Structure-activity relationships of pregabalin and analogues that target the alpha(2)-delta protein
Belliotti, TR, Capiris, T, Ekhato, Kinsora, JJ, Field, MJ, Heffner, TG, Meltzer, LT, Schwarz, JB, Taylor, CP, Thorpe, AJ, Vartanian, MG, Wise, LD, Zhi-Su, T, Weber, ML, Wustrow, DJ
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
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Activity profile of pregabalin in rodent models of epilepsy and ataxia
Vartanian, Mark G., Radulovic, Louis L., Kinsora, Jack J., Serpa, Kevin A., Vergnes, Marguerite, Bertram, Edward, Taylor, Charles P.
Published in Epilepsy research (01.03.2006)
Published in Epilepsy research (01.03.2006)
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Novel cyclopropyl beta-amino acid analogues of pregabalin and gabapentin that target the alpha(2)-delta protein
Schwarz, JB, Gibbons, SE, Graham, Colbry, NL, Guzzo, PR, Le, VD, Vartanian, MG, Kinsora, JJ, Lotarski, SM, Li, Z, Dickerson, MR, Su, TZ, Weber, ML, El-Kattan, A, Thorpe, AJ, Donevan, SD, Taylor, CP, Wustrow, DJ
Published in Journal of medicinal chemistry (21.04.2005)
Published in Journal of medicinal chemistry (21.04.2005)
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Carboxylate bioisosteres of gabapentin
Burgos-Lepley, Carmen E., Thompson, Lisa R., Kneen, Clare O., Osborne, Simon A., Bryans, Justin S., Capiris, Thomas, Suman-Chauhan, Nirmala, Dooley, David J., Donovan, Cindy M., Field, Mark J., Vartanian, Mark G., Kinsora, Jack J., Lotarski, Susan M., El-Kattan, Ayman, Walters, Karen, Cherukury, Madhu, Taylor, Charles P., Wustrow, David J., Schwarz, Jacob B.
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
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Carboxylate bioisosteres of pregabalin
Schwarz, Jacob B., Colbry, Norman L., Zhu, Zhijian, Nichelson, Brian, Barta, Nancy S., Lin, Kristin, Hudack, Raymond A., Gibbons, Sian E., Galatsis, Paul, DeOrazio, Russell J., Manning, David D., Vartanian, Mark G., Kinsora, Jack J., Lotarski, Susan M., Li, Zheng, Dickerson, Melvin R., El-Kattan, Ayman, Thorpe, Andrew J., Donevan, Sean D., Taylor, Charles P., Wustrow, David J.
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
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Milameline (CI-979/RU35926): A Muscarinic Receptor Agonist with Cognition-Activating Properties: Biochemical and In Vivo Characterization
Schwarz, R D, Callahan, M J, Coughenour, L L, Dickerson, M R, Kinsora, J J, Lipinski, W J, Raby, C A, Spencer, C J, Tecle, H
Published in The Journal of pharmacology and experimental therapeutics (01.11.1999)
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Published in The Journal of pharmacology and experimental therapeutics (01.11.1999)
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Continuous ICV infusion of scopolamine impairs sustained attention of rhesus monkeys
Callahan, M.J., Kinsora, J.J., Harbaugh, R.E., Reeder, T.M., Davis, R.E.
Published in Neurobiology of aging (01.03.1993)
Published in Neurobiology of aging (01.03.1993)
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