Paolo, Bianchi, Elisabetta, Pessi, Antonello
Published in Journal of peptide science (01.06.2003)
Published in Journal of peptide science (01.06.2003)
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A Functionally Orthogonal Estrogen Receptor-Based Transcription Switch Specifically Induced by a Nonsteroid Synthetic Ligand
Gallinari, Paola, Lahm, Armin, Koch, Uwe, Paolini, Chantal, Nardi, Maria Chiara, Roscilli, Giuseppe, Kinzel, Olaf, Fattori, Daniela, Muraglia, Ester, Toniatti, Carlo, Cortese, Riccardo, De Francesco, Raffaele, Ciliberto, Gennaro
Published in Chemistry & biology (01.08.2005)
Published in Chemistry & biology (01.08.2005)
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