Design and Synthesis of Cyclopenta[g]quinazoline-Based Antifolates as Inhibitors of Thymidylate Synthase and Potential Antitumor Agents
Bavetsias, Vassilios, Marriott, Jonathan H, Melin, Camille, Kimbell, Rosemary, Matusiak, Zbigniew S, Boyle, F. Thomas, Jackman, Ann L
Published in Journal of medicinal chemistry (18.05.2000)
Published in Journal of medicinal chemistry (18.05.2000)
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Journal Article
Biological Activity and Intracellular Metabolism of ZD1694 in Human Leukemia Cell Lines with Different Resistance Mechanisms to Antifolate Drugs
Takemura, Yuzuru, Kobayashi, Hiroyuki, Miyachi, Hayato, Gibson, William, Kimbell, Rosemary, Jackman, Ann L.
Published in Cancer science (01.07.1996)
Published in Cancer science (01.07.1996)
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Journal Article
Cellular pharmacology and in vivo activity of a new anticancer agent, ZD9331: a water-soluble, nonpolyglutamatable, quinazoline-based inhibitor of thymidylate synthase
JACKMAN, A. L, KIMBELL, R, AHERNE, G. W, BRUNTON, L, JANSEN, G, STEPHENS, T. C, SMITH, M. N, WARDLEWORTH, J. M, BOYLE, F. T
Published in Clinical cancer research (01.06.1997)
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Published in Clinical cancer research (01.06.1997)
Journal Article
Does breakfast-club attendance affect schoolchildren's nutrient intake? A study of dietary intake at three schools
Belderson, Pippa, Harvey, Ian, Kimbell, Rosemary, O'Neill, Jennifer, Russell, Jean, Barker, Margo E.
Published in British journal of nutrition (01.12.2003)
Published in British journal of nutrition (01.12.2003)
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Journal Article
Design and Synthesis of Potent Non-Polyglutamatable Quinazoline Antifolate Thymidylate Synthase Inhibitors
Marsham, Peter R, Wardleworth, J. Michael, Boyle, F. Thomas, Hennequin, Laurent F, Kimbell, Rosemary, Brown, Melody, Jackman, Ann L
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
A rationale for the clinical development of the thymidylate synthase inhibitor ZD9331 in ovarian and other solid tumours
Jackman, Ann L, Melin, Camille J, Kimbell, Rosemary, Brunton, Lisa, Aherne, G.Wynne, Theti, Davinder S, Walton, Mike
Published in BBA - Molecular Basis of Disease (18.07.2002)
Published in BBA - Molecular Basis of Disease (18.07.2002)
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Synthesis of novel quinazoline-based antifolates with modified glutamate side chains as potential inhibitors of thymidylate synthase and antitumour agents
Bavetsias, Vassilios, Bisset, Graham M.F., Kimbell, Rosemary, Boyle, F.Thomas, Jackman, Ann L.
Published in Tetrahedron (29.09.1997)
Published in Tetrahedron (29.09.1997)
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Quinazoline Antifolate Thymidylate Synthase Inhibitors: γ-Linked l-d, d-d, and d-l Dipeptide Analogues of 2-Desamino-2-methyl-N 10-propargyl-5,8-dideazafolic Acid (ICI 198583)
Bavetsias, Vassilios, Jackman, Ann L, Kimbell, Rosemary, Gibson, William, Boyle, F. Thomas, Bisset, Graham M. F
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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Journal Article
Folate-Based Inhibitors of Thymidylate Synthase: Synthesis and Antitumor Activity of γ-Linked Sterically Hindered Dipeptide Analogues of 2-Desamino-2-methyl-N 10-propargyl-5,8-dideazafolic Acid (ICI 198583)
Bavetsias, Vassilios, Jackman, Ann L, Marriott, Jonathan H, Kimbell, Rosemary, Gibson, William, Boyle, F. Thomas, Bisset, Graham M. F
Published in Journal of medicinal chemistry (09.05.1997)
Published in Journal of medicinal chemistry (09.05.1997)
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Journal Article
The influence of drug‐exposure conditions on the development of resistance to methotrexate or ZD1694 in cultured human leukaemia cells
Takemura, Yuzuru, Kobayashi, Hiroyuki, Gibson, William, Kimbell, Rosemary, Miyachi, Hayato, Jackman, Ann L.
Published in International journal of cancer (28.03.1996)
Published in International journal of cancer (28.03.1996)
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Journal Article
Folate-Based Inhibitors of Thymidylate Synthase: Synthesis and Antitumor Activity of γ-Linked Sterically Hindered Dipeptide Analogues of 2-Desamino-2-methyl-N10-propargyl-5,8-dideazafolic Acid (ICI 198583)
BAVETSIAS, Vassilios, JACKMAN, Ann L., MARRIOTT, Jonathan H., KIMBELL, Rosemary, GIBSON, William, BOYLE, F. Thomas, BISSET, Graham M. F.
Published in Journal of medicinal chemistry (09.05.1997)
Published in Journal of medicinal chemistry (09.05.1997)
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Journal Article
Quinazoline Antifolates Thymidylate Synthase Inhibitors: Lipophilic Analogues with Modification to the C2-Methyl Substituent
Hennequin, Laurent F, Boyle, F. Thomas, Wardleworth, J. Michael, Marsham, Peter R, Kimbell, Rosemary, Jackman, Ann L
Published in Journal of medicinal chemistry (02.02.1996)
Published in Journal of medicinal chemistry (02.02.1996)
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Journal Article
Quinazoline Antifolate Thymidylate Synthase Inhibitors: Replacement of Glutamic Acid in the C2-Methyl Series
Marsham, Peter R, Jackman, Ann L, Barker, Andrew J, Boyle, F. Thomas, Pegg, Stephen J, Wardleworth, J. Michael, Kimbell, Rosemary, O'Connor, Brigid M, Calvert, A. Hilary, Hughes, Leslie R
Published in Journal of medicinal chemistry (01.03.1995)
Published in Journal of medicinal chemistry (01.03.1995)
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Journal Article
Carboxylic acid bioisosteres of γ-linked dipeptide analogues of the folate-based thymidylate synthase (TS) inhibitor, 2-desamino-2-methyl- N10-propargyl-5,8-dideazafolic acid (ICI 198583)
Bavetsias, Vassilios, Jackman, Ann L., Kimbell, Rosemary, Thomas Boyle, F., Bisset, Graham M.F.
Published in Bioorganic & medicinal chemistry letters (01.03.1996)
Published in Bioorganic & medicinal chemistry letters (01.03.1996)
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Journal Article
Quinazoline Antifolate Thymidylate Synthase Inhibitors: γ-Linked l-d, d-d, and d-l Dipeptide Analogues of 2-Desamino-2-methyl-N10-propargyl-5,8-dideazafolic Acid (ICI 198583)
BAVETSIAS, Vassilios, JACKMAN, Ann L., KIMBELL, Rosemary, GIBSON, William, BOYLE, F. Thomas, BISSET, Graham M. F.
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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Journal Article
The duration of the inhibition of thymidylate synthase in intact L1210 cells exposed to two different classes of quinazoline analogues
Kimbell, R, Jackman, A L, Boyle, F T, Hardcastle, A, Aherne, W
Published in Advances in experimental medicine and biology (1993)
Published in Advances in experimental medicine and biology (1993)
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