Discovery of potent, orally active benzimidazole glucagon receptor antagonists
Kim, Ronald M., Chang, Jiang, Lins, Ashley R., Brady, Ed, Candelore, Mari R., Dallas-Yang, Qing, Ding, Victor, Dragovic, Jasminka, Iliff, Susan, Jiang, Guoqiang, Mock, Steven, Qureshi, Sajjad, Saperstein, Richard, Szalkowski, Deborah, Tamvakopoulos, Constantin, Tota, Laurie, Wright, Michael, Yang, Xiaodong, Tata, James R., Chapman, Kevin, Zhang, Bei B., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Na v 1.7 target modulation and efficacy can be measured in nonhuman primate assays
Kraus, Richard L, Zhao, Fuqiang, Pall, Parul S, Zhou, Dan, Vardigan, Joshua D, Danziger, Andrew, Li, Yuxing, Daley, Christopher, Ballard, Jeanine E, Clements, Michelle K, Klein, Rebecca M, Holahan, Marie A, Greshock, Thomas J, Kim, Ronald M, Layton, Mark E, Burgey, Christopher S, Serra, Jordi, Henze, Darrell A, Houghton, Andrea K
Published in Science translational medicine (19.05.2021)
Published in Science translational medicine (19.05.2021)
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Journal Article
Discovery of 3-morpholino-imidazole[1,5-a]pyrazine BTK inhibitors for rheumatoid arthritis
Boga, Sobhana Babu, Alhassan, Abdul-Basit, Liu, Jian, Guiadeen, Deodial, Krikorian, Arto, Gao, Xiaolei, Wang, James, Yu, Younong, Anand, Rajan, Liu, Shilan, Yang, Chundao, Wu, Hao, Cai, Jiaqiang, Zhu, Hugh, Desai, Jagdish, Maloney, Kevin, Gao, Ying-Duo, Fischmann, Thierry O., Presland, Jeremy, Mansueto, My, Xu, Zangwei, Leccese, Erica, Knemeyer, Ian, Garlisi, Charles G., Bays, Nathan, Stivers, Peter, Brandish, Philip E., Hicks, Alexandra, Cooper, Alan, Kim, Ronald M., Kozlowski, Joseph A.
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
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Journal Article
Mimicry of Erythropoietin by a Nonpeptide Molecule
Qureshi, Sajjad A., Kim, Ronald M., Konteatis, Zenon, Biazzo, Dawn E., Motamedi, Haideh, Rodrigues, Robert, Boice, Judith A., Calaycay, Jimmy R., Bednarek, Maria A., Griffin, Patrick, Gao, Ying-Duo, Chapman, Kevin, Mark, David F.
Published in Proceedings of the National Academy of Sciences - PNAS (12.10.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (12.10.1999)
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Journal Article
인플루엔자를 치료 또는 예방하기 위한 폴리시클릭 캡-의존성 엔도뉴클레아제 억제제
SHURTLEFF VALERIE W, CHOBANIAN HARRY R, PLOTKIN MICHAEL A, SU HUA, EMBREY MARK W, KIM RONALD M, DEJESUS REYNALDA KEH, MORRIELLO GREGORI J, GUO LIANGQIN, MCCAULEY JOHN A, ZHANG YONGLIAN, FELLS JAMES, CROWLEY BRENDAN M, LO MICHAEL MAN CHU, ZHAO KAKE, DE LERA RUIZ MANUEL, BENNETT FRANK
Year of Publication 03.04.2023
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Year of Publication 03.04.2023
Patent
P1′ oxadiazole protease inhibitors with excellent activity against native and protease inhibitor-resistant HIV-1
Kim, Ronald M., Rouse, Elizabeth A., Chapman, Kevin T., Schleif, William A., Olsen, David B., Stahlhut, Mark, Rutkowski, Carrie A., Emini, Emilio A., Tata, James R.
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
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Journal Article
Dendrimer-Supported Combinatorial Chemistry
Kim, Ronald M., Manna, Mahua, Hutchins, Steven M., Griffin, Patrick R., Yates, Nathan A., Bernick, Amy M., Chapman, Kevin T.
Published in Proceedings of the National Academy of Sciences - PNAS (17.09.1996)
Published in Proceedings of the National Academy of Sciences - PNAS (17.09.1996)
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Journal Article
전압-게이팅 나트륨 채널에서 선택적 활성을 갖는 히드록시알킬아민- 및 히드록시시클로알킬아민-치환된 디아민-아릴술폰아미드 화합물
KIM RONALD M, ROECKER ANTHONY J, ZHOU GANG, WON WALTER, GUO LIANGQIN, GRESHOCK THOMAS J, MULHEARN JAMES, ZHANG TING, NANTERMET PHILIPPE, WANG DEPING, ANAND RAJAN, ZHENG JUNYING
Year of Publication 27.08.2018
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Year of Publication 27.08.2018
Patent
전압-게이팅 나트륨 채널에서 선택적 활성을 갖는 디아미노-알킬아미노-연결 아릴술폰아미드 화합물
ROECKER ANTHONY J, JIAN TIANYING, ZHOU GANG, WON WALTER, GRESHOCK THOMAS J, MULHEARN JAMES, ZHANG TING, ANAND RAJAN, KIM RONALD M, GUO LIANGQIN, KELLY MICHAEL J. III, WANG DEPING, NANTERMET PHILIPPE, LAYTON MARK E
Year of Publication 29.08.2018
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Year of Publication 29.08.2018
Patent
Antibacterial activity of G6-quaternary ammonium derivatives of a lipophilic vancomycin analogue
BLIZZARD, Timothy A, KIM, Ronald M, MORGAN, Jerry D, JIANG CHANG, KOHLER, Joyce, KILBURN, Ruth, CHAPMAN, Kevin, HAMMOND, Milton L
Published in Bioorganic & medicinal chemistry letters (25.03.2002)
Published in Bioorganic & medicinal chemistry letters (25.03.2002)
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Journal Article
SOLUBLE GUANYLATE CYCLASE ACTIVATORS
KIM RONALD M, ZIOUZINA OLGA A, PARMEE EMMA R, SINZ CHRISTOPHER JOSEPH
Year of Publication 09.12.2011
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Year of Publication 09.12.2011
Patent
Intercalation of aminophenyl- and pyridinium-substituted porphyrins into zirconium hydrogen phosphate: evidence for substituent-derived orientational selectivity
Kim, Ronald M, Pillion, John E, Burwell, David A, Groves, John T, Thompson, Mark E
Published in Inorganic chemistry (01.10.1993)
Published in Inorganic chemistry (01.10.1993)
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Journal Article
SOLUBLE GUANYLATE CYCLASE ACTIVATORS
KIM RONALD M, MIRC J. W, PARMEE EMMA R, TAN QIANG, BITTNER AMY R, CHANG JIANG, SINZ CHRISTOPHER JOSEPH
Year of Publication 04.06.2010
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Year of Publication 04.06.2010
Patent
BTK INHIBITORS
OUBRIE ARTHUR, ZHU HUGH Y, REWINKEL JOHANNES B.M, LIU SHILAN, YANG CHUNDAO, LIU JIAN, KAPTEIN ALLARD, BARF TJEERD A, JANS CHRISTIAAN G.J.M, ANAND RAJAN, WU HAO, STERRENBURG JAN GERARD, WIJKMANS JACOBUS C.H.M, WANG JAMES, YU YOUNONG, RAAIJMAKERS HANS C.A, KIM RONALD M, YAO XIN, COOPER ALAN B, VACCARO HENRY M, DE MAN ADRIANUS P.A, GAO XIAOLEI, ALHASSAN ABDUL BASIT, BOGA SOBHANA BABU
Year of Publication 05.06.2014
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Year of Publication 05.06.2014
Patent
Facile Synthesis of Trisubstituted Thioindoles via a Novel Tricyclic Thiolactone Intermediate
Yang, Cangming, Kim, Ronald M., Parmee, Emma R., Tan, Qiang
Published in Synthetic communications (10.03.2009)
Published in Synthetic communications (10.03.2009)
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Journal Article
Abstract 17305: Activation of Soluble Guanylate Cyclase Ameliorates the Progression of Glucose Intolerance and Nephropathy in Obese ZSF1 Rats
da Cunha, Valdeci, Shah, Kashmira, Price, Olga, Sinz, Christopher J, Kim, Ronald M
Published in Circulation (New York, N.Y.) (11.11.2016)
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Published in Circulation (New York, N.Y.) (11.11.2016)
Journal Article
Direct interaction of a vancomycin derivative with bacterial enzymes involved in cell wall biosynthesis
Sinha Roy, Ranabir, Yang, Ping, Kodali, Srinivas, Xiong, Yusheng, Kim, Ronald M, Griffin, Patrick R, Onishi, H.Russell, Kohler, Joyce, Silver, Lynn L, Chapman, Kevin
Published in Chemistry & biology (01.11.2001)
Published in Chemistry & biology (01.11.2001)
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